Solubility and dissolution enhancement strategies: current understanding and recent trends
出版年份 2014 全文链接
标题
Solubility and dissolution enhancement strategies: current understanding and recent trends
作者
关键词
-
出版物
DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY
Volume 41, Issue 6, Pages 875-887
出版商
Informa UK Limited
发表日期
2014-10-24
DOI
10.3109/03639045.2014.971027
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- (2014) Koneti Venkata Mahesh et al. POWDER TECHNOLOGY
- Nano-extrusion: a One-Step Process for Manufacturing of Solid Nanoparticle Formulations Directly from the Liquid Phase
- (2013) Johannes Khinast et al. AAPS PHARMSCITECH
- Lattice energy calculation – A quick tool for screening of cocrystals and estimation of relative solubility. Case of flavonoids
- (2013) L.N. Kuleshova et al. CHEMICAL PHYSICS LETTERS
- Norfloxacin salts with benzenedicarboxylic acids: charge-assisted hydrogen-bonding recognition and solubility regulation
- (2013) Xian-Feng Huang et al. CRYSTENGCOMM
- Application of the combinative particle size reduction technology H 42 to produce fast dissolving glibenclamide tablets
- (2013) Jaime Salazar et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Preparation of an amorphous sodium furosemide salt improves solubility and dissolution rate and leads to a faster Tmax after oral dosing to rats
- (2013) Line Hagner Nielsen et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Spray granulation: Importance of process parameters on in vitro and in vivo behavior of dried nanosuspensions
- (2013) Carlos E. Figueroa et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Improved group contribution parameter set for the application of solubility parameters to melt extrusion
- (2013) Susann Just et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Miniaturized screening of polymers for amorphous drug stabilization (SPADS): Rapid assessment of solid dispersion systems
- (2013) Nicole Wyttenbach et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- The influence of salt formation on electrostatic and compression properties of flurbiprofen salts
- (2013) Enes Šupuk et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Stability of nanosuspensions in drug delivery
- (2013) Yancai Wang et al. JOURNAL OF CONTROLLED RELEASE
- A portable fiber-optic Raman analyzer for fast real-time screening and identifying cocrystal formation of drug-coformer via grinding process
- (2013) Hong-Liang Lin et al. MICROCHEMICAL JOURNAL
- Stability and solubility enhancement of ellagic acid in cellulose ester solid dispersions
- (2012) Bin Li et al. CARBOHYDRATE POLYMERS
- Physicochemical and Pharmacokinetic Characterization of Amorphous Solid Dispersion of Tranilast with Enhanced Solubility in Gastric Fluid and Improved Oral Bioavailability
- (2012) Satomi Onoue et al. Drug Metabolism and Pharmacokinetics
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- (2012) Elham Shoghi et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Nanocrystals: Comparison of the size reduction effectiveness of a novel combinative method with conventional top-down approaches
- (2012) Jaime Salazar et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Development of an oral solid dispersion formulation for use in low-dose metronomic chemotherapy of paclitaxel
- (2012) Johannes Moes et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Coformer selection based on degradation pathway of drugs: A case study of adefovir dipivoxil–saccharin and adefovir dipivoxil–nicotinamide cocrystals
- (2012) Yuan Gao et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- A new cocrystal and salts of itraconazole: Comparison of solid-state properties, stability and dissolution behavior
- (2012) Anna Shevchenko et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Aqueous solubility: Simple predictive methods (in silico, in vitro and bio-relevant approaches)
- (2012) David Elder et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Emerging trends in the stabilization of amorphous drugs
- (2012) Riikka Laitinen et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Drug nanocrystals in the commercial pharmaceutical development process
- (2012) Jan P. Möschwitzer INTERNATIONAL JOURNAL OF PHARMACEUTICS
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- Rational Coformer or Solvent Selection for Pharmaceutical Cocrystallization or Desolvation
