Cobalt(ii)-catalyzed remote C5-selective C–H sulfonylation of quinolines via insertion of sulfur dioxide

A copper-catalyzed sulfonylative C–H bond functionalization from sulfur dioxide and aryldiazonium tetrafluoroborates

(2018) Hongguang Xia et al.   Organic Chemistry Frontiers

Synthesis of sulfonated naphthols via C–H bond functionalization with the insertion of sulfur dioxide

(2018) Kaida Zhou et al.   Organic Chemistry Frontiers

Pd-Catalyzed Conversion of Aryl Iodides to Sulfonyl Fluorides Using SO2 Surrogate DABSO and Selectfluor

(2017) Ariana L. Tribby et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective remote esterification of 8-aminoquinoline amides via copper(ii)-catalyzed C(sp2)–O cross-coupling reaction

(2017) Chengcai Xia et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of sulfones via selective C–H-functionalization

(2017) Saad Shaaban et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Pd-Catalyzed Selective Synthesis of Cyclic Sulfonamides and Sulfinamides Using K2S2O5 as a Sulfur Dioxide Surrogate

(2017) Hideyuki Konishi et al.   ORGANIC LETTERS

N-Radical Initiated Aminosulfonylation of Unactivated C(sp3)–H Bond through Insertion of Sulfur Dioxide

(2017) Yuewen Li et al.   ORGANIC LETTERS

Copper(i)-catalyzed sulfonylative Suzuki–Miyaura cross-coupling

(2017) Yiding Chen et al.   Chemical Science

Domino C–H/N–H Allylations of Imidates by Cobalt Catalysis

(2017) Hui Wang et al.   ACS Catalysis

Copper(i) and N-fluorobenzenesulfonimide-mediated direct regioselective halogenation of 8-amidoquinolines on the C5 position

(2017) Xin He et al.   Organic Chemistry Frontiers

Nickel-catalyzed selective C-5 fluorination of 8-aminoquinolines with NFSI

(2017) Junshuai Ding et al.   Organic Chemistry Frontiers

Site-selective oxidative C–H sulfonylation of 8-acylaminoquinolines and anilides under metal-free conditions

(2017) Yang Wang et al.   Organic Chemistry Frontiers

Synthesis of 3-(((2,3-dihydrobenzofuran-3-yl)methyl)sulfonyl) coumarins through the reaction of 2-(allyloxy)anilines, sulfur dioxide, and aryl propiolates

(2017) Xuefeng Wang et al.   Organic Chemistry Frontiers

Radical cyclization of benzene-tethered 1,7-enynes with aryldiazonium tetrafluoroborates: a facile route to benzo[j]phenanthridines

(2017) Yuanyuan An et al.   Organic Chemistry Frontiers

Synthesis of 3-((arylsulfonyl)methyl)indolin-2-ones via insertion of sulfur dioxide using anilines as the aryl source

(2017) Tong Liu et al.   Organic Chemistry Frontiers

Generation of benzosultams via a radical process with the insertion of sulfur dioxide

(2017) Kaida Zhou et al.   Organic Chemistry Frontiers

Reductive insertion of sulfur dioxide for the synthesis of trifluoromethyl thiolsulphonates through a one-pot reaction of aniline and trifluoromethanesulfanylamide

(2017) Jie Sheng et al.   Organic Chemistry Frontiers

Transition-metal-free oxidative reaction of hydrazines and potassium metabisulfite for preparation of sulfonohydrazides

(2017) Yang Wang et al.   Organic Chemistry Frontiers

Synthesis of β-keto sulfones via a multicomponent reaction through sulfonylation and decarboxylation

(2017) Jiyao Yu et al.   Organic Chemistry Frontiers

Copper-Catalyzed Remote C-H Sulfonylation of 8-Aminoquinoline Amides with Arylsulfonyl Hydrazides

(2017) Guoshu Chen et al.   ChemistrySelect

Copper-Catalyzed Remote C−H Functionalization of 8-Aminoquinolines with Sodium and Lithium Sulfinates

(2016) Shuai Liang et al.   ADVANCED SYNTHESIS & CATALYSIS

A First Example of Cobalt-Catalyzed Remote CH Functionalization of 8-Aminoquinolines Operating through a Single Electron Transfer Mechanism

(2016) Christopher J. Whiteoak et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-Catalyzed Remote C−H Amination of Quinolines withN-Fluorobenzenesulfonimide

