Multicomponent coupling and macrocyclization enabled by Rh(III)-catalyzed dual C–H activation: Macrocyclic oxime inhibitor of influenza H1N1
出版年份 2022 全文链接
标题
Multicomponent coupling and macrocyclization enabled by Rh(III)-catalyzed dual C–H activation: Macrocyclic oxime inhibitor of influenza H1N1
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关键词
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出版物
Chem
Volume -, Issue -, Pages -
出版商
Elsevier BV
发表日期
2022-11-10
DOI
10.1016/j.chempr.2022.10.019
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Marine furanocembranoids-inspired macrocycles enabled by Pd-catalyzed unactivated C(sp3)-H olefination mediated by donor/donor carbenes
- (2021) Jiping Hao et al. Nature Communications
- Mechanism-Guided Development of Transition-Metal-Catalyzed C–N Bond-Forming Reactions Using Dioxazolones as the Versatile Amidating Source
- (2021) Seung Youn Hong et al. ACCOUNTS OF CHEMICAL RESEARCH
- Use of Strain-Release for the Diastereoselective Construction of Quaternary Carbon Centers
- (2021) Tobias Pinkert et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Nitrene-mediated intermolecular N–N coupling for efficient synthesis of hydrazides
- (2021) Hao Wang et al. Nature Chemistry
- Zearalenone and the Immune Response
- (2021) Cristina Valeria Bulgaru et al. Toxins
- Late-stage C–H functionalization offers new opportunities in drug discovery
- (2021) Lucas Guillemard et al. Nature Reviews Chemistry
- Transition-Metal-Catalyzed, Coordination-Assisted Functionalization of Nonactivated C(sp3)–H Bonds
- (2021) Bin Liu et al. CHEMICAL REVIEWS
- Pd-Catalyzed Decarboxylative Olefination: Stereoselective Synthesis of Polysubstituted Butadienes and Macrocyclic P-glycoprotein Inhibitors
- (2020) Bichao Song et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Evaluation of 3-Dimensionality in Approved and Experimental Drug Space
- (2020) Kathleen E. Prosser et al. ACS Medicinal Chemistry Letters
- A modular biomimetic strategy for the synthesis of macrolide P-glycoprotein inhibitors via Rh-catalyzed C-H activation
- (2020) Lu Chen et al. Nature Communications
- Dioxazolones: Stable Substrates for the Catalytic Transfer of Acyl Nitrenes
- (2020) Kaj M. van Vliet et al. ACS Catalysis
- The rise of molecular simulations in fragment-based drug design (FBDD): an overview
- (2020) Maicol Bissaro et al. DRUG DISCOVERY TODAY
- DrugSpaceX: a large screenable and synthetically tractable database extending drug space
- (2020) Tianbiao Yang et al. NUCLEIC ACIDS RESEARCH
- Unconventional Macrocyclizations in Natural Product Synthesis
- (2020) Iakovos Saridakis et al. ACS Central Science
- Palladium-Catalyzed C(sp3)–H Bond Functionalization of Aliphatic Amines
- (2019) Chuan He et al. Chem
- Structure-Based Macrocycle Design in Small-Molecule Drug Discovery and Simple Metrics To Identify Opportunities for Macrocyclization of Small-Molecule Ligands
- (2019) Maxwell D. Cummings et al. JOURNAL OF MEDICINAL CHEMISTRY
- Iridium-Catalyzed Enantioselective C(sp3)–H Amidation Controlled by Attractive Noncovalent Interactions
- (2019) Hao Wang et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Strategies for the Diversity-Oriented Synthesis of Macrocycles
- (2019) Kim T. Mortensen et al. CHEMICAL REVIEWS
- α-Branched amines by catalytic 1,1-addition of C–H bonds and aminating agents to terminal alkenes
- (2019) Soham Maity et al. Nature Catalysis
- Synthesis of Biaryl-Bridged Cyclic Peptides via Catalytic Oxidative Cross-Coupling Reactions
- (2019) Mor Ben-Lulu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- A general strategy for synthesis of cyclophane-braced peptide macrocycles via palladium-catalysed intramolecular sp3 C−H arylation
- (2018) Xuekai Zhang et al. Nature Chemistry
- Selective formation of γ-lactams via C–H amidation enabled by tailored iridium catalysts
- (2018) Seung Youn Hong et al. SCIENCE
- Revisiting Arene C(sp2 )−H Amidation by Intramolecular Transfer of Iridium Nitrenoids: Evidence for a Spirocyclization Pathway
- (2018) Yeongyu Hwang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Backbone-Enabled Directional Peptide Macrocyclization through Late-Stage Palladium-Catalyzed δ-C(sp2 )−H Olefination
- (2018) Zengbing Bai et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Chromopynones are pseudo natural product glucose uptake inhibitors targeting glucose transporters GLUT-1 and -3
- (2018) George Karageorgis et al. Nature Chemistry
- Rapamycin-inspired macrocycles with new target specificity
- (2018) Zufeng Guo et al. Nature Chemistry
- Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
- (2016) Yu Zhou et al. CHEMICAL REVIEWS
- Palladium-Catalyzed Transformations of Alkyl C–H Bonds
- (2016) Jian He et al. CHEMICAL REVIEWS
- Twenty years on: the impact of fragments on drug discovery
- (2016) Daniel A. Erlanson et al. NATURE REVIEWS DRUG DISCOVERY
- Functionalization of C(sp3)-H bonds using a transient directing group
- (2016) F.-L. Zhang et al. SCIENCE
- Rhodium(III)-Catalyzed Amidation of Unactivated C(sp3)H Bonds
- (2015) He Wang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds
- (2015) Albert Isidro-Llobet et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- A C–H bond activation-based catalytic approach to tetrasubstituted chiral allenes
- (2015) Shangze Wu et al. Nature Communications
- New peptide architectures through C–H activation stapling between tryptophan–phenylalanine/tyrosine residues
- (2015) Lorena Mendive-Tapia et al. Nature Communications
- Peptide Nanotubes
- (2014) Ian W. Hamley ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Diversity-Oriented Synthesis of Drug-Like Macrocyclic Scaffolds Using an Orthogonal Organo- and Metal Catalysis Strategy
- (2014) André Grossmann et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Macrocyclic Drugs and Synthetic Methodologies toward Macrocycles
- (2013) Xufen Yu et al. MOLECULES
- A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling
- (2013) Henning S. G. Beckmann et al. Nature Chemistry
- Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation
- (2012) Huijun Dong et al. CHEMICAL COMMUNICATIONS
- C–C, C–O and C–N bond formation via rhodium(iii)-catalyzed oxidative C–H activation
- (2012) Guoyong Song et al. CHEMICAL SOCIETY REVIEWS
- Gold(I)-Catalyzed Coupling Reactions for the Synthesis of Diverse Small Molecules Using the Build/Couple/Pair Strategy
- (2009) Tuoping Luo et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- The rise of fragment-based drug discovery
- (2009) Christopher W. Murray et al. Nature Chemistry
- The exploration of macrocycles for drug discovery — an underexploited structural class
- (2008) Edward M. Driggers et al. NATURE REVIEWS DRUG DISCOVERY
- Towards the Optimal Screening Collection: A Synthesis Strategy
- (2007) Thomas E. Nielsen et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
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