Copper Carbenoid, Reactant and Catalyst for One-Pot Diazo Ester Coupling Cascade Rearrangement of Enediynes: Formation of Two Contiguous Tetrasubstituted Stereocenters

One-pot Crabbé homologation-radical cascade cyclisation with memory of chirality

(2012) Shovan Mondal et al.   CHEMICAL COMMUNICATIONS

Mechanistic Investigation of Enediyne-Connected Amino Ester Rearrangement. Theoretical Rationale for the Exclusive Preference for 1,6- or 1,5-Hydrogen Atom Transfer Depending on the Substrate. A Potential Route to Chiral Naphthoazepines

(2012) Damien Campolo et al.   JOURNAL OF ORGANIC CHEMISTRY

An efficient and recyclable hybrid nanocatalyst to promote enantioselective radical cascade rearrangements of enediynes

(2011) Malek Nechab et al.   CHEMICAL COMMUNICATIONS

Design of Novel Neurokinin 1 Receptor Antagonists Based on Conformationally Constrained Aromatic Amino Acids and Discovery of a Potent Chimeric Opioid Agonist-Neurokinin 1 Receptor Antagonist

(2011) Steven Ballet et al.   JOURNAL OF MEDICINAL CHEMISTRY

Development of Tetrahydroisoquinoline-Based Hydroxamic Acid Derivatives: Potent Histone Deacetylase Inhibitors with Marked in Vitro and in Vivo Antitumor Activities

(2011) Yingjie Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Discovery of a Tetrahydroisoquinoline-Based Hydroxamic Acid Derivative (ZYJ-34c) as Histone Deacetylase Inhibitor with Potent Oral Antitumor Activities

(2011) Yingjie Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cu(i)-catalyzed tandem benzyldiazoester coupling with terminal alkyne–allene formation–Michael reaction: Application to the syntheses of oxa and azacycles

(2011) Gullapalli Kumaraswamy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalyzed Synthesis of 2,4-Disubstituted Allenoates from α-Diazoesters

(2011) Matthew Hassink et al.   ORGANIC LETTERS

Copper-catalyzed cascade coupling/cyclization of terminal alkynes with diazoacetates: a straightforward route for trisubstituted furans

(2011) Lei Zhou et al.   TETRAHEDRON LETTERS

Brønsted Base-Catalyzed Tandem Isomerization-Michael Reactions of Alkynes: Synthesis of Oxacycles and Azacycles

(2010) Hongjun Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Coupling of N-Tosylhydrazones with Terminal Alkynes Catalyzed by Copper(I): Synthesis of Trisubstituted Allenes

(2010) Qing Xiao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, synthesis and preliminary activity assay of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid derivatives as novel Histone deacetylases (HDACs) inhibitors

(2010) Yingjie Zhang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of enediyne-based peptide with selective peptide-cleaving activity

(2010) Snigdha Roy et al.   CHEMICAL COMMUNICATIONS

Bergman Cyclization of Acyclic Amino Acid Derived Enediynes Leads to the Formation of 2,3-Dihydrobenzo[f]isoindoles

(2010) Matija Gredičak et al.   JOURNAL OF ORGANIC CHEMISTRY

Memory of Chirality in Cascade Rearrangements of Enediynes

(2010) Malek Nechab et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Memory of Axial Chirality in Aryl Radical Phosphanylations

(2010) Achim Bruch et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chemistry of allenic/propargylic anions generated by base treatment of sulfonylallenes: synthesis of 1-alkynyl-1-sulfonylcycloalkanes and cycloalkanols

(2010) Shinji Kitagaki et al.   TETRAHEDRON

Design and synthesis of enediyne–peptide conjugates and their inhibiting activity against chymotrypsin

(2009) Sansa Dutta et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Catalytic Carbene Insertion into C−H Bonds

(2009) Michael P. Doyle et al.   CHEMICAL REVIEWS

Construction of Contiguous Tetrasubstituted Chiral Carbon Stereocenters via Direct Catalytic Asymmetric Aldol Reaction of α-Isothiocyanato Esters with Ketones

(2009) Tatsuhiko Yoshino et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

C-Lysine Conjugates: pH-Controlled Light-Activated Reagents for Efficient Double-Stranded DNA Cleavage with Implications for Cancer Therapy

(2009) Wang-Yong Yang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Stereoselective Synthesis of the Epicoccin Core

(2009) Ulrike Gross et al.   ORGANIC LETTERS

Synthesis and DNA-cleaving activity of lactenediynes conjugated with DNA-complexing moieties

(2008) Luca Banfi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Asymmetric synthesis of β-lactams using chiral-memory effect on photochemical γ-hydrogen abstraction by thiocarbonyl group

(2008) Masami Sakamoto et al.   CHEMICAL COMMUNICATIONS

Design, synthesis and DNA-cleaving efficiency of photoswitchable dimeric azobenzene-based C2-symmetric enediynes

(2008) Amit Basak et al.   CHEMICAL COMMUNICATIONS

Synthesis and aromatisation of cyclic enediyne-containing amino acids

(2008) Jasper Kaiser et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Ruthenium-Catalyzed One-Pot Carbenoid N−H Insertion Reactions and Diastereoselective Synthesis of Prolines

(2008) Qing-Hai Deng et al.   ORGANIC LETTERS