The Dopamine Stabilizer (−)-OSU6162 Occupies a Subpopulation of Striatal Dopamine D2/D3 Receptors: An [11C]Raclopride PET Study in Healthy Human Subjects
出版年份 2014 全文链接
标题
The Dopamine Stabilizer (−)-OSU6162 Occupies a Subpopulation of Striatal Dopamine D2/D3 Receptors: An [11C]Raclopride PET Study in Healthy Human Subjects
作者
关键词
-
出版物
NEUROPSYCHOPHARMACOLOGY
Volume 40, Issue 2, Pages 472-479
出版商
Springer Nature
发表日期
2014-09-24
DOI
10.1038/npp.2014.195
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- Rostrocaudal gradients of dopamine D2/3 receptor binding in striatal subregions measured with [11C]raclopride and high-resolution positron emission tomography
- (2013) Kati Alakurtti et al. NEUROIMAGE
- Placebo-controlled cross-over study of the monoaminergic stabiliser (−)-OSU6162 in mental fatigue following stroke or traumatic brain injury.
- (2012) Birgitta Johansson et al. ACTA NEUROPSYCHIATRICA
- In vivo quantification of striatal dopamine D2 receptor occupancy by JNJ-37822681 using [11C]raclopride and positron emission tomography
- (2012) Erik T te Beek et al. JOURNAL OF PSYCHOPHARMACOLOGY
- The dopamine stabilizers ACR16 and (−)-OSU6162 display nanomolar affinities at the σ-1 receptor
- (2012) K Sahlholm et al. MOLECULAR PSYCHIATRY
- No association between bone mass and prolactin levels among patients with schizophrenia
- (2011) Norio Sugawara et al. HUMAN PSYCHOPHARMACOLOGY-CLINICAL AND EXPERIMENTAL
- II. In vitro evidence that (−)-OSU6162 and (+)-OSU6162 produce their behavioral effects through 5-HT2A serotonin and D2 dopamine receptors
- (2011) Ethan S. Burstein et al. JOURNAL OF NEURAL TRANSMISSION
- I. In vivo evidence for partial agonist effects of (−)-OSU6162 and (+)-OSU6162 on 5-HT2A serotonin receptors
- (2011) Maria L. Carlsson et al. JOURNAL OF NEURAL TRANSMISSION
- Effects of the dopamine stabilizers (S)-(-)-OSU6162 and ACR16 on prolactin secretion in drug-naive and monoamine-depleted rats
- (2011) Johan P. Rung et al. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
- Analysis of the actions of the novel dopamine receptor-directed compounds (S)-OSU6162 and ACR16 at the D2 dopamine receptor
- (2010) Elodie Kara et al. BRITISH JOURNAL OF PHARMACOLOGY
- Application of Stable Isotope Methodology in the Evaluation of the Pharmacokinetics of (S,S)-3-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine Hydrochloride in Rats
- (2009) S. Yamazaki et al. DRUG METABOLISM AND DISPOSITION
- The dopaminergic stabilizers pridopidine (ACR16) and (−)-OSU6162 display dopamine D2 receptor antagonism and fast receptor dissociation properties
- (2009) Tino Dyhring et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- Co-operativity in agonist binding at the D2dopamine receptor: evidence from agonist dissociation kinetics
- (2009) Elodie Kara et al. JOURNAL OF NEUROCHEMISTRY
- Allosteric communication between protomers of dopamine class A GPCR dimers modulates activation
- (2009) Yang Han et al. Nature Chemical Biology
- Effects of (−)-OSU6162 and ACR16 on motor activity in rats, indicating a unique mechanism of dopaminergic stabilization
- (2008) Johan P. Rung et al. JOURNAL OF NEURAL TRANSMISSION
Add your recorded webinar
Do you already have a recorded webinar? Grow your audience and get more views by easily listing your recording on Peeref.
Upload NowCreate your own webinar
Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.
Create Now