Catalytic Enantioselective Ring-Opening Reaction ofmeso-Aziridines with α-Isothiocyanato Imides

Enantioselective Synthesis and Stereoselective Ring Opening ofN-Acylaziridines

(2012) Jennifer Cockrell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Synthesis of Spirooxindoles by a Mannich-Type Reaction of Isothiocyanato Oxindoles

(2012) Shota Kato et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Ion-Pairing Catalysis

(2012) Katrien Brak et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of structurally-diverse inhibitor scaffolds by high-throughput screening of a fragment library with dimethylarginine dimethylaminohydrolase

(2012) Thomas W. Linsky et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Highly Efficient Enantioselective Construction of Bispirooxindoles Containing Three Stereocenters through an Organocatalytic Cascade Michael-Cyclization Reaction

(2012) Hao Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric Michael Addition/Cyclization of Isothiocyanato Oxindoles: Highly Efficient and Versatile Approach for the Synthesis of 3,2′-Pyrrolidinyl Mono- and Bi-spirooxindole Frameworks

(2012) Yi-Ming Cao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Core Scaffold-Inspired Stereoselective Synthesis of Spiropyrazolones via an Organocatalytic Michael/Cyclization Sequence

(2012) Luping Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Cinchona Alkaloid Amides/Dialkylzinc Catalyzed Enantioselective Desymmetrization of Aziridines with Phosphites

(2012) Masashi Hayashi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Asymmetric Ring Openings of Meso and Terminal Aziridines with Halides Mediated by Chiral 1,2,3-Triazolium Silicates

(2012) Kohsuke Ohmatsu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Efficient and Stereoselective Construction of Dispiro-[oxazolidine-2-thione]bisoxindoles and Dispiro[imidazolidine-2-thione]bisoxindoles

(2012) Yan-Yan Han et al.   ORGANIC LETTERS

Studies on the true catalyst in the phosphate-promoted desymmetrization of meso-aziridines with silylated nucleophiles

(2012) Giorgio Della Sala   TETRAHEDRON

Stereodivergent Direct Catalytic Asymmetric Mannich-Type Reactions of α-Isothiocyanato Ester with Ketimines

(2011) Gang Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Michael/Cyclization Reaction Sequence: Scaffold-Inspired Synthesis of Spirooxindoles with Multiple Stereocenters

(2011) Yiming Cao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Guanidine-catalyzed enantioselective desymmetrization of meso-aziridines

(2011) Yan Zhang et al.   CHEMICAL COMMUNICATIONS

Core Structure-Based Design of Organocatalytic [3+2]-Cycloaddition Reactions: Highly Efficient and Stereocontrolled Syntheses of 3,3′-Pyrrolidonyl Spirooxindoles

(2011) Bin Tan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Guanidine Organocatalyst for the Asymmetric Mannich-Type Reaction between α-Isothiocyanato Imide and Sulfonyl Imines

(2011) Xiaohong Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric Ring-Opening ofmeso-Aziridines with Malonates under Heterodinuclear Rare Earth Metal Schiff Base Catalysis

(2011) Yingjie Xu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Direct Asymmetric Aldol Reactions of 3-Isothiocyanato Oxindoles to Ketones: Stereocontrolled Synthesis of Spirooxindoles Bearing Highly Congested Contiguous Tetrasubstituted Stereocenters

(2011) Wen-Bing Chen et al.   ORGANIC LETTERS

Catalytic enantioselective aldol additions of α-isothiocyanato imides to α-ketoesters

(2010) Matthew K. Vecchione et al.   CHEMICAL COMMUNICATIONS

Efficient Synthesis of β-Hydroxy-α-Amino Acid Derivatives via Direct Catalytic Asymmetric Aldol Reaction of α-Isothiocyanato Imide with Aldehydes

(2010) Xiaohong Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

A rationale for the activity profile of arylpiperazinylthioalkyls as 5-HT1A-serotonin and α1-adrenergic receptor ligands

(2010) Brij Kishore Sharma et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Unique Approach to the Concise Synthesis of Highly Optically Active Spirooxazolines and the Discovery of a More Potent Oxindole-Type Phytoalexin Analogue

(2010) Xianxing Jiang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct Organocatalytic Asymmetric Aldol Reaction of α-Isothiocyanato Imides to α-Ketoesters under Low Ligand Loading: A Doubly Stereocontrolled Approach to Cyclic Thiocarbamates Bearing Chiral Quaternary Stereocenters†

(2010) Xianxing Jiang et al.   ORGANIC LETTERS

Recent developments in regioselective ring opening of aziridines

(2010) Pengfei Lu   TETRAHEDRON

Enantioselective desymmetrization of meso-N-(heteroarenesulfonyl)aziridines with TMSN3 catalyzed by chiral Lewis acids

(2010) Shuichi Nakamura et al.   TETRAHEDRON LETTERS

Organocatalytic Asymmetric Synthesis of Protected α,β-Diamino Acids

(2009) Zugui Shi et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic, Enantioselective Ring Opening of Aziridines

(2009) Christoph Schneider   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Titanium Binolate Catalyzed Aminolysis ofmeso Aziridines: A Highly Enantioselective and Direct Access to 1,2-Diamines

(2009) Saravanan Peruncheralathan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and evaluation of a series of 2,4-diaminopyridine derivatives as potential positron emission tomography tracers for neuropeptide Y Y1 receptors

(2009) Minoru Kameda et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Cinchona-based phase-transfer catalysts for asymmetric synthesis

(2009) Sang-sup Jew et al.   CHEMICAL COMMUNICATIONS

Desymmetrization of meso-N-Acylaziridines with Benzenethiols Promoted by α,α-Diaryl-L-prolinols

(2009) Alessandra Lattanzi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Catalytic Enantioselective Synthesis of α,β-Diamino Acid Derivatives

(2009) Le Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Construction of Contiguous Tetrasubstituted Chiral Carbon Stereocenters via Direct Catalytic Asymmetric Aldol Reaction of α-Isothiocyanato Esters with Ketones

(2009) Tatsuhiko Yoshino et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chiral Phosphoric Acid-Catalyzed Desymmetrization ofmeso-Aziridines with Functionalized Mercaptans

(2009) Shawn E. Larson et al.   ORGANIC LETTERS

Highly Enantioselective Synthesis of β-Amidophenylthioethers by Organocatalytic Desymmetrization ofmeso-Aziridines

(2009) Giorgio Della Sala et al.   ORGANIC LETTERS

Enantioselective Desymmetrization ofmeso-Aziridines with TMSN3or TMSCN Catalyzed by Discrete Yttrium Complexes

(2008) Bin Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of New Arylpiperazinylalkylthiobenzimidazole, Benzothiazole, or Benzoxazole Derivatives as Potent and Selective 5-HT1ASerotonin Receptor Ligands†

(2008) Maria A. Siracusa et al.   JOURNAL OF MEDICINAL CHEMISTRY

Catalytic Enantioselective Aldol Additions of α-Isothiocyanato Imides to Aldehydes

(2008) Le Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantio- and Diastereoselective Catalytic Alkylation Reactions with Aziridines

(2008) Thomas A. Moss et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic asymmetric ring-opening of aziridines

(2008) Márcio W. Paixão et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Practical Aspects of Recent Asymmetric Phase-Transfer Catalysis

(2008) Keiji Maruoka   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Quinine-catalyzed enantioselective desymmetrization of meso-aziridines with benzenethiols

(2008) Zhiyong Wang et al.   TETRAHEDRON-ASYMMETRY