Persulfate-promoted oxidative C–N bond coupling of quinoxalinones and NH-sulfoximines

Sulfoximines from a Medicinal Chemist's Perspective: Physicochemical and in vitro Parameters Relevant for Drug Discovery

(2017) Marcus Frings et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Hydroxymethylation of Quinolines with Na2 S2 O8 by a Radical Pathway

(2017) Luan Zhou et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Transition-metal-free and organic solvent-free conversion of N-substituted 2-aminobiaryls into corresponding carbazoles via intramolecular oxidative radical cyclization induced by peroxodisulfate

(2017) Palani Natarajan et al.   GREEN CHEMISTRY

Iodine-Catalyzed C–N Bond Formation: Synthesis of 3-Aminoquinoxalinones under Ambient Conditions

(2017) Abhishek Gupta et al.   JOURNAL OF ORGANIC CHEMISTRY

(Diacetoxy)iodobenzene-Mediated Oxidative C–H Amination of Imidazopyridines at Ambient Temperature

(2017) Susmita Mondal et al.   JOURNAL OF ORGANIC CHEMISTRY

“A Jack of Trio”-robust one-pot metal free oxidative amination, azidation and peroxidation of phenols

(2017) Debayan Sarkar et al.   NEW JOURNAL OF CHEMISTRY

Copper-catalyzed oxidative decarboxylative coupling of α-keto acids and sulfoximines

(2017) Chaleena Pimpasri et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper promoted N-alkylation of sulfoximines with alkylboronic acid under mild conditions

(2017) Surabhi Gupta et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Silver-catalyzed decarboxylative acylation of quinoxalin-2(1H)-ones with α-oxo-carboxylic acids

(2017) Xiaobao Zeng et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition-Metal-Free Direct C–H Arylation of Quinoxalin-2(1H)-ones with Diaryliodonium Salts at Room Temperature

(2017) Kun Yin et al.   ORGANIC LETTERS

Transfer of Electrophilic NH Using Convenient Sources of Ammonia: Direct Synthesis of NH Sulfoximines from Sulfoxides

(2016) Marina Zenzola et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct phosphonation of quinoxalin-2(1H)-ones under transition-metal-free conditions

(2016) Ming Gao et al.   CHEMICAL COMMUNICATIONS

Non-Deprotonative Primary and Secondary Amination of (Hetero)Arylmetals

(2016) Zhe Zhou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-catalysed oxidative amination of quinoxalin-2(1H)-ones with aliphatic amines

(2016) Yi Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Direct and Practical Synthesis of Primary Anilines through Iron-Catalyzed C–H Bond Amination

(2016) Luca Legnani et al.   ACS Catalysis

Pyrazino[2,3-g]quinoxaline-2,7-dione based π-conjugated polymers with affinity towards acids and semiconductor performance in organic thin film transistors

(2016) Jesse Quinn et al.   RSC Advances

tert-Butyl Hydroperoxide and Tetrabutylammonium Iodide-Promoted Free Radical Cyclization of α-Imino-N-arylamides and α-Azido-N-arylamides

(2015) Dianjun Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-catalyzed aerobic radical C–C bond cleavage of N–H ketimines

(2015) Ya Lin Tnay et al.   Beilstein Journal of Organic Chemistry

Palladium/Copper-Cocatalyzed Oxidative Amidobrominations of Alkenes

(2015) Xiao Yun Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Designing novel building blocks is an overlooked strategy to improve compound quality

(2015) Frederick W. Goldberg et al.   DRUG DISCOVERY TODAY

Drugging ATR: progress in the development of specific inhibitors for the treatment of cancer

(2015) Kevin M Foote et al.   Future Medicinal Chemistry

Catalyst-Free Regioselective C-3 Thiocyanation of Imidazopyridines

(2015) Daoshan Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Microwave-Promoted Tin-Free Iminyl Radical Cyclization with TEMPO Trapping: A Practical Synthesis of 2-Acylpyrroles

(2015) Yu Cai et al.   ORGANIC LETTERS

Development of a Scalable Process for the Crop Protection Agent Isoclast

(2015) Kim E. Arndt et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Catalytic Methods for Aromatic C–H Amination: An Ideal Strategy for Nitrogen-Based Functional Molecules

(2015) Jiao Jiao et al.   ACS Catalysis

Fluorinated sulfoximines: syntheses, properties and applications

(2014) Vincent Bizet et al.   CHEMICAL SOCIETY REVIEWS

Structure–activity relationships studies of quinoxalinone derivatives as aldose reductase inhibitors

(2014) Saghir Hussain et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Fluorinated Sulfoximines: Preparation, Reactions and Applications

(2014) Xiao Shen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Advances in the Chemistry of Quinoxalinone Derivatives

