A Conformationally Frozen Peptoid Boosts CXCR4 Affinity and Anti-HIV Activity

Synthesis of N-methylated cyclic peptides

(2012) Jayanta Chatterjee et al.   Nature Protocols

PET Imaging of CXCR4 Receptors in Cancer by a New Optimized Ligand

(2011) Oliver Demmer et al.   ChemMedChem

Drug Discovery Research Targeting the CXC Chemokine Receptor 4 (CXCR4)

(2011) Won-Tak Choi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Design, Synthesis, and Functionalization of Dimeric Peptides Targeting Chemokine Receptor CXCR4

(2011) Oliver Demmer et al.   JOURNAL OF MEDICINAL CHEMISTRY

PET of CXCR4 Expression by a 68Ga-Labeled Highly Specific Targeted Contrast Agent

(2011) E. Gourni et al.   JOURNAL OF NUCLEAR MEDICINE

EASY-HIT: HIV Full-Replication Technology for Broad Discovery of Multiple Classes of HIV Inhibitors

(2010) S. Kremb et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Structures of the CXCR4 Chemokine GPCR with Small-Molecule and Cyclic Peptide Antagonists

(2010) B. Wu et al.   SCIENCE

Coreceptors and HIV-1 Pathogenesis

(2010) Paul R. Gorry et al.   Current HIV/AIDS Reports

The AMD3100 story: The path to the discovery of a stem cell mobilizer (Mozobil)

(2009) Erik De Clercq   BIOCHEMICAL PHARMACOLOGY

Synthetic therapeutic peptides: science and market

(2009) Patrick Vlieghe et al.   DRUG DISCOVERY TODAY

Mobilization of hematopoietic stem cells: state of the art

(2008) Jean-Pierre Levesque et al.   Current Opinion in Organ Transplantation

Introduction of Functional Groups into Peptides viaN-Alkylation

(2008) O. Demmer et al.   ORGANIC LETTERS