Aminoboronic acids and esters: from synthetic challenges to the discovery of unique classes of enzyme inhibitors
出版年份 2011 全文链接
标题
Aminoboronic acids and esters: from synthetic challenges to the discovery of unique classes of enzyme inhibitors
作者
关键词
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出版物
CHEMICAL SOCIETY REVIEWS
Volume 40, Issue 7, Pages 3895
出版商
Royal Society of Chemistry (RSC)
发表日期
2011-03-23
DOI
10.1039/c0cs00154f
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- Synthesis and carbohydrate binding studies of fluorescent α-amidoboronic acids and the corresponding bisboronic acids
- (2010) Shan Jin et al. BIOORGANIC & MEDICINAL CHEMISTRY
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- (2010) Xianfeng Li et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Structure–activity relationship of boronic acid derivatives of tyropeptin: Proteasome inhibitors
- (2010) Takumi Watanabe et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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- (2010) Xianfeng Li et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- 4,7-Dichloro benzothien-2-yl sulfonylaminomethyl boronic acid: First boronic acid-derived beta-lactamase inhibitor with class A, C, and D activity
- (2010) Qiang Tan et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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- (2010) E. Kupperman et al. CANCER RESEARCH
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- (2010) Valery M. Dembitsky et al. CHEMICAL REVIEWS
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- (2010) S. M. Drawz et al. CLINICAL MICROBIOLOGY REVIEWS
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- (2010) E. Genin et al. CURRENT TOPICS IN MEDICINAL CHEMISTRY
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- (2010) Lawrence R. Dick et al. DRUG DISCOVERY TODAY
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- (2010) Nuruddeen D. Lewis et al. JOURNAL OF IMMUNOLOGY
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- (2010) Kenneth Knott et al. ORGANIC & BIOMOLECULAR CHEMISTRY
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- (2010) Paul C. Trippier et al. MedChemComm
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- (2009) Irene Georgiou et al. ACCOUNTS OF CHEMICAL RESEARCH
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- (2009) Sarah M. Drawz et al. BIOCHEMISTRY
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- (2009) Aaron M. LeBeau et al. BIOORGANIC & MEDICINAL CHEMISTRY
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- (2009) Amogh Boloor et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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- (2009) Eric Sanchez et al. BRITISH JOURNAL OF HAEMATOLOGY
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- (2009) Heiko Zettl et al. ChemMedChem
- Not boring at all. Boron is the new carbon in the quest for novel drug candidates
- (2009) Philip Hunter EMBO REPORTS
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- (2009) Stephen J Baker et al. Future Medicinal Chemistry
- Arginase inhibition restores NOS coupling and reverses endothelial dysfunction and vascular stiffness in old rats
- (2009) Jae Hyung Kim et al. JOURNAL OF APPLIED PHYSIOLOGY
- Design, Synthesis, Biological Evaluation, and Structure−Activity Relationship (SAR) Discussion of Dipeptidyl Boronate Proteasome Inhibitors, Part I: Comprehensive Understanding of the SAR of α-Amino Acid Boronates
- (2009) Yongqiang Zhu et al. JOURNAL OF MEDICINAL CHEMISTRY
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- (2009) Nobuaki Suzuki et al. JOURNAL OF MEDICINAL CHEMISTRY
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- (2008) Harm Maarsingh et al. AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE
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- (2008) George W. Kabalka et al. APPLIED ORGANOMETALLIC CHEMISTRY
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- (2008) Aaron M. LeBeau et al. CHEMISTRY & BIOLOGY
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- (2007) Donald S. Matteson MEDICINAL RESEARCH REVIEWS
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