(2014) Leilei Shi et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Iron-Catalyzed Hetero-Cross-Dehydrogenative Coupling Reactions of Sulfoximines with Diarylmethanes: A New Route to N-Alkylated Sulfoximines

(2014) Ying Cheng et al.   ORGANIC LETTERS

The Copper-Catalyzed OxidativeN-Acylation of Sulfoximines

(2013) Long Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Sulfoximines: A Neglected Opportunity in Medicinal Chemistry

(2013) Ulrich Lücking   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Oxidative Cross-Coupling of Sulfoximines and Alkynes

(2013) Long Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Lab Oddity Prevails: Discovery of Pan-CDK Inhibitor (R)-S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-hydroxy-1-methylpropyl]oxy}-5-(trifluoromethyl)pyrimidin-2-yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer

(2013) Ulrich Lücking et al.   ChemMedChem

Metal-Free Oxidative Carbon-Heteroatom Bond Formation Through C-H Bond Functionalization

(2013) Rajarshi Samanta et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Sulfoxaflor and the sulfoximine insecticides: Chemistry, mode of action and basis for efficacy on resistant insects

(2013) Thomas C. Sparks et al.   PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY

Syntheses and biological activities of sulfoximine-based acyclic triaryl olefins

(2012) Xiao Yun Chen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

N-Cyano Sulfoximines: COX Inhibition, Anticancer Activity, Cellular Toxicity, and Mutagenicity

(2012) Seong Jun Park et al.   ChemMedChem

An Efficient Synthesis of Quinoxalinone Derivatives as Potent Inhibitors of Aldose Reductase

(2012) Yanchun Yang et al.   ChemMedChem

Comparison of symmetric and asymmetric bipolar type high triplet energy host materials for deep blue phosphorescent organic light-emitting diodes

(2012) Soon Ok Jeon et al.   JOURNAL OF MATERIALS CHEMISTRY

Bioactive sulfoximines: Syntheses and properties of Vioxx® analogs

(2011) Seong Jun Park et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, In Vitro Antitubercular Activity and 3D-QSAR of Novel Quinoxaline Derivatives

(2011) Ayarivan Puratchikody et al.   Chemical Biology & Drug Design

UV promoted phenanthridine syntheses from oxime carbonate derived iminyl radicals

(2011) Roy T. McBurney et al.   CHEMICAL COMMUNICATIONS

Recent advances in the transition metal-catalyzed twofold oxidative C–H bond activation strategy for C–C and C–N bond formation

(2011) Seung Hwan Cho et al.   CHEMICAL SOCIETY REVIEWS

Metal-Free Intermolecular Oxidative C–N Bond Formation via Tandem C–H and N–H Bond Functionalization

(2011) Abhishek A. Kantak et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Metal-Free Amination of Benzoxazoles – The First Example of an Iodide-Catalyzed Oxidative Amination of Heteroarenes

(2011) Tanja Froehr et al.   ORGANIC LETTERS

Quinoxalinoneinhibitors of the lectin DC-SIGN

(2011) Shane L. Mangold et al.   Chemical Science

An Efficient Domino Synthesis of Quinoxalin-2(1H)-ones via an SNAr/Coupling/Demesylation Reaction Catalyzed by Copper(I) as Key Step

(2010) Dingben Chen et al.   ADVANCED SYNTHESIS & CATALYSIS

Direct Azole Amination: CH Functionalization as a New Approach to Biologically Important Heterocycles

(2010) Alan Armstrong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective synthesis of highly functionalised amides by copper-catalysed vinylogous Mukaiyama aldol reaction

(2010) Marcus Frings et al.   CHEMICAL COMMUNICATIONS

Synthesis of some new pyrimido[2′,1′:2,3]thiazolo[4,5-b]quinoxaline derivatives as anti-inflammatory and analgesic agents

(2010) A.A. Abu-Hashem et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Part I: Synthesis, cancer chemopreventive activity and molecular docking study of novel quinoxaline derivatives

(2010) Shadia A. Galal et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Discovery and Characterization of Sulfoxaflor, a Novel Insecticide Targeting Sap-Feeding Pests

(2010) Yuanming Zhu et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Iron(II) Triflate as an Efficient Catalyst for the Imination of Sulfoxides

(2009) Olga García Mancheño et al.   ORGANIC LETTERS

In vitro and in vivo anti-tumoral activities of imidazo[1,2-a]quinoxaline, imidazo[1,5-a]quinoxaline, and pyrazolo[1,5-a]quinoxaline derivatives

(2008) Georges Moarbess et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Oxidative alkylamination of azinones as a direct route to aminoazinones: study of some condensed diazinones

(2007) Anna V. Gulevskaya et al.   TETRAHEDRON