1,2,3-Triazoles in Peptidomimetic Chemistry

Cyclative Cleavage through Dipolar Cycloaddition: Polymer-Bound Azidopeptidylphosphoranes Deliver Locked cis-Triazolylcyclopeptides as Privileged Protein Binders

(2010) Ahsanullah et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cyclopeptide Smac mimetics as antagonists of IAP proteins

(2010) Haiying Sun et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

1,2,3-Triazolyl amino acids as AMPA receptor ligands

(2010) N.J. Stanley et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

In situ click chemistry: probing the binding landscapes of biological molecules

(2010) Sreeman K. Mamidyala et al.   CHEMICAL SOCIETY REVIEWS

Tricks with clicks: modification of peptidomimetic oligomers via copper-catalyzed azide-alkyne [3 + 2] cycloaddition

(2010) Justin M. Holub et al.   CHEMICAL SOCIETY REVIEWS

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

Development of Stable Phosphohistidine Analogues

(2010) Jung-Min Kee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bioorthogonal Chemical Reporters for Monitoring Protein Acetylation

(2010) Yu-Ying Yang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rapid Cu-Free Click Chemistry with Readily Synthesized Biarylazacyclooctynones

(2010) John C. Jewett et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-free click chemistry in living animals

(2010) P. V. Chang et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Evaluation of triazolamers as active site inhibitors of HIV-1 protease

(2009) Andrea L. Jochim et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Peptidomimetics - A Versatile Route to Biologically Active Compounds

(2009) Andreas Grauer et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

CuI-Catalyzed Azide–Alkyne Intramoleculari-to-(i+4) Side-Chain-to-Side-Chain Cyclization Promotes the Formation of Helix-Like Secondary Structures

(2009) Mario Scrima et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Peptide Cyclization and Cyclodimerization by CuI-Mediated Azide−Alkyne Cycloaddition

(2009) Reshma Jagasia et al.   JOURNAL OF ORGANIC CHEMISTRY

Microwave-Assisted Intramolecular Huisgen Cycloaddition of Azido Alkynes Derived from α-Amino Acids

(2009) Evita Balducci et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Azide-Alkyne Fragments for “Click” Chemical Applications. Part 2. Formation of Oligomers from Orthogonally Protected Chiral Trialkylsilylhomopropargyl Azides and Homopropargyl Alcohols

(2009) Oliver D. Montagnat et al.   JOURNAL OF ORGANIC CHEMISTRY

Side chain-to-side chain cyclization by click reaction

(2009) Alexandra Le Chevalier Isaad et al.   JOURNAL OF PEPTIDE SCIENCE

Genetic Encoding and Labeling of Aliphatic Azides and Alkynes in Recombinant Proteinsviaa Pyrrolysyl-tRNA Synthetase/tRNACUAPair and Click Chemistry

(2009) Duy P. Nguyen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Microwave-assisted click polymerization for the synthesis of Aβ(16–22) cyclic oligomers and their self-assembly into polymorphous aggregates

(2009) Ronald C. Elgersma et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Structure–function relationships in peptoids: Recent advances toward deciphering the structural requirements for biological function

(2009) Sarah A. Fowler et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Novel triazolopeptides: chirospecific synthesis and conformational studies of proline derived analogs

(2009) Andreas Paul et al.   TETRAHEDRON

Unnatural Amino Acid Incorporation into Virus-Like Particles

(2008) Erica Strable et al.   BIOCONJUGATE CHEMISTRY

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Backbone Amide Linker Strategy for the Synthesis of 1,4-Triazole-Containing Cyclic Tetra- and Pentapeptides

(2008) Jasper Springer et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Structural Determinants for Affinity Enhancement of a Dual Antagonist Peptide Entry Inhibitor of Human Immunodeficiency Virus Type-1

(2008) Hosahudya Gopi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Conformational Analysis of a Cyclic Peptide Obtained viaitoi+4 Intramolecular Side-Chain to Side-Chain Azide−Alkyne 1,3-Dipolar Cycloaddition

(2008) Sonia Cantel et al.   JOURNAL OF ORGANIC CHEMISTRY

Ribosomal Synthesis of Bicyclic Peptides via Two Orthogonal Inter-Side-Chain Reactions

(2008) Yusuke Sako et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Design and synthesis of cyclo[-Arg-Gly-Asp-Ψ(triazole)-Gly-Xaa-] peptide analogues by click chemistry

(2008) Yaqin Liu et al.   TETRAHEDRON

Design of azidoproline containing gluten peptides to suppress CD4+ T-cell responses associated with Celiac disease

(2007) Varsha V. Kapoerchan et al.   BIOORGANIC & MEDICINAL CHEMISTRY