Rational Design of Amine Nucleophiles for Dynamic Kinetic Resolution of Azlactones Leading to Highly Enantioselective Synthesis of Bisamides

Catalytic Asymmetric Inverse-Electron-Demand Oxa-Diels-Alder Reaction of In Situ Generatedortho-Quinone Methides with 3-Methyl-2-Vinylindoles

(2015) Jia-Jia Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic dynamic kinetic resolution of azlactones to construct chiral N-acyl amino acid oxime esters

(2015) Kunru Yu et al.   CHEMICAL COMMUNICATIONS

Brine-Stabilized 2,2,2-Trifluorodiazoethane and Its Application in the Synthesis of CF3–Substituted Cyclopropane α-Amino Acids

(2015) Chuan-Le Zhu et al.   ORGANIC LETTERS

Chiral Phosphoric Acid Catalyzed Asymmetric Synthesis of 2-Substituted 2,3-Dihydro-4-quinolones by a Protecting-Group-Free Approach

(2015) Kodai Saito et al.   ORGANIC LETTERS

Recent Advances in Chiral Phosphoric Acid Catalyzed Asymmetric Reactions for the Synthesis of Enantiopure Indole Derivatives

(2015) Hua Wu et al.   SYNTHESIS-STUTTGART

A Practical Aryl Unit for Azlactone Dynamic Kinetic Resolution: Orthogonally Protected Products and A Ligation-Inspired Coupling Process

(2014) Sean Tallon et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric Arylative Dearomatization of 2,3-Disubstituted Indoles Enabled by Tandem Reactions

(2014) Yu-Chen Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Formation of All-Carbon Quaternary Stereocenters from Indoles and Tertiary Alcohols Bearing A Directing Group

(2014) Wanxiang Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Diastereoselectivity in prebiotically relevant 5(4H)-oxazolone-mediated peptide couplings

(2014) Damien Beaufils et al.   CHEMICAL COMMUNICATIONS

Complete Field Guide to Asymmetric BINOL-Phosphate Derived Brønsted Acid and Metal Catalysis: History and Classification by Mode of Activation; Brønsted Acidity, Hydrogen Bonding, Ion Pairing, and Metal Phosphates

(2014) Dixit Parmar et al.   CHEMICAL REVIEWS

Peptide-Catalyzed Conversion of Racemic Oxazol-5(4H)-ones into Enantiomerically Enriched α-Amino Acid Derivatives

(2014) Anthony J. Metrano et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Transfer Hydrogenation of Ketimines by Indoline as Recyclable Hydrogen Donor

(2014) Kodai Saito et al.   ORGANIC LETTERS

Discussion of absolute configuration for bioactive Griseusins by comparing computed optical rotations and electronic circular dichroism with the experimental results

(2014) Hua-Jie Zhu et al.   TETRAHEDRON

Vibrational circular dichroism study for natural bioactive schizandrin and reassignment of its absolute configuration

(2014) Ping He et al.   TETRAHEDRON LETTERS

Histone Deacetylase Inhibitors with Enhanced Enzymatic Inhibition Effects and Potent in vitro and in vivo Antitumor Activities

(2013) Lei Zhang et al.   ChemMedChem

C-5′-Substituted Cinchona Alkaloid Derivatives Catalyse the First Highly Enantioselective Dynamic Kinetic Resolutions of Azlactones by Thiolysis

(2013) Carole Palacio et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Mimicking hemoproteins: a new synthetic metalloenzyme based on a Fe(III)-mesoporphyrin functionalized by two helical decapeptides

(2013) Mariano Venanzi et al.   JOURNAL OF PEPTIDE SCIENCE

Pd-Catalyzed Asymmetric Allylic Alkylation of Pyrazol-5-ones with Allylic Alcohols: The Role of the Chiral Phosphoric Acid in C–O Bond Cleavage and Stereocontrol

(2013) Zhong-Lin Tao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Challenges in the assignment of relative and absolute configurations of complex molecules: computation can resolve conflicts between theory and experiment