(2016) Yao Yin et al.   ADVANCED SYNTHESIS & CATALYSIS

Generation of Sulfonyl Radicals from Aryldiazonium Tetrafluoroborates and Sulfur Dioxide: The Synthesis of 3-Sulfonated Coumarins

(2016) Danqing Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-catalyzed synthesis of arylsulfinates through radical coupling reaction

(2016) Weixi Zhang et al.   CHEMICAL COMMUNICATIONS

Transition-Metal-Catalyzed C–H Bond Addition to Carbonyls, Imines, and Related Polarized π Bonds

(2016) Joshua R. Hummel et al.   CHEMICAL REVIEWS

Transition metal-catalysed couplings between arenes and strained or reactive rings: combination of C–H activation and ring scission

(2016) Fen Wang et al.   CHEMICAL SOCIETY REVIEWS

Vicinal Difluoroalkylation and Aminosulfonylation of Alkynes under Photoinduced Conditions

(2016) Yuanchao Xiang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Remote C−H Activation of Quinolines through Copper-Catalyzed Radical Cross-Coupling

(2016) Jun Xu et al.   Chemistry-An Asian Journal

In Situ Generated HypoIodite Activator for the C2 Sulfonylation of Heteroaromatic N-oxides

(2016) Yuan Su et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Regioselective C–H Sulfonylation of 8-Aminoquinolines

(2016) Jun Wei et al.   JOURNAL OF ORGANIC CHEMISTRY

Transition-metal-free oxidative C5 C–H-halogenation of 8-aminoquinoline amides using sodium halides

(2016) Ying Wang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper(ii)-catalyzed C5 and C7 halogenation of quinolines using sodium halides under mild conditions

(2016) Jun Xu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Metal-Free Remote C–H Bond Amidation of 8-Amidoquinolines on the C5 Position under Mild Conditions

(2016) Dezhong Ji et al.   ORGANIC LETTERS

Cu-Catalyzed Deoxygenative C2-Sulfonylation Reaction of Quinoline N-Oxides with Sodium Sulfinate

(2016) Bingnan Du et al.   ORGANIC LETTERS

Amidines for Versatile Cobalt(III)-Catalyzed Synthesis of Isoquinolines through C–H Functionalization with Diazo Compounds

(2016) Jie Li et al.   ORGANIC LETTERS

Reaction of Alkyl Halides with Rongalite: One-Pot and Telescoped Syntheses of Aliphatic Sulfonamides, Sulfonyl Fluorides, and Unsymmetrical Sulfones

(2016) Andre Shavnya et al.   ORGANIC LETTERS

Nickel-Catalyzed Site-Selective C–H Bond Difluoroalkylation of 8-Aminoquinolines on the C5-Position

(2016) Hao Chen et al.   ORGANIC LETTERS

Regio- and Chemoselective Mono- and Bisnitration of 8-Amino quinoline Amides with Fe(NO3)3·9H2O as Promoter and Nitro Source

(2016) Yan He et al.   ORGANIC LETTERS

Copper-catalyzed C5-regioselective C H sulfonylation of 8-aminoquinoline amides with aryl sulfonyl chlorides

(2016) Jun-Ming Li et al.   TETRAHEDRON LETTERS

Copper(ii)-catalyzed remote sulfonylation of aminoquinolines with sodium sulfinates via radical coupling

(2016) Chengcai Xia et al.   RSC Advances

Oxidative Remote C−H Trifluoromethylation of Quinolineamides on the C5 Position with Iodobenzene Diacetate as the Oxidizing Agent

(2016) Zhaoyang Wu et al.   Asian Journal of Organic Chemistry

A general route to sulfones via insertion of sulfur dioxide promoted by cobalt oxide

(2016) Danqing Zheng et al.   Organic Chemistry Frontiers

Copper-catalyzed 8-amido chelation-induced regioselective C–H fluoroalkylation of quinolines

(2016) Li-Kun Jin et al.   Organic Chemistry Frontiers

A copper(ii)-catalyzed three-component reaction of aryldiazonium tetrafluoroborates, sulfur dioxide, with alkenes

(2016) Runyu Mao et al.   Organic Chemistry Frontiers

Palladium(II)-Catalyzed Synthesis of Sulfinates from Boronic Acids and DABSO: A Redox-Neutral, Phosphine-Free Transformation

(2015) Alex S. Deeming et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Synthesis of (Hetero)Aryl Alkyl Sulfones from (Hetero)Aryl Boronic Acids, Unactivated Alkyl Halides, and Potassium Metabisulfite

