Neuropeptides and Neuropeptide Receptors: Drug Targets, and Peptide and Non-Peptide Ligands: a Tribute to Prof.Dieter Seebach
出版年份 2012 全文链接
标题
Neuropeptides and Neuropeptide Receptors: Drug Targets, and Peptide and Non-Peptide Ligands: a Tribute to Prof.Dieter Seebach
作者
关键词
-
出版物
CHEMISTRY & BIODIVERSITY
Volume 9, Issue 11, Pages 2367-2387
出版商
Wiley
发表日期
2012-11-19
DOI
10.1002/cbdv.201200288
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- Orexin Receptor Antagonism, a New Sleep-Enabling Paradigm: A Proof-of-Concept Clinical Trial
- (2012) P Hoever et al. CLINICAL PHARMACOLOGY & THERAPEUTICS
- Orexin receptor antagonism: an ascending multiple-dose study with almorexant
- (2012) Petra Hoever et al. JOURNAL OF PSYCHOPHARMACOLOGY
- Structure of the δ-opioid receptor bound to naltrindole
- (2012) Sébastien Granier et al. NATURE
- Structure of the human κ-opioid receptor in complex with JDTic
- (2012) Huixian Wu et al. NATURE
- Structure of the nociceptin/orphanin FQ receptor in complex with a peptide mimetic
- (2012) Aaron A. Thompson et al. NATURE
- Crystal structure of the µ-opioid receptor bound to a morphinan antagonist
- (2012) Aashish Manglik et al. NATURE
- Structure and dynamics of the M3 muscarinic acetylcholine receptor
- (2012) Andrew C. Kruse et al. NATURE
- Apo-Ghrelin Receptor Forms Heteromers with DRD2 in Hypothalamic Neurons and Is Essential for Anorexigenic Effects of DRD2 Agonism
- (2012) Andras Kern et al. NEURON
- Crystal Structure of a Lipid G Protein-Coupled Receptor
- (2012) M. A. Hanson et al. SCIENCE
- Structure-based drug screening for G-protein-coupled receptors
- (2012) Brian K. Shoichet et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- New insights from structural biology into the druggability of G protein-coupled receptors
- (2012) Jonathan S. Mason et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- Nanobody stabilization of G protein-coupled receptor conformational states
- (2011) Jan Steyaert et al. CURRENT OPINION IN STRUCTURAL BIOLOGY
- Promotion of Sleep by Suvorexant—A Novel Dual Orexin Receptor Antagonist
- (2011) Christopher J. Winrow et al. JOURNAL OF NEUROGENETICS
- Conformational Dynamics of Single G Protein-Coupled Receptors in Solution
- (2011) Samuel Bockenhauer et al. JOURNAL OF PHYSICAL CHEMISTRY B
- Phase I studies on the safety, tolerability, pharmacokinetics and pharmacodynamics of SB-649868, a novel dual orexin receptor antagonist
- (2011) Paolo Bettica et al. JOURNAL OF PSYCHOPHARMACOLOGY
- Reaction Development and Mechanistic Study of a Ruthenium Catalyzed Intramolecular Asymmetric Reductive Amination en Route to the Dual Orexin Inhibitor Suvorexant (MK-4305)
- (2011) Neil A. Strotman et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- The truncated ghrelin receptor polypeptide (GHS-R1b) is localized in the endoplasmic reticulum where it forms heterodimers with ghrelin receptors (GHS-R1a) to attenuate their cell surface expression
- (2011) Kevin B.S. Chow et al. MOLECULAR AND CELLULAR ENDOCRINOLOGY
- Conformational changes in the G protein Gs induced by the β2 adrenergic receptor
- (2011) Ka Young Chung et al. NATURE
- Crystal structure of the β2 adrenergic receptor–Gs protein complex
- (2011) Søren G. F. Rasmussen et al. NATURE
- Structural insights into adrenergic receptor function and pharmacology
- (2011) Brian K. Kobilka TRENDS IN PHARMACOLOGICAL SCIENCES
- Reaction of Fe3(CO)12 with octreotide—chemical, electrochemical and biological investigations
- (2010) Ulf-Peter Apfel et al. DALTON TRANSACTIONS
- Anticonvulsant effects and behavioural outcomes of rAAV serotype 1 vector-mediated neuropeptide Y overexpression in rat hippocampus
- (2010) F Noe et al. GENE THERAPY
- Neuropeptide receptor positive allosteric modulation in epilepsy: Galanin modulation revealed
- (2010) D. Hoyer PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- GalR2-positive allosteric modulator exhibits anticonvulsant effects in animal models
- (2010) X. Lu et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- RAMP-ing up Class-B GPCR ECD Structural Coverage
- (2010) Fai Y. Siu et al. STRUCTURE
- Crystal Structure of the Ectodomain Complex of the CGRP Receptor, a Class-B GPCR, Reveals the Site of Drug Antagonism
- (2010) Ernst ter Haar et al. STRUCTURE
- Non-peptidic antagonists of the CGRP receptor, BIBN4096BS and MK-0974, interact with the calcitonin receptor-like receptor via methionine-42 and RAMP1 via tryptophan-74
- (2009) Philip S. Miller et al. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
- Novel CGRP receptor antagonists through a design strategy of target simplification with addition of molecular flexibility
- (2009) Michael R. Wood et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Almorexant
- (2009) R.T. Owen et al. DRUGS OF THE FUTURE
- NMR-Solution Structures and Affinities for the Human Somatostatin G-Protein-Coupled Receptors hsst1â5 of CF3 Derivatives of Sandostatin® (Octreotide)
- (2009) Dieter Seebach et al. HELVETICA CHIMICA ACTA
- The structure and function of G-protein-coupled receptors
- (2009) Daniel M. Rosenbaum et al. NATURE
- Developing novel antiepileptic drugs: Characterization of NAX 5055, a systemically-active galanin analog, in epilepsy models
- (2009) H. Steve White et al. Neurotherapeutics
- The role of CGRP in the pathophysiology of migraine and efficacy of CGRP receptor antagonists as acute antimigraine drugs
- (2009) Carlos M. Villalón et al. PHARMACOLOGY & THERAPEUTICS
- β-Peptidic Peptidomimetics
- (2008) Dieter Seebach et al. ACCOUNTS OF CHEMICAL RESEARCH
- Molecular biology of 5-HT receptors
- (2008) Jason Hannon et al. BEHAVIOURAL BRAIN RESEARCH
- Neuropeptide Y gene therapy decreases chronic spontaneous seizures in a rat model of temporal lobe epilepsy
- (2008) Francesco Noè et al. BRAIN
- Increased exploratory activity of APP23 mice in a novel environment is reversed by siRNA
- (2008) Yann Senechal et al. BRAIN RESEARCH
- The Enantiomer of Octreotate Binds to All Five Somatostatin Receptors with Almost Equal Micromolar Affinity - A Comparison withSANDOSTATIN®
- (2008) James Gardiner et al. CHEMISTRY & BIODIVERSITY
- New Open-Chain and Cyclic Tetrapeptides, Consisting ofα-,β2-, andβ3-Amino-Acid Residues, as Somatostatin Mimics - A Survey
- (2008) Dieter Seebach et al. HELVETICA CHIMICA ACTA
- Pharmacological profile of somatostatin and cortistatin receptors
- (2007) Sandra Siehler et al. MOLECULAR AND CELLULAR ENDOCRINOLOGY
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreFind the ideal target journal for your manuscript
Explore over 38,000 international journals covering a vast array of academic fields.
Search