(2013) Jie Ren et al.   TETRAHEDRON

Brønsted acid catalyzed azlactone ring opening by nucleophiles

(2013) Adriane A. Pereira et al.   TETRAHEDRON

Highly stereoselective Michael addition of azlactones to electron-deficient triple bonds under P-spiro chiral iminophosphorane catalysis: importance of protonation pathway

(2013) Daisuke Uraguchi et al.   Chemical Science

Efficient Routes to Carbon–Silicon Bond Formation for the Synthesis of Silicon-Containing Peptides and Azasilaheterocycles

(2012) Geanna K. Min et al.   ACCOUNTS OF CHEMICAL RESEARCH

Enantioselective Construction of Pyrroloindolines Catalyzed by Chiral Phosphoric Acids: Total Synthesis of (−)-Debromoflustramine B

(2012) Zuhui Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Progression of Absolute Configuration Determination in Natural Product Chemistry Using Optical Rotation (Dispersion), Matrix Determinant and Electronic Circular Dichroism Methods

(2012) Sheng-Ding Zhao et al.   CURRENT ORGANIC CHEMISTRY

The Dynamic Kinetic Resolution of Azlactones with Thiol Nucleophiles Catalyzed by Arylated, Deoxygenated Cinchona Alkaloids

(2012) Zaida Rodríguez-Docampo et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Regio-, Diastereo-, and Enantioselective 1,6- and 1,8-Additions of Azlactones to Di- and Trienyl N-Acylpyrroles

(2012) Daisuke Uraguchi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly enantioselective trapping of zwitterionic intermediates by imines

(2012) Huang Qiu et al.   Nature Chemistry

Origin of Enantioselectivity in Benzotetramisole-Catalyzed Dynamic Kinetic Resolution of Azlactones

(2012) Peng Liu et al.   ORGANIC LETTERS

Brønsted-Acid-Catalyzed Asymmetric Multicomponent Reactions for the Facile Synthesis of Highly Enantioenriched Structurally Diverse Nitrogenous Heterocycles

(2011) Jie Yu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Enantioselective synthesis of α-deuterium labelled chiral α-amino acids via dynamic kinetic resolution of racemic azlactones

(2011) Joong-Suk Oh et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Solid-phase de novo synthesis of a (±)-2-deoxy-glycoside

(2010) Céline Lucchesi et al.   CARBOHYDRATE RESEARCH

Benzotetramisole-Catalyzed Dynamic Kinetic Resolution of Azlactones

(2010) Xing Yang et al.   ORGANIC LETTERS

Dynamic Kinetic Resolution of Azlactones Catalyzed by Chiral Brønsted Acids

(2010) Guojian Lu et al.   ORGANIC LETTERS

Chiral Phosphoric Acids as Versatile Catalysts for Enantioselective Transformations

(2010) Masahiro Terada   SYNTHESIS-STUTTGART

Assignment of the Absolute Configuration ofConcentricolide- Absolute Configuration Determination of Its Bioactive Analogs Using DFT Methods

(2009) Jie Ren et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Site-Directed Asymmetric Quaternization of a Peptide Backbone at a C-Terminal Azlactone

(2008) Daisuke Uraguchi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Binaphthol-derived phosphoric acid as a versatile catalyst for enantioselective carbon–carbon bond forming reactions

(2008) Masahiro Terada   CHEMICAL COMMUNICATIONS

Organocatalytic Asymmetric Addition of Alcohols and Thiols to Activated Electrophiles: Efficient Dynamic Kinetic Resolution and Desymmetrization Protocols

(2008) Aldo Peschiulli et al.   JOURNAL OF ORGANIC CHEMISTRY

Chemoenzymatic preparation of enantiopure l-benzofuranyl- and l-benzo[b]thiophenyl alanines

(2008) Paula Veronica Podea et al.   TETRAHEDRON-ASYMMETRY

Structural Parameter Characterization and Bioactivity Simulation Based on Peptide Sequence

(2008) Mao Shu et al.   Quantitative structure-activity relationships & combinatorial science

Amino acid derivatives as histone deacetylase inhibitors

(2007) Jed L. Hubbs et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS