Development of a Fluorescence-based Trypanosoma cruzi CYP51 Inhibition Assay for Effective Compound Triaging in Drug Discovery Programmes for Chagas Disease

标题
Development of a Fluorescence-based Trypanosoma cruzi CYP51 Inhibition Assay for Effective Compound Triaging in Drug Discovery Programmes for Chagas Disease
作者
关键词
Trypanosoma cruzi, Chagas disease, Drug discovery, Parasitic diseases, Sterols, Drug metabolism, High throughput screening, Enzyme metabolism
出版物
PLoS Neglected Tropical Diseases
Volume 9, Issue 9, Pages e0004014
出版商
Public Library of Science (PLoS)
发表日期
2015-09-23
DOI
10.1371/journal.pntd.0004014

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