Development of a Fluorescence-based Trypanosoma cruzi CYP51 Inhibition Assay for Effective Compound Triaging in Drug Discovery Programmes for Chagas Disease
Development of a Fluorescence-based Trypanosoma cruzi CYP51 Inhibition Assay for Effective Compound Triaging in Drug Discovery Programmes for Chagas Disease
作者
关键词
Trypanosoma cruzi, Chagas disease, Drug discovery, Parasitic diseases, Sterols, Drug metabolism, High throughput screening, Enzyme metabolism
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