Ligand-Enabled Triple CH Activation Reactions: One-Pot Synthesis of Diverse 4-Aryl-2-quinolinones from Propionamides

Aerobic Double Dehydrogenative Cross Coupling between Cyclic Saturated Ketones and Simple Arenes

(2014) Nicolas Gigant et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ligand-enabled cross-coupling of C(sp3)–H bonds with arylboron reagents via Pd(II)/Pd(0) catalysis

(2014) Kelvin S. L. Chan et al.   Nature Chemistry

Ligand-Controlled C(sp3)-H Arylation and Olefination in Synthesis of Unnatural Chiral  -Amino Acids

(2014) J. He et al.   SCIENCE

Palladium-Catalyzed Through-Space C(sp3)H and C(sp2)H Bond Activation by 1,4-Palladium Migration: Efficient Synthesis of [3,4]-Fused Oxindoles

(2013) Tiffany Piou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Oxidative C–H amination reactions

(2013) Marie-Laure Louillat et al.   CHEMICAL SOCIETY REVIEWS

Catalytic Direct β-Arylation of Simple Ketones with Aryl Iodides

(2013) Zhongxing Huang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Aerobic Dehydrogenation of Cyclohexanone to Cyclohexenone Catalyzed by Pd(DMSO)2(TFA)2: Evidence for Ligand-Controlled Chemoselectivity

(2013) Tianning Diao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium(0)-Catalyzed Alkynylation of C(sp3)–H Bonds

(2013) Jian He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 2(1H)-Quinolinones via Pd-Catalyzed Oxidative Cyclocarbonylation of 2-Vinylanilines

(2013) Jamie Ferguson et al.   ORGANIC LETTERS

Activation of a C(sp3)H Bond by a Transient σ-Alkylpalladium(II) Complex: Synthesis of Spirooxindoles Through a Palladium-Catalyzed Domino Carbopalladation/C(sp3)C(sp3) Bond-Forming Process

(2012) Tiffany Piou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Tandem-type Pd(ii)-catalyzed oxidative Heck reaction/intramolecular C–H amidation sequence: a novel route to 4-aryl-2-quinolinones

(2012) Kiyofumi Inamoto et al.   CHEMICAL COMMUNICATIONS

4-Aryl-2-quinolones from 3,3-Diarylacrylamides through Intramolecular Copper-Catalyzed C–H Functionalization/C–N Bond Formation

(2012) Roberta Berrino et al.   JOURNAL OF ORGANIC CHEMISTRY

Ligand-Enabled Methylene C(sp3)–H Bond Activation with a Pd(II) Catalyst

(2012) Masayuki Wasa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Spirocyclization by Palladium-Catalyzed Domino Heck–Direct C–H Arylation Reactions: Synthesis of Spirodihydroquinolin-2-ones

(2012) Tiffany Piou et al.   ORGANIC LETTERS

Diastereoselective synthesis of 3,3-disubstituted oxindoles from atropisomeric N-aryl oxindole derivatives

(2012) Atsuo Nakazaki et al.   TETRAHEDRON LETTERS

Palladium-Catalyzed Enantioselective Intramolecular Hydroarylation of Alkynes To Form Axially Chiral 4-Aryl 2-Quinolinones

(2011) Tetsuro Shibuya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-Pot Formation of CC and CN Bonds through Palladium-Catalyzed Dual CH Activation: Synthesis of Phenanthridinones

(2011) Guan-Wu Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Phenanthridinones from N-Methoxybenzamides and Arenes by Multiple Palladium-Catalyzed CH Activation Steps at Room Temperature

(2011) Jaganathan Karthikeyan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Cyclic Enones via Direct Palladium-Catalyzed Aerobic Dehydrogenation of Ketones

(2011) Tianning Diao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct aerobic α,β-dehydrogenation of aldehydes and ketones with a Pd(TFA)2/4,5-diazafluorenone catalyst

(2011) Tianning Diao et al.   Chemical Science

General palladium-catalyzed aerobic dehydrogenation to generate double bonds

(2011) Weiming Gao et al.   Chemical Science

Second Generation Analogues of the Cancer Drug Clinical Candidate Tipifarnib for Anti-Chagas Disease Drug Discovery

(2010) James M. Kraus et al.   JOURNAL OF MEDICINAL CHEMISTRY

Palladium-Catalyzed Intramolecular Amidation of C(sp2)−H Bonds: Synthesis of 4-Aryl-2-quinolinones

(2010) Kiyofumi Inamoto et al.   JOURNAL OF ORGANIC CHEMISTRY

Rational Modification of a Candidate Cancer Drug for Use Against Chagas Disease

(2009) James M. Kraus et al.   JOURNAL OF MEDICINAL CHEMISTRY

Pd(0)/PR3-Catalyzed Intermolecular Arylation of sp3C−H Bonds

(2009) Masayuki Wasa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diverse Functionalization of Corannulene: Easy Access to Pentagonal Superstructure

(2009) Doron Pappo et al.   ORGANIC LETTERS

Synthesis and evaluation of novel 3,4,6-substituted 2-quinolones as FMS kinase inhibitors

(2008) Mark J. Wall et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and in vitro anti-hepatitis B virus activities of 4-aryl-6-chloro-quinolin-2-one and 5-aryl-7-chloro-1,4-benzodiazepine derivatives

(2008) Pi Cheng et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of β-, γ-, and δ-Lactams via Pd(II)-Catalyzed C−H Activation Reactions

(2008) Masayuki Wasa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis and biological activity of quinolinone and dihydroquinolinone p38 MAP kinase inhibitors

(2006) Meng-Hsin Chen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS