Tautomeric origin of dual effects of N1-nicotinoyl-3-(4′-hydroxy-3′-methyl phenyl)-5-[(sub)phenyl]-2-pyrazolines on bacterial and viral strains: POM analyses as new efficient bioinformatics’ platform to predict and optimize bioactivity of drugs

Synthesis, studies and in-vitro antibacterial activity of N-substituted 5-(furan-2-yl)-phenyl pyrazolines

(2015) Mamta Rani et al.   Arabian Journal of Chemistry

Synthesis, antibacterial and antifungal activities of 3-aryl-5-(pyridin-3-yl)-4,5-dihydropyrazole-1-carbothioamide derivatives

(2012) M. Shekarchi et al.   Journal of the Iranian Chemical Society

Development of selective and reversible pyrazoline based MAO-B inhibitors: Virtual screening, synthesis and biological evaluation

(2011) Nibha Mishra et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide as anticancer and anti-inflammatory agents

(2011) Rafia Bashir et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Design, synthesis and antimycobacterial evaluation of novel 3-substituted-N-aryl-6,7-dimethoxy-3a,4-dihydro-3H-indeno[1,2-c]pyrazole-2-carboxamide analogues

(2011) Mohamed Jawed Ahsan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Chemical scaffolds with structural similarities to siderophores of nonribosomal peptide–polyketide origin as novel antimicrobials against Mycobacterium tuberculosis and Yersinia pestis

(2011) Julian A. Ferreras et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, molecular docking and evaluation of thiazolyl-pyrazoline derivatives as EGFR TK inhibitors and potential anticancer agents

(2011) Peng-Cheng Lv et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Pyrazoline based MAO inhibitors: Synthesis, biological evaluation and SAR studies

(2011) Monika Jagrat et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A novel class of trans-methylpyrazoline analogs of combretastatins: Synthesis and in-vitro biological testing

(2011) Megan Lee et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of some new 2-pyrazolines bearing benzene sulfonamide moiety as potential anti-inflammatory and anti-cancer agents

(2011) Sameena Bano et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of some novel benzofuran-2-yl(4,5-dihyro-3,5-substituted diphenylpyrazol-1-yl) methanones and studies on the antiproliferative effects and reversal of multidrug resistance of human MDR1-gene transfected mouse lymphoma cells in vitro

(2011) Shrey Parekh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Pregnenolone derivatives as potential anticancer agents

(2011) M. Iqbal Choudhary et al.   STEROIDS

Synthesis and in-vitro-antibacterial activity of [5-(furan-2-yl)-phenyl]-4,5-carbothioamide-pyrazolines

(2011) Mamta Rani et al.   Journal of Saudi Chemical Society

Synthesis and in vitro biology of Co(II), Ni(II), Cu(II) and Zinc(II) complexes of functionalized beta-diketone bearing energy buried potential antibacterial and antiviral O,O pharmacophore sites

(2011) Javed Sheikh et al.   Journal of Saudi Chemical Society

Synthesis, studies and in vitro antibacterial activity of some 5-(thiophene-2-yl)-phenyl pyrazoline derivatives

(2011) Mamta Rani et al.   Journal of Saudi Chemical Society

Development of selective and reversible pyrazoline based MAO-A inhibitors: Synthesis, biological evaluation and docking studies

(2010) Muthukumar Karuppasamy et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, analgesic and anti-inflammatory activities of some novel pyrazolines derivatives

(2010) Ratnadeep S. Joshi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and pharmacological study of 1-acetyl/propyl-3-aryl-5-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-2-pyrazoline

(2010) K.S. Girisha et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis, and antitubercular evaluation of novel series of 3-benzofuran-5-aryl-1-pyrazolyl-pyridylmethanone and 3-benzofuran-5-aryl-1-pyrazolylcarbonyl-4-oxo-naphthyridin analogs

(2010) Kuntal Manna et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and biological evaluation of N-substituted-3,5-diphenyl-2-pyrazoline derivatives as cyclooxygenase (COX-2) inhibitors

(2010) Rossella Fioravanti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal based biologically active compounds: Design, synthesis, and antibacterial/antifungal/cytotoxic properties of triazole-derived Schiff bases and their oxovanadium(IV) complexes

(2010) Zahid H. Chohan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Theoretical Calculations and Experimental Verification of the Antibacterial Potential of Some Monocyclic β-Lactams Containing Two Synergetic Buried Antibacterial Pharmacophore Sites

(2010) Ali Parvez et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

Studies on novel D-ring substituted steroidal pyrazolines as potential anticancer agents

(2010) Abid H. Banday et al.   STEROIDS

Towards development of selective and reversible pyrazoline based MAO-inhibitors: Synthesis, biological evaluation and docking studies

(2009) Anasuya Sahoo et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, anticonvulsant activity and 3D-QSAR study of some prop-2-eneamido and 1-acetyl-pyrazolin derivatives of aminobenzothiazole

(2009) Nikhil D. Amnerkar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Identification of antibacterial and antifungal pharmacophore sites for potent bacteria and fungi inhibition: Indolenyl sulfonamide derivatives

(2009) Zahid H. Chohan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and pharmacological evaluation of pyrazoline derivatives as new anti-inflammatory and analgesic agents

(2008) Mohammad Amir et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Pyrazoline-based mycobactin analogues as MAO-inhibitors

(2008) Venkatesan Jayaprakash et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide

(2008) I.G. Rathish et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of pyrazoline analogues with β-amino acyl group as dipeptidyl peptidase IV inhibitors

(2008) Mi Ae Jun et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives

(2008) Franco Chimenti et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and investigation of anti-inflammatory activity and gastric ulcerogenicity of novel nitric oxide-donating pyrazoline derivatives

(2008) Mai E. Shoman et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antimicrobial evaluation of 1-(benzofuran-2-yl)-4-nitro-3-arylbutan-1-ones and 3-(benzofuran-2-yl)-4,5-dihydro-5-aryl-1-[4-(aryl)-1,3-thiazol-2-yl]-1H-pyrazoles

(2008) Bakr F. Abdel-Wahab et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of novel thiazolone-based compounds containing pyrazoline moiety and evaluation of their anticancer activity

(2008) Dmytro Havrylyuk et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A novel synthesis of 1,3,5-trisubstituted pyrazoles through a spiro-pyrazoline intermediate via a tandem 1,3-dipolar cycloaddition/elimination

(2008) Sureshbabu Dadiboyena et al.   TETRAHEDRON LETTERS