- (2012) Yuriy A. Abramov et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Drug Salt Formation via Mechanochemistry: The Case Study of Vincamine
- (2012) Dritan Hasa et al. MOLECULAR PHARMACEUTICS
- Preparation and characterization of vitexin powder micronized by a supercritical antisolvent (SAS) process
- (2012) Yuangang Zu et al. POWDER TECHNOLOGY
- Improvement in physicochemical properties of ezetimibe using a crystal engineering technique
- (2012) Snehal P. Mulye et al. POWDER TECHNOLOGY
- Formation of itraconazole/L-malic acid cocrystals by gas antisolvent cocrystallization
- (2012) Courtney A. Ober et al. POWDER TECHNOLOGY
- Mechanochemistry: opportunities for new and cleaner synthesis
- (2011) Stuart L. James et al. CHEMICAL SOCIETY REVIEWS
- Physicochemical characterization and dissolution study of solid dispersions of diacerein with polyethylene glycol 6000
- (2011) Amit Kumar Aggarwal et al. DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY
- Impact of the counterion on the solubility and physicochemical properties of salts of carboxylic acid drugs
- (2011) S.E. David et al. DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY
- Effect of counterions on the properties of amorphous atorvastatin salts
- (2011) Vishal M. Sonje et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
- Counter-intuitive enhancement in the dissolution of indomethacin with the incorporation of cohesive poorly water-soluble inorganic salt additives
- (2011) Tracy Tay et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Investigation of preparation parameters of nanosuspension by top-down media milling to improve the dissolution of poorly water-soluble glyburide
- (2011) Sachin Kumar Singh et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
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- (2011) Michael Lee Branham et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
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- (2011) Mohammad Amin Mohammad et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
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- (2011) Yohei Kawabata et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
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- (2011) Shunichirou Tsutsumi et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
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- (2011) Ken K. Qian et al. JOURNAL OF PHARMACEUTICAL SCIENCES
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- (2011) Ann Newman et al. JOURNAL OF PHARMACEUTICAL SCIENCES
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- (2011) Dritan Hasa et al. PHARMACEUTICAL RESEARCH
- Cocrystal Eutectic Constants and Prediction of Solubility Behavior
- (2010) David J. Good et al. CRYSTAL GROWTH & DESIGN
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- (2010) David Good et al. CRYSTENGCOMM
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- (2010) Haibing He et al. DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY
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- (2010) Krzysztof J. Paluch et al. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
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- (2010) Satomi Onoue et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
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- (2010) Yasuhiro Miyako et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
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- (2010) Jean-Philippe Sylvestre et al. JOURNAL OF CONTROLLED RELEASE
- Hydrocortisone nanosuspensions for ophthalmic delivery: A comparative study between microfluidic nanoprecipitation and wet milling
- (2010) Hany S.M. Ali et al. JOURNAL OF CONTROLLED RELEASE
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- (2010) Gregory A. Stephenson et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Screening for pharmaceutical cocrystals using the supercritical fluid enhanced atomization process
- (2010) Luis Padrela et al. JOURNAL OF SUPERCRITICAL FLUIDS
- Formulation development of Carbamazepine–Nicotinamide co-crystals complexed with γ-cyclodextrin using supercritical fluid process
- (2010) Abhijat Shikhar et al. JOURNAL OF SUPERCRITICAL FLUIDS
- Aqueous solubility of crystalline and amorphous drugs: Challenges in measurement
- (2010) Sharad B. Murdande et al. PHARMACEUTICAL DEVELOPMENT AND TECHNOLOGY
