Linear Aliphatic Dialkynes as Alternative Linkers for Double-Click Stapling of p53-Derived Peptides
出版年份 2014 全文链接
标题
Linear Aliphatic Dialkynes as Alternative Linkers for Double-Click Stapling of p53-Derived Peptides
作者
关键词
-
出版物
CHEMBIOCHEM
Volume 15, Issue 18, Pages 2680-2683
出版商
Wiley
发表日期
2014-10-29
DOI
10.1002/cbic.201402374
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- Comparative α-Helicity of Cyclic Pentapeptides in Water
- (2014) Aline D. de Araujo et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Investigating peptide sequence variations for ‘double-click’ stapled p53 peptides
- (2014) Yu Heng Lau et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Functionalised staple linkages for modulating the cellular activity of stapled peptides
- (2014) Yu Heng Lau et al. Chemical Science
- Distinct BimBH3 (BimSAHB) Stapled Peptides for Structural and Cellular Studies
- (2013) Greg H. Bird et al. ACS Chemical Biology
- Stabilisation of a shortα-helical VIP fragment by side chain to side chain cyclisation: a comparison of common cyclisation motifs by circular dichroism
- (2013) Lukasz Frankiewicz et al. JOURNAL OF PEPTIDE SCIENCE
- A Perfluoroaryl-Cysteine SNAr Chemistry Approach to Unprotected Peptide Stapling
- (2013) Alexander M. Spokoyny et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Inhibition of α-helix-mediated protein–protein interactions using designed molecules
- (2013) Valeria Azzarito et al. Nature Chemistry
- Stapled α−helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy
- (2013) Yong S. Chang et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Stapled Peptides with Improved Potency and Specificity That Activate p53
- (2012) Christopher J. Brown et al. ACS Chemical Biology
- Development of α-Helical Calpain Probes by Mimicking a Natural Protein–Protein Interaction
- (2012) Hyunil Jo et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Synthesis of cell-permeable stapled peptide dual inhibitors of the p53-Mdm2/Mdmx interactions via photoinduced cycloaddition
- (2011) Michael M. Madden et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Peptides and Proteins as a Continuing Exciting Source of Inspiration for Peptidomimetics
- (2011) Rob M. J. Liskamp et al. CHEMBIOCHEM
- Achieving cell penetration with distance-matching cysteine cross-linkers: a facile route to cell-permeable peptide dual inhibitors of Mdm2/Mdmx
- (2011) Avinash Muppidi et al. CHEMICAL COMMUNICATIONS
- 1,2,3-Triazoles in Peptidomimetic Chemistry
- (2011) Daniel Sejer Pedersen et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Design of Triazole-Stapled BCL9 α-Helical Peptides to Target the β-Catenin/B-Cell CLL/lymphoma 9 (BCL9) Protein–Protein Interaction
- (2011) Steven A. Kawamoto et al. JOURNAL OF MEDICINAL CHEMISTRY
- Structure of the Stapled p53 Peptide Bound to Mdm2
- (2011) Sohee Baek et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Design and Structure of Stapled Peptides Binding to Estrogen Receptors
- (2011) Chris Phillips et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- On Resin Side-Chain Cyclization of Complex Peptides Using CuAAC
- (2011) Sampat Ingale et al. ORGANIC LETTERS
- Stapled peptides in the p53 pathway: Computer simulations reveal novel interactions of the staples with the target protein
- (2010) Thomas Leonard Joseph et al. CELL CYCLE
- The MCL-1 BH3 helix is an exclusive MCL-1 inhibitor and apoptosis sensitizer
- (2010) Michelle L Stewart et al. Nature Chemical Biology
- Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency
- (2010) R. S. Harrison et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Reactivation of p53: from peptides to small molecules
- (2010) Christopher J. Brown et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- Facile synthesis of stapled, structurally reinforced peptide helices via a photoinduced intramolecular 1,3-dipolar cycloaddition reaction
- (2009) Michael M. Madden et al. CHEMICAL COMMUNICATIONS
- Peptidomimetics - A Versatile Route to Biologically Active Compounds
- (2009) Andreas Grauer et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- CuI-Catalyzed AzideâAlkyne Intramoleculari-to-(i+4) Side-Chain-to-Side-Chain Cyclization Promotes the Formation of Helix-Like Secondary Structures
- (2009) Mario Scrima et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Photocontrollable Peptide-Based Switches Target the Anti-Apoptotic Protein Bcl-xL
- (2008) Sabine Kneissl et al. CHEMBIOCHEM
- Development of a Series of Cross-Linking Agents that Effectively Stabilize α-Helical Structures in Various Short Peptides
- (2007) Kazuhisa Fujimoto et al. CHEMISTRY-A EUROPEAN JOURNAL
Create your own webinar
Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.
Create NowAsk a Question. Answer a Question.
Quickly pose questions to the entire community. Debate answers and get clarity on the most important issues facing researchers.
Get Started