Journal
MOLECULAR DIVERSITY
Volume 19, Issue 3, Pages 473-480Publisher
SPRINGER
DOI: 10.1007/s11030-015-9583-5
Keywords
Indazolone; Hydrazines; Oxazolone; beta-Triketones
Categories
Funding
- MIUR [PRIN 20109Z2XRJ_010]
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A straightforward and efficient method for the synthesis of novel highly substituted and diversely functionalized indazolone derivatives has been developed. The transformation consists of a cyclocondensation of selected -tricarbonyls with monosubstituted hydrazines. The starting -triketones were prepared by an efficient chemo- and regioselective method under MW irradiation, exploiting the oxazolone chemistry. The reaction is easily accomplished under mild conditions and appears versatile, providing a synthetic diversification method with potential for drug-like compounds preparation.
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