A facile synthesis of 2H-indazoles under neat conditions and further transformation into aza-γ-carboline alkaloid analogues in a tandem one-pot fashion

Synthesis and biological activity ofN-substituted-tetrahydro-γ-carbolines containing peptide residues

(2014) Nadezhda V Sokolova et al.   Beilstein Journal of Organic Chemistry

A direct access to bioactive fused N-heterocyclic acetic acid derivatives

(2014) Raju Adepu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Isovanillin derived N-(un)substituted hydroxylamines possessing an ortho-allylic group: valuable precursors to bioactive N-heterocycles

(2014) Balakrishna Dulla et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Regioselective Synthesis of 2H-Indazoles Using a Mild, One-Pot Condensation–Cadogan Reductive Cyclization

(2014) Nathan E. Genung et al.   ORGANIC LETTERS

Microwave-assisted facile synthesis of [a]-annelated pyrazolopyrroloindoles via intramolecular azomethine imine 1,3-dipolar cycloaddition

(2014) Anand H. Shinde et al.   TETRAHEDRON LETTERS

Surfactant-Type Brønsted Acid Catalyzed Stereoselective Synthesis oftrans-3-Alkenyl Indazoles from Triazenylaryl Allylic Alcohols in Water

(2013) Weijun Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, Synthesis and Biological Evaluation of Pazopanib Derivatives as Antitumor Agents

(2013) Yuping Jia et al.   Chemical Biology & Drug Design

Metal-free nitro-carbocyclization of activated alkenes: a direct approach to synthesize oxindoles by cascade C–N and C–C bond formation

(2013) Tao Shen et al.   CHEMICAL COMMUNICATIONS

How to measure reaction temperature in microwave-heated transformations

(2013) C. Oliver Kappe   CHEMICAL SOCIETY REVIEWS

Benign by design: catalyst-free in-water, on-water green chemical methodologies in organic synthesis

(2013) Manoj B. Gawande et al.   CHEMICAL SOCIETY REVIEWS

Solvent-Free and Catalysts-Free Chemistry: A Benign Pathway to Sustainability

(2013) Manoj B. Gawande et al.   ChemSusChem

A facile protocol for the synthesis of 3-aminoimidazo-fused heterocycles via the Groebke–Blackburn–Bienayme reaction under catalyst-free and solvent-free conditions

(2013) Shinde Vidyacharan et al.   GREEN CHEMISTRY

Process Development of C–N Cross-Coupling and Enantioselective Biocatalytic Reactions for the Asymmetric Synthesis of Niraparib

(2013) Cheol K. Chung et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

A robust protocol for Pd(ii)-catalyzed C-3 arylation of (1H) indazoles and pyrazoles: total synthesis of nigellidine hydrobromide

(2013) Mengchun Ye et al.   Chemical Science

CuO nanoparticle catalysed synthesis of 2H-indazoles under ligand free conditions

(2013) Nilufa Khatun et al.   RSC Advances

Green synthesis and anti-infective activities of fluorinated pyrazoline derivatives

(2012) Sharad N. Shelke et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Regioselective zincation of indazoles using TMP2Zn and Negishi cross-coupling with aryl and heteroaryl iodides

(2012) Andreas Unsinn et al.   CHEMICAL COMMUNICATIONS

Chemistry and Biology Of Multicomponent Reactions

(2012) Alexander Dömling et al.   CHEMICAL REVIEWS

A One-Pot, Copper-Catalyzed Cascade Route to 2-Indolyl-C-glycosides

(2012) Parthasarathi Subramanian et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

From biomass to medicines. A simple synthesis of indolo[3,2-c]quinolines, antimalarial alkaloid isocryptolepine, and its derivatives

(2012) Maxim G. Uchuskin et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

An efficient synthesis of 2H-indazoles via reductive cyclization of 2-nitrobenzylamines induced by low-valent titanium reagent

(2012) Fang Sun et al.   TETRAHEDRON

Acid and base catalyzed Davis–Beirut reaction: experimental and theoretical mechanistic studies and synthesis of novel 3-amino-2H-indazoles

(2012) Belem Avila et al.   TETRAHEDRON LETTERS

Synthesis and antimalarial evaluation of novel isocryptolepine derivatives

(2011) Louise R. Whittell et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A general and efficient approach to 2H-indazoles and 1H-pyrazoles through copper-catalyzed intramolecular N–N bond formation under mild conditions

(2011) Jiantao Hu et al.   CHEMICAL COMMUNICATIONS

Green chemistry oriented organic synthesis in water

(2011) Marc-Olivier Simon et al.   CHEMICAL SOCIETY REVIEWS

Environmentally benign synthesis of heterocyclic compounds by combined microwave-assisted heterogeneous catalytic approaches†

(2011) Arif Daştan et al.   GREEN CHEMISTRY

Synthesis of 2H-Indazoles by the [3 + 2] Dipolar Cycloaddition of Sydnones with Arynes

(2011) Yuesi Fang et al.   JOURNAL OF ORGANIC CHEMISTRY

Consecutive Condensation, C–N and N–N Bond Formations: A Copper- Catalyzed One-Pot Three-Component Synthesis of 2H-Indazole

(2011) Manian Rajesh Kumar et al.   ORGANIC LETTERS

An efficient new route towards biologically active isocryptolepine and γ-carboline derivatives using an intramolecular thermal electrocyclization strategy

(2011) Dattatray G. Hingane et al.   TETRAHEDRON LETTERS

SMT-A07, a 3-(Indol-2-yl) indazole derivative, induces apoptosis of leukemia cells in vitro

(2010) Shijing Qian et al.   MOLECULAR AND CELLULAR BIOCHEMISTRY

Synthesis of 2H-Indazoles by the [3 + 2] Cycloaddition of Arynes and Sydnones

(2010) Chunrui Wu et al.   ORGANIC LETTERS

Intramolecular Fe(II)-Catalyzed N−O or N−N Bond Formation from Aryl Azides

(2010) Benjamin J. Stokes et al.   ORGANIC LETTERS

A General and Mild Palladium-Catalyzed Domino Reaction for the Synthesis of 2H-Indazoles

(2009) Nis Halland et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Solvent-Free Heterocyclic Synthesis

(2009) Marcos A. P. Martins et al.   CHEMICAL REVIEWS

Efficient Traceless Solid-Phase Synthesis of 3,4-Dihydropyrazino[1,2-b]indazoles and Their 6-Oxides

(2009) Naděžda Pudelová et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Microwave-assisted Cadogan reaction for the synthesis of 2-aryl-2H-indazoles, 2-aryl-1H-benzimidazoles, 2-carbonylindoles, carbazole, and phenazine

(2009) Evelyn Cuevas Creencia et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Oxadiazolylindazole Sodium Channel Modulators are Neuroprotective toward Hippocampal Neurones

(2009) Lisa A. Clutterbuck et al.   JOURNAL OF MEDICINAL CHEMISTRY

Indazoles: Regioselective Protection and Subsequent Amine Coupling Reactions

(2009) David J. Slade et al.   JOURNAL OF ORGANIC CHEMISTRY

Four-Component Domino Reaction Leading to Multifunctionalized Quinazolines

(2009) Bo Jiang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Preparation of Polyfunctional Indazoles and Heteroarylazo Compounds Using Highly Functionalized Zinc Reagents

(2009) Benjamin Haag et al.   ORGANIC LETTERS

Direct Arylations of 2H-Indazoles On Water

(2009) Stephan A. Ohnmacht et al.   ORGANIC LETTERS

Microwave dielectric heating in synthetic organic chemistry

(2008) C. Oliver Kappe   CHEMICAL SOCIETY REVIEWS

Recent Advances in the Chemistry of Indazoles

(2008) Andreas Schmidt et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

New Route to the Synthesis of the Isocryptolepine Alkaloid and Its Related Skeletons Using a Modified Pictet-Spengler Reaction

(2008) Piyush K. Agarwal et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Solid-Phase Synthesis of Biologically Active Benzoannelated Nitrogen Heterocycles: An Update

(2008) Carmen Gil et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Synthesis of Annulated 2H-Indazoles and 1,2,3- and 1,2,4-Triazoles via a One-Pot Palladium-Catalyzed Alkylation/Direct Arylation Reaction

(2008) Benoît Laleu et al.   JOURNAL OF ORGANIC CHEMISTRY

A Practical, Metal-Free Synthesis of 1H-Indazoles

(2008) Carla M. Counceller et al.   ORGANIC LETTERS