Dialkylbiaryl phosphines in Pd-catalyzed amination: a user's guide

Bases and Basic Materials in Chemical and Environmental Processes. Liquid versus Solid Basicity

(2010) Guido Busca   CHEMICAL REVIEWS

Pd-Catalyzed Cross-Coupling Reactions of Amides and Aryl Mesylates

(2010) Karin Dooleweerdt et al.   ORGANIC LETTERS

Palladium-catalyzed coupling of functionalized primary and secondary amines with aryl and heteroaryl halides: two ligands suffice in most cases

(2010) Debabrata Maiti et al.   Chemical Science

Nine Times Fluoride can be Good for your Syntheses.Not just Cheaper: Nonafluorobutanesulfonates as Intermediates for Transition Metal-Catalyzed Reactions

(2009) Jens Högermeier et al.   ADVANCED SYNTHESIS & CATALYSIS

Recent Applications of Palladium-Catalyzed Coupling Reactions in the Pharmaceutical, Agrochemical, and Fine Chemical Industries

(2009) Christian Torborg et al.   ADVANCED SYNTHESIS & CATALYSIS

Room-Temperature Copper-Catalyzed Carbon-Nitrogen Coupling of Aryl Iodides and Bromides Promoted by Organic Ionic Bases

(2009) Chu-Ting Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organotrifluoroborates and Monocoordinated Palladium Complexes as Catalysts—A Perfect Combination for Suzuki–Miyaura Coupling

(2009) Gary A. Molander et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Phenylaminopyrimidines as inhibitors of Janus kinases (JAKs)

(2009) Christopher J. Burns et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

N-substituted 2′-(aminoaryl)benzothiazoles as kinase inhibitors: Hit identification and scaffold hopping

(2009) Stefan Tasler et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Benzo[c][2,7]naphthyridines as inhibitors of PDK-1

(2009) Kyung-Hee Kim et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Part 1: Structure–Activity Relationship (SAR) investigations of fused pyrazoles as potent, selective and orally available inhibitors of p38α mitogen-activated protein kinase

(2009) Ryan P. Wurz et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Hydrophilic Ligands and Their Application in Aqueous-Phase Metal-Catalyzed Reactions

(2009) Kevin H. Shaughnessy   CHEMICAL REVIEWS

Sterically demanding trialkylphosphines for palladium-catalyzed cross coupling reactions—alternatives to PtBu3

(2009) Christoph A. Fleckenstein et al.   CHEMICAL SOCIETY REVIEWS

A General Palladium-Catalyzed Amination of Aryl Halides with Ammonia

(2009) Thomas Schulz et al.   CHEMISTRY-A EUROPEAN JOURNAL

Kinase Domain Mutations in Cancer: Implications for Small Molecule Drug Design Strategies

(2009) Jack A. Bikker et al.   JOURNAL OF MEDICINAL CHEMISTRY

On the behavior of amines in the presence of Pd0 and PdII species

(2009) Jacques Muzart   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Room-Temperature Pd-Catalyzed Amidation of Aryl Bromides Usingtert-Butyl Carbamate

(2009) Swapna Bhagwanth et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed N-Arylation of Secondary Acyclic Amides: Catalyst Development, Scope, and Computational Study

(2009) Jacqueline D. Hicks et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd-Catalyzed Conversion of Aryl Chlorides, Triflates, and Nonaflates to Nitroaromatics

(2009) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Orthogonal Cu- and Pd-Based Catalyst Systems for the O- and N-Arylation of Aminophenols

(2009) Debabrata Maiti et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Efficient Process for Pd-Catalyzed C−N Cross-Coupling Reactions of Aryl Iodides: Insight Into Controlling Factors

(2009) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Coupling of Ammonia with Aryl Chlorides, Bromides, Iodides, and Sulfonates: A General Method for the Preparation of Primary Arylamines

(2009) Giang D. Vo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Influence of Biaryl Phosphine Structure on C−N and C−C Bond Formation

(2009) Ramendra Pratap et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Modular Synthesis of Indoles from Imines ando-Dihaloarenes oro-Chlorosulfonates by a Pd-Catalyzed Cascade Process

(2009) José Barluenga et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Theoretical Bond Dissociation Energies of Halo-Heterocycles: Trends and Relationships to Regioselectivity in Palladium-Catalyzed Cross-Coupling Reactions

(2009) Yeimy Garcia et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

[2.2]Paracyclophane-based monophosphine ligand for palladium-catalyzed cross-coupling reactions of aryl chlorides

(2009) Jiwu Ruan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A General Method for the Synthesis of Unsymmetrically Substituted Ureas via Palladium-Catalyzed Amidation

(2009) Brian J. Kotecki et al.   ORGANIC LETTERS

An efficient system for the Pd-catalyzed cross-coupling of amides and aryl chlorides

(2009) Brett P. Fors et al.   TETRAHEDRON

An improved synthesis of N-aryl and N-heteroaryl substituted homopiperazines—from conventional thermal conditions to scaling-up using microwave heating