(2015) Andre Shavnya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selective remote C–H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis

(2015) Hong-Wen Liang et al.   CHEMICAL COMMUNICATIONS

H-phosphonate-mediated sulfonylation of heteroaromatic N-oxides: a mild and metal-free one-pot synthesis of 2-sulfonyl quinolines/pyridines

(2015) Kai Sun et al.   CHEMICAL COMMUNICATIONS

Recent advances in C–S bond formation via C–H bond functionalization and decarboxylation

(2015) Chao Shen et al.   CHEMICAL SOCIETY REVIEWS

Transition metal-catalyzed ketone-directed or mediated C–H functionalization

(2015) Zhongxing Huang et al.   CHEMICAL SOCIETY REVIEWS

Recent advances in transition metal-catalyzed C–H bond functionalization of ferrocene derivatives

(2015) Luis A. López et al.   DALTON TRANSACTIONS

Nickel-Catalyzed Alkynylation of a C(sp2)–H Bond Directed by an 8-Aminoquinoline Moiety

(2015) Jun Yi et al.   JOURNAL OF ORGANIC CHEMISTRY

Fixation of sulfur dioxide into small molecules

(2015) Gang Liu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Regioselective, Molecular Iodine-Mediated C3 Iodination of Quinolines

(2015) Kai Sun et al.   ORGANIC LETTERS

Copper-Mediated Remote C–H Bond Chalcogenation of Quinolines on the C5 Position

(2015) Longzhi Zhu et al.   ORGANIC LETTERS

One-Pot, Three-Component Arylalkynyl Sulfone Synthesis

(2015) C. Chun Chen et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Sulfonylation of 8-Aminoquinoline Amides with Sulfonyl Chlorides in Air

(2015) Huijie Qiao et al.   ORGANIC LETTERS

Pd(II)-Catalyzed Direct Sulfonylation of Unactivated C(sp3)–H Bonds with Sodium Sulfinates

(2015) Wei-Hao Rao et al.   ORGANIC LETTERS

Cobalt-Catalyzed C–H Activation

(2015) Marc Moselage et al.   ACS Catalysis

Transition metal-catalyzed C–H bond functionalizations by the use of diverse directing groups

(2015) Zhengkai Chen et al.   Organic Chemistry Frontiers

Metal-Free Aminosulfonylation of Aryldiazonium Tetrafluoroborates with DABCO⋅(SO2)2and Hydrazines

(2014) Danqing Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Synthesis of Ammonium Sulfinates from Aryl Halides and a Sulfur Dioxide Surrogate: A Gas- and Reductant-Free Process

(2014) Edward J. Emmett et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Application of Fundamental Organometallic Chemistry to the Development of a Gold-Catalyzed Synthesis of Sulfinate Derivatives

(2014) Miles W. Johnson et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Combining Organometallic Reagents, the Sulfur Dioxide Surrogate DABSO, and Amines: A One-Pot Preparation of Sulfonamides, Amenable to Array Synthesis

(2014) Alex S. Deeming et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium(III)-Catalyzed CC and CO Coupling of QuinolineN-Oxides with Alkynes: Combination of CH Activation with O-Atom Transfer

(2014) Xueyun Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-catalyzed aerobic difunctionalization of alkenes: a highly efficient approach to construct oxindoles by C–S and C–C bond formation

(2014) Tao Shen et al.   CHEMICAL COMMUNICATIONS

Direct regioselective phosphonation of heteroaryl N-oxides with H-phosphonates under metal and external oxidant free conditions

(2014) Hui Wang et al.   CHEMICAL COMMUNICATIONS

Syntheses, Radiolabelings, and in Vitro Evaluations of Fluorinated PET Radioligands of 5-HT6 Serotoninergic Receptors

(2014) Julie Colomb et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cobalt-Catalyzed C–H Arylations, Benzylations, and Alkylations with Organic Electrophiles and Beyond

(2014) Lutz Ackermann   JOURNAL OF ORGANIC CHEMISTRY

Regioselective Introduction of Heteroatoms at the C-8 Position of Quinoline N-Oxides: Remote C–H Activation Using N-Oxide as a Stepping Stone

(2014) Heejun Hwang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(III)-Catalyzed C–C Bond Formation of Quinoline N-Oxides at the C-8 Position under Mild Conditions

(2014) Jisu Jeong et al.   ORGANIC LETTERS

Iron-Catalyzed, Chelation-Induced Remote C–H Allylation of Quinolines via 8-Amido Assistance

(2014) Xuefeng Cong et al.   ORGANIC LETTERS

A Copper-Catalyzed Three-Component Reaction of Triethoxysilanes, Sulfur Dioxide, and Hydrazines

(2014) Xianbo Wang et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Amination of Quinoline N-Oxides via C–H Bond Activation under Mild Conditions

(2014) Chongwei Zhu et al.   ORGANIC LETTERS

Rediscovering the Chemistry of Sulfur Dioxide: New Developments in Synthesis and Catalysis

(2014) Michael Willis et al.   SYNTHESIS-STUTTGART

Recent advances in directed C–H functionalizations using monodentate nitrogen-based directing groups

(2014) Min Zhang et al.   Organic Chemistry Frontiers

Palladium-Catalyzed Three-Component Diaryl Sulfone Synthesis Exploiting the Sulfur Dioxide Surrogate DABSO

(2013) Edward J. Emmett et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Aerobic Oxysulfonylation of Alkenes Leading to Secondary and Tertiary β-Hydroxysulfones

(2013) Qingquan Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A tandem Friedel–Crafts based method for the construction of a tricyclic pyrroloquinoline skeleton and its application in the synthesis of ammosamide B

(2013) Yohei Takayama et al.   CHEMICAL COMMUNICATIONS

The antitumor activity of zinc(II) and copper(II) complexes with 5,7-dihalo-substituted-8-quinolinoline

(2013) Yan-Cheng Liu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Dioxygen-Triggered Oxidative Radical Reaction: Direct Aerobic Difunctionalization of Terminal Alkynes toward β-Keto Sulfones

(2013) Qingquan Lu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Taming sulfur dioxide: a breakthrough for its wide utilization in chemistry and biology

(2013) Philippe Bisseret et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalyzed Intermolecular Dehydrogenative Amidation/Amination of Quinoline N-Oxides with Lactams/Cyclamines

(2013) Gang Li et al.   ORGANIC LETTERS

Palladium-Catalyzed Sulfination of Aryl and Heteroaryl Halides: Direct Access to Sulfones and Sulfonamides

(2013) Andrei Shavnya et al.   ORGANIC LETTERS

Synthesis of Sulfones from Organozinc Reagents, DABSO, and Alkyl Halides

(2013) Benjamin N. Rocke et al.   ORGANIC LETTERS

1,4-Diazabicyclo[2.2.2]octane Bis(sulfur dioxide) Adduct (DABSO)

(2013) Ludovic Martial   SYNLETT

On the Interpretation of Deuterium Kinetic Isotope Effects in CH Bond Functionalizations by Transition-Metal Complexes

(2012) Eric M. Simmons et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A palladium-catalyzed reaction of aryl halides, potassium metabisulfite, and hydrazines

(2012) Shengqing Ye et al.   CHEMICAL COMMUNICATIONS

Palladium-catalysed aminosulfonylation of aryl-, alkenyl- and heteroaryl halides: scope of the three-component synthesis of N-aminosulfonamides

(2012) Edward J. Emmett et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Nitroxoline (8-hydroxy-5-nitroquinoline) is more a potent anti-cancer agent than clioquinol (5-chloro-7-iodo-8-quinoline)

(2011) Hongchao Jiang et al.   CANCER LETTERS

Kinetic Isotope Effects in the Study of Organometallic Reaction Mechanisms

(2011) Mar Gómez-Gallego et al.   CHEMICAL REVIEWS

5-HT6 receptor and cognition

(2011) Xabier Codony et al.   CURRENT OPINION IN PHARMACOLOGY

Ruthenium-Catalyzed Meta Sulfonation of 2-Phenylpyridines

(2011) Ourida Saidi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Quinolines and structurally related heterocycles as antimalarials

(2010) Kirandeep Kaur et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Imide-Catalyzed Oxidation System: Sulfides to Sulfoxides and Sulfones

(2010) Naohiro Fukuda et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis of the Ammosamides

(2010) Chambers C. Hughes et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Aminosulfonylation of Aryl Halides

(2010) Bao Nguyen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Direct Arylation of Azine and AzoleN-Oxides: Reaction Development, Scope and Applications in Synthesis

(2009) Louis-Charles Campeau et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed C−H Bond Functionalization with Arylsulfonyl Chlorides

(2009) Xiaodan Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Ammosamides: Structures of Cell Cycle Modulators from a Marine-DerivedStreptomycesSpecies

(2008) Chambers C. Hughes et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS