Selective S-arylation of 2-oxazolidinethiones and selective N-arylation of 2-benzoxazolinones/2-benzimidazolinones

Employing Arynes in Diels–Alder Reactions and Transition-Metal-Free Multicomponent Coupling and Arylation Reactions

(2016) Sachin Suresh Bhojgude et al.   ACCOUNTS OF CHEMICAL RESEARCH

Superacid-Catalyzed Trifluoromethylthiolation of Aromatic Amines

(2016) Longin Justin Clair Bonazaba Milandou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-free C–H thioarylation of arenes using sulfoxides: a direct, general diaryl sulfide synthesis

(2016) José A. Fernández-Salas et al.   CHEMICAL COMMUNICATIONS

Chemoselective cross-coupling reaction of sodium sulfinates with phenols under aqueous conditions

(2016) Fuhong Xiao et al.   GREEN CHEMISTRY

Catalytic Synthesis of 3-Thioindoles Using Bunte Salts as Sulfur Sources under Metal-Free Conditions

(2016) Hong Qi et al.   JOURNAL OF ORGANIC CHEMISTRY

Reactions of HDDA-Derived Benzynes with Sulfides: Mechanism, Modes, and Three-Component Reactions

(2016) Junhua Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Aryne 1,2,3-Trifunctionalization with Aryl Allyl Sulfoxides

(2016) Yuanyuan Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Reactions of Hexadehydro-Diels–Alder (HDDA)-Derived Benzynes with Thioamides: Synthesis of Dihydrobenzothiazino-Heterocyclics

(2016) Vignesh Palani et al.   ORGANIC LETTERS

Synthesis of Aryl Ketoamides via Aryne Insertion into Imides

(2016) Austin C. Wright et al.   ORGANIC LETTERS

TFA-promoted direct C–H sulfenylation at the C2 position of non-protected indoles

(2015) Thomas Hostier et al.   CHEMICAL COMMUNICATIONS

Domino Aryne Precursor: Efficient Construction of 2,4-Disubstituted Benzothiazoles

(2015) Jiarong Shi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

CuI/Oxalic Diamide Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amines

(2015) Wei Zhou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Reaction of Arynes with Sulfoxides

(2015) Hong-Ying Li et al.   ORGANIC LETTERS

Synthesis of Aryl Sulfides: Metal-Free C–H Sulfenylation of Electron-Rich Arenes

(2015) Thomas Hostier et al.   ORGANIC LETTERS

Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sodium Sulfinates

(2014) Fuhong Xiao et al.   ADVANCED SYNTHESIS & CATALYSIS

Regioselective Thiolation of Arenes and Heteroarenes: C–H Functionalization Strategy for C–S Bond Formation

(2014) Begur Vasanthkumar Varun et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine-Mediated Thiolation of Substituted Naphthols/Naphthylamines and Arylsulfonyl Hydrazides via C(sp2)–H Bond Functionalization

(2014) Xing Kang et al.   JOURNAL OF ORGANIC CHEMISTRY

Diaryl and Heteroaryl Sulfides: Synthesis via Sulfenyl Chlorides and Evaluation as Selective Anti-Breast-Cancer Agents

(2014) Ivelina M. Yonova et al.   JOURNAL OF ORGANIC CHEMISTRY

The Role of Aryne Distortions, Steric Effects, and Charges in Regioselectivities of Aryne Reactions

(2014) Jose M. Medina et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

N-Chlorosuccinimide-Promoted Regioselective Sulfenylation of Imidazoheterocycles at Room Temperature

(2014) Chitrakar Ravi et al.   ORGANIC LETTERS

Interception of benzyne with thioethers: a facile access to sulfur ylides under mild conditions

(2014) Hua-Dong Xu et al.   RSC Advances

Iodine-Catalyzed Regioselective Sulfenylation of Indoles with Sulfonyl Hydrazides

(2013) Fu-Lai Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

C–N bond forming cross-coupling reactions: an overview

(2013) Jitender Bariwal et al.   CHEMICAL SOCIETY REVIEWS

Addition of Cyclic Ureas and 1-Methyl-2-oxazolidone to Pyridynes: A New Approach to Pyridodiazepines, Pyridodiazocines, and Pyridooxazepines

(2013) Nozomi Saito et al.   ORGANIC LETTERS

Iodine-catalyzed oxidative system for 3-sulfenylation of indoles with disulfides using DMSO as oxidant under ambient conditions in dimethyl carbonate

(2012) Wenlei Ge et al.   GREEN CHEMISTRY

Mechanistic Assessment of SNAr Displacement of Halides from 1-Halo-2,4-dinitrobenzenes by Selected Primary and Secondary Amines: Brønsted and Mayr Analyses

(2012) Ik-Hwan Um et al.   JOURNAL OF ORGANIC CHEMISTRY

Steric Effects Compete with Aryne Distortion To Control Regioselectivities of Nucleophilic Additions to 3-Silylarynes

(2012) Sarah M. Bronner et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Use of benzynes for the synthesis of heterocycles

(2012) Anton V. Dubrovskiy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition-Metal-Free Electrophilic Amination of Arylboroxines

(2012) Qing Xiao et al.   ORGANIC LETTERS

Organocatalytic, Oxidative, Intermolecular Amination and Hydrazination of Simple Arenes at Ambient Temperature

(2012) Rajarshi Samanta et al.   ORGANIC LETTERS

A C–N insertion of β-lactam to benzyne: unusual formation of acridone

(2012) Jimin Kim et al.   TETRAHEDRON LETTERS

Synthesis of di(hetero)aryl sulfides by directly using arylsulfonyl chlorides as a sulfur source

(2011) Qian Wu et al.   CHEMICAL COMMUNICATIONS

Benzimidazolones: A New Class of Selective Peroxisome Proliferator-Activated Receptor γ (PPARγ) Modulators

(2011) Weiguo Liu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Intermolecular Oxidative C–N Bond Formation under Metal-Free Conditions: Control of Chemoselectivity between Aryl sp2and Benzylic sp3C–H Bond Imidation

(2011) Hyun Jin Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Free Intermolecular Oxidative C–N Bond Formation via Tandem C–H and N–H Bond Functionalization

(2011) Abhishek A. Kantak et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Insertion of Arynes into Thioureas: A New Amidine Synthesis

(2011) Kallolmay Biswas et al.   ORGANIC LETTERS

Identification and Development of Novel Inhibitors ofToxoplasma gondiiEnoyl Reductase

(2010) Suresh K. Tipparaju et al.   JOURNAL OF MEDICINAL CHEMISTRY

Indolyne and Aryne Distortions and Nucleophilic Regioselectivites

(2010) Paul H.-Y. Cheong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indolyne Experimental and Computational Studies: Synthetic Applications and Origins of Selectivities of Nucleophilic Additions

(2010) G-Yoon J. Im et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Quantitative Structure Activity Relationship (QSAR) Analysis of Substituted 4-Oxothiazolidines and 5-Arylidines as Lipoxygenase Inhibitors

(2010) A.N. Choudhary et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Regioselective Reactions of Highly Substituted Arynes

(2010) Pamela M. Tadross et al.   ORGANIC LETTERS

Transition-Metal-Free Electrophilic Amination between Aryl Grignard Reagents andN-Chloroamines

(2010) Takuji Hatakeyama et al.   ORGANIC LETTERS

Dialkylbiaryl phosphines in Pd-catalyzed amination: a user's guide

(2010) David S. Surry et al.   Chemical Science

A 1,8-Naphthyridone Derivative Targets the HIV-1 Tat-Mediated Transcription and Potently Inhibits the HIV-1 Replication

(2009) Serena Massari et al.   JOURNAL OF MEDICINAL CHEMISTRY

Insertion of Benzene Rings into the Amide Bond: One-Step Synthesis of Acridines and Acridones from Aryl Amides

(2009) Didier G. Pintori et al.   ORGANIC LETTERS

Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

(2008) John F. Hartwig   ACCOUNTS OF CHEMICAL RESEARCH

Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles†

(2008) Dawei Ma et al.   ACCOUNTS OF CHEMICAL RESEARCH

Sequential Metal-CatalyzedN-Heteroarylation and C–C Cross-Coupling Reactions: An Expedient Route to Tris(hetero)aryl Systems

(2008) Jamie S. Siddle et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 1. Synthesis and Structure−Activity Relationship of a Class of Human Immunodeficiency Virus type 1 Integrase Inhibitors†

(2008) Serena Pasquini et al.   JOURNAL OF MEDICINAL CHEMISTRY