(2009) Uwe Schön et al.   TETRAHEDRON

Mild conditions for Pd-catalyzed conversion of aryl bromides to primary anilines using benzophenone imine

(2009) Swapna Bhagwanth et al.   TETRAHEDRON LETTERS

Simple, efficient protocols for the Pd-catalyzed cross-coupling reaction of aryl chlorides and dimethylamine

(2009) Brian K. Lee et al.   TETRAHEDRON LETTERS

Palladium-Catalyzed Suzuki−Miyaura Cross-Coupling Reactions Employing Dialkylbiaryl Phosphine Ligands

(2008) Ruben Martin et al.   ACCOUNTS OF CHEMICAL RESEARCH

Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

(2008) John F. Hartwig   ACCOUNTS OF CHEMICAL RESEARCH

Well-Defined N-Heterocyclic Carbenes−Palladium(II) Precatalysts for Cross-Coupling Reactions

(2008) Nicolas Marion et al.   ACCOUNTS OF CHEMICAL RESEARCH

A New Hybrid Phosphine Ligand for Palladium-Catalyzed Amination of Aryl Halides

(2008) Ken Suzuki et al.   ADVANCED SYNTHESIS & CATALYSIS

Electron-Rich, Bicyclic Biaryl-Like KITPHOS Monophosphinesvia[4+2] Cycloaddition between 1-Alkynylphosphine Oxides and Anthracene: Highly Efficient Ligands for Palladium-Catalysed CN and CC Bond Formation

(2008) Simon Doherty et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium-Catalyzed Amination of Aryl Mesylates

(2008) Chau Ming So et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Biaryl Phosphane Ligands in Palladium-Catalyzed Amination

(2008) David S. Surry et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Evaluation of indazole-based compounds as a new class of potent KDR/VEGFR-2 inhibitors

(2008) David Bauer et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Pd-catalyzed diarylation of aniline—a way to a non-linear bis(terpyridyl) ligand providing increased electronic communication

(2008) Olof Johansson et al.   DALTON TRANSACTIONS

Role of the ligand in the palladium-catalyzed C-2 and C-3 arylation of the indole magnesium salt

(2008) M. V. Nikulin et al.   DOKLADY CHEMISTRY

Irregularities in the Effect of Potassium Phosphate in Ynamide Synthesis

(2008) Karin Dooleweerdt et al.   JOURNAL OF ORGANIC CHEMISTRY

Vinylation of Aromatic Halides Using Inexpensive Organosilicon Reagents. Illustration of Design of Experiment Protocols

(2008) Scott E. Denmark et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Highly Active Catalyst for Pd-Catalyzed Amination Reactions: Cross-Coupling Reactions Using Aryl Mesylates and the Highly Selective Monoarylation of Primary Amines Using Aryl Chlorides

(2008) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Reactive, General and Long-Lived Catalysts for Palladium-Catalyzed Amination of Heteroaryl and Aryl Chlorides, Bromides, and Iodides: Scope and Structure–Activity Relationships

(2008) Qilong Shen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A New Class of Easily Activated Palladium Precatalysts for Facile C−N Cross-Coupling Reactions and the Low Temperature Oxidative Addition of Aryl Chlorides

(2008) Mark R. Biscoe et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

[(CyPF-tBu)PdCl2]: An Air-Stable, One-Component, Highly Efficient Catalyst for Amination of Heteroaryl and Aryl Halides

(2008) Qilong Shen et al.   ORGANIC LETTERS

Water-Mediated Catalyst Preactivation: An Efficient Protocol for C−N Cross-Coupling Reactions

(2008) Brett P. Fors et al.   ORGANIC LETTERS

A Rapid, Large-Scale Synthesis of a Potent Cholecystokinin (CCK) 1R Receptor Agonist

(2008) Jeffrey T. Kuethe et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

A Practical Synthesis of a Diazepinylbenzoic Acid, a Retinoid X Receptor Antagonist

(2008) Xinglong Jiang et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Streamlined Synthesis of the Bippyphos Family of Ligands and Cross-Coupling Applications

(2008) Gregory J. Withbroe et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Study of the microwave-assisted hydrolysis of nitriles and esters and the implementation of this system in rapid microwave-assisted Pd-catalyzed amination

(2008) Gitte Van Baelen et al.   TETRAHEDRON

Delineating ligand effects in intramolecular aryl amidation reactions: formation of a novel spiro-heterocycle by a tandem cyclisation process

(2008) Emma L. Cropper et al.   TETRAHEDRON

Pd-catalyzed coupling of arylamines and 2-bromo-3,3,3-trifluoropropene

(2007) Tatsuhito Kino et al.   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Multicomponent and one-pot synthesis of trisubstituted pyridines through a Pd-catalyzed cross-coupling/cross-coupling/cycloaddition sequence

(2007) José Barluenga et al.   TETRAHEDRON