Catalytic Asymmetric Synthesis of [2,3]-Fused Indoline Heterocycles through Inverse-Electron-Demand Aza-Diels-Alder Reaction of Indoles with Azoalkenes

Copper-Catalyzed Enantioselective Inverse Electron-Demand Hetero-Diels-Alder Reactions of Diazadienes with Enol Ethers: Efficient Synthesis of Chiral Pyridazines

(2013) Shuang Gao et al.   ADVANCED SYNTHESIS & CATALYSIS

Complex Bioactive Alkaloid-Type Polycycles through Efficient Catalytic Asymmetric Multicomponent Aza-Diels-Alder Reaction of Indoles with Oxetane as Directing Group

(2013) Zhilong Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric 1,3-Dipolar Cycloaddition of Two Different Ylides: Facile Access to Chiral 1,2,4-Triazinane Frameworks

(2013) Min-Chao Tong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent Developments in Catalytic Asymmetric Inverse-Electron-Demand Diels–Alder Reaction

(2013) Xianxing Jiang et al.   CHEMICAL REVIEWS

Copper-Catalyzed Highly Enantioselective Cyclopentannulation of Indoles with Donor–Acceptor Cyclopropanes

(2013) Hu Xiong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bifunctional Organocatalytic Strategy for Inverse-Electron-Demand Diels-Alder Reactions: Highly Efficient In Situ Substrate Generation and Activation to Construct Azaspirocyclic Skeletons

(2012) Xianxing Jiang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

FeCl3-Mediated Friedel-Crafts Hydroarylation with ElectrophilicN-Acetyl Indoles for the Synthesis of Benzofuroindolines

(2012) Rodolphe Beaud et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Dearomatization Reactions

(2012) Chun-Xiang Zhuo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Synthesis of Dihydropyrazoles by Formal [4+1] Cycloaddition of in Situ-Derived Azoalkenes and Sulfur Ylides

(2012) Jia-Rong Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalyzed Enantioselective Formal [4 + 2] Cycloaddition of 2,3-Disubstituted Indole and Methyl Vinyl Ketone

(2012) Quan Cai et al.   ORGANIC LETTERS

Enantioselective Gold-Catalyzed Synthesis of Polycyclic Indolines

(2012) Gianpiero Cera et al.   ORGANIC LETTERS

Asymmetric Diels–Alder reaction of β,β-disubstituted enals and chromone-fused dienes: construction of collections with high molecular complexity and skeletal diversity

(2012) Jun-Long Li et al.   Chemical Science

A Novel Assembly of Substituted Pyrroles by Acid-Catalyzed Sequential Three-Component Reaction of Amines, Alkynoates, and 1,2-Diaza-1,3-dienes

(2011) Orazio A. Attanasi et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Michael/Mannich Polycyclization Cascade of Indolyl Enones Catalyzed by Quinine-Derived Primary Amines

(2011) Quan Cai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Exploiting the Electrophilic Properties of Indole Intermediates: New Options in Designing Asymmetric Reactions

(2011) Charles C. J. Loh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct Asymmetric Hydrosilylation of Indoles: Combined Lewis Base and Brønsted Acid Activation

(2011) You-Cai Xiao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalyzed Enantioselective Fluorocyclizations

(2011) Oscar Lozano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Cycloaddition of β,γ-Unsaturated α-Ketoesters with Electron-Rich Alkenes Catalyzed by a Chiral Er(OTf)3/N,N′-Dioxide Complex: Highly Enantioselective Synthesis of 3,4-Dihydro-2 H-pyrans

(2011) Yin Zhu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Chiral Phosphoric Acid-Catalyzed Enantioselective Three-Component Povarov Reaction Using Enecarbamates as Dienophiles: Highly Diastereo- and Enantioselective Synthesis of Substituted 4-Aminotetrahydroquinolines

(2011) Guillaume Dagousset et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Efficient Hydrogen-Bonding Catalysis of the Diels–Alder Reaction of 3-Vinylindoles and Methyleneindolinones Provides Carbazolespirooxindole Skeletons

(2011) Bin Tan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxaziridine-Mediated Oxyamination of Indoles: An Approach to 3-Aminoindoles and Enantiomerically Enriched 3-Aminopyrroloindolines

(2010) Tamas Benkovics et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Synthesis of Pyrroloindolines by a Formal [3 + 2] Cycloaddition Reaction

(2010) Lindsay M. Repka et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cultivating the Passion to Build Heterocycles from 1,2-Diaza-1,3-dienes: the Force of Imagination

(2009) Orazio A. Attanasi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Asymmetric C2−C3 Cyclopentannulation of the Indole Ring

(2009) José Barluenga et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium-Catalyzed [3 + 2] Annulation of Indoles

(2009) Yajing Lian et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper(II)/Copper(I)-Catalyzed Aza-Michael Addition/Click Reaction of in Situ Generated α-Azidohydrazones: Synthesis of Novel Pyrazolone−Triazole Framework

(2009) Orazio A. Attanasi et al.   ORGANIC LETTERS

Au-Containing All-Carbon 1,4-Dipoles:  Generation and [4 + 2] Annulation in the Formation of Carbo-/Heterocycles

(2008) Guozhu Zhang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Flexible Protocol for the Chemo- and Regioselective Building of Pyrroles and Pyrazoles by Reactions of Danishefsky’s Dienes with 1,2-Diaza-1,3-butadienes

(2008) Orazio A. Attanasi et al.   ORGANIC LETTERS