- A biopharmaceutical classification-based Right-First-Time formulation approach to reduce human pharmacokinetic variability and project cycle time from First-In-Human to clinical Proof-Of-Concept
- (2010) M. Sherry Ku et al. PHARMACEUTICAL DEVELOPMENT AND TECHNOLOGY
- Effect of Crystal Size on the In Vitro Dissolution and Oral Absorption of Nitrendipine in Rats
- (2010) Dengning Xia et al. PHARMACEUTICAL RESEARCH
- Understanding the Behavior of Amorphous Pharmaceutical Systems during Dissolution
- (2010) David E. Alonzo et al. PHARMACEUTICAL RESEARCH
- Bottom-Up Preparation Techniques for Nanocrystals of Lipophilic Drugs
- (2010) Hans de Waard et al. PHARMACEUTICAL RESEARCH
- Solubility of Pioglitazone Hydrochloride in Aqueous Solutions of Ethanol, Propylene Glycol, and N-Methyl-2-Pyrrolidone at 298.2°K
- (2009) Shahla Soltanpour et al. AAPS PHARMSCITECH
- Water-soluble prodrugs of an Aurora kinase inhibitor
- (2009) Johan D. Oslob et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Prodrug Approaches for Enhancing the Bioavailability of Drugs with Low Solubility
- (2009) Christaâ E. Müller CHEMISTRY & BIODIVERSITY
- Understanding and Predicting the Effect of Cocrystal Components and pH on Cocrystal Solubility
- (2009) Sarah J. Bethune et al. CRYSTAL GROWTH & DESIGN
- Solubility Advantage of Pharmaceutical Cocrystals
- (2009) David J. Good et al. CRYSTAL GROWTH & DESIGN
- Synthesis and Structural Characterization of Cocrystals and Pharmaceutical Cocrystals: Mechanochemistry vs Slow Evaporation from Solution
- (2009) David R. Weyna et al. CRYSTAL GROWTH & DESIGN
- Enhancement of solubility and dissolution of Coenzyme Q10 using solid dispersion formulation
- (2009) Pushp R. Nepal et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- Supersaturating Drug Delivery Systems: The Answer to Solubility-Limited Oral Bioavailability?
- (2009) Joachim Brouwers et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Fusion processing of itraconazole solid dispersions by kinetisol® dispersing: A comparative study to hot melt extrusion
- (2009) James C. DiNunzio et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Solubility Improvement of Drugs using N-Methyl Pyrrolidone
- (2008) Ritesh Sanghvi et al. AAPS PHARMSCITECH
- Applying Hot-Stage Microscopy to Co-Crystal Screening: A Study of Nicotinamide with Seven Active Pharmaceutical Ingredients
- (2008) David J. Berry et al. CRYSTAL GROWTH & DESIGN
- Effect of the Counterion on the Solubility of Isostructural Pharmaceutical Lamotrigine Salts
- (2008) Judit Galcera et al. CRYSTAL GROWTH & DESIGN
- Cocrystals and Salts of Gabapentin: pH Dependent Cocrystal Stability and Solubility
- (2008) L. Sreenivas Reddy et al. CRYSTAL GROWTH & DESIGN
- Screening strategies based on solubility and solution composition generate pharmaceutically acceptable cocrystals of carbamazepine
- (2008) Scott L. Childs et al. CRYSTENGCOMM
- Effect of polymer type on the dissolution profile of amorphous solid dispersions containing felodipine
- (2008) Hajime Konno et al. EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
- Enhancement of oral bioavailability of an HIV-attachment inhibitor by nanosizing and amorphous formulation approaches
- (2008) Michael G. Fakes et al. INTERNATIONAL JOURNAL OF PHARMACEUTICS
- A novel bottom–up process to produce drug nanocrystals: Controlled crystallization during freeze-drying
- (2008) H. de Waard et al. JOURNAL OF CONTROLLED RELEASE
- Preparation and Characterization of Salt Forms of Enalapril
- (2008) Lokesh Kumar et al. PHARMACEUTICAL DEVELOPMENT AND TECHNOLOGY
- Dissolution Improvement and the Mechanism of the Improvement from Cocrystallization of Poorly Water-soluble Compounds
- (2008) Koji Shiraki et al. PHARMACEUTICAL RESEARCH
- Particle design of poorly water-soluble drug substances using supercritical fluid technologies
- (2007) Takehiko Yasuji et al. ADVANCED DRUG DELIVERY REVIEWS
- Engineering of Pharmaceutical Materials: An Industrial Perspective
- (2007) Kwok Chow et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Supercritical fluid-micronized ipratropium bromide for pulmonary drug delivery
- (2007) Yong Ho Kim et al. POWDER TECHNOLOGY
- Preparation of griseofulvin microparticles by supercritical fluid expansion depressurization process
- (2007) Li Zhiyi et al. POWDER TECHNOLOGY
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