A general and convenient method for the synthesis of 2,4-dinitrobenzyl ketones. Almost unlimited access to 2-substituted 6-nitroindoles from 2,4-dinitrotoluene and aldehydes

A copper-catalyzed tandem reaction for the construction of coumarin fused 9H-pyrrolo[1,2-a]indoles

(2017) Shao-Jing Jin et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Gold(i)-catalyzed synthesis of 2-substituted indoles from 2-alkynylnitroarenes with diboron as reductant

(2017) Wenqiang Fu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Concise synthesis of carbazole-1,4-quinones and evaluation of their antiproliferative activity against HCT-116 and HL-60 cells

(2016) Takashi Nishiyama et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Application of nucleophilic substitution of hydrogen in nitroarenes to the chemistry of indoles

(2015) Mieczysław Mąkosza et al.   Chemistry of Heterocyclic Compounds

Amino derivatives of indolone-N-oxide: Preparation and antiplasmodial properties

(2014) Ennaji Najahi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Robust, Well-Defined Homogeneous Silver(I) Catalyst for Mild Intramolecular Hydroamination of 2-Ethynylanilines Leading to Indoles

(2014) James McNulty et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

The PdCl2-catalyzed sequential heterocyclization/Michael addition cascade in the synthesis of 2,3-disubstituted indoles

(2013) Donala Janreddy et al.   TETRAHEDRON

Chemoselective N-Acylation of Indoles and Oxazolidinones with Carbonylazoles

(2012) Stephen T. Heller et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 3-Carboxylated Indoles through a Tandem Process Involving Cyclization of 2-Ethynylanilines Followed by CO2 Fixation in the Absence of Transition Metal Catalysts

(2012) Kiyofumi Inamoto et al.   ORGANIC LETTERS

Ready synthesis of free N-H 2-arylindoles via the copper-catalyzed amination of 2-bromo-arylacetylenes with aqueous ammonia and sequential intramolecular cyclization

(2011) Huifeng Wang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition-Metal-Free Formal Sonogashira Coupling and α-Carbonyl Arylation Reactions

(2010) Birgit Prüger et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Combined Experimental and Density Functional Theory Study on the Pd-Mediated Cycloisomerization of o-Alkynylnitrobenzenes - Synthesis of Isatogens and Their Evaluation as Modulators of ROS-Mediated Cell Death

(2010) Chepuri V. Ramana et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Iron-Catalyzed Regio- and Stereoselective Substitution of γ,δ-Epoxy-α,β-unsaturated Esters and Amides with Grignard Reagents

(2010) Takeshi Hata et al.   ORGANIC LETTERS

Cupric Halide-Mediated Intramolecular Halocyclization of N-Electron-Withdrawing Group-Substituted 2-Alkynylanilines for the Synthesis of 3-Haloindoles

(2009) Zengming Shen et al.   ADVANCED SYNTHESIS & CATALYSIS

One-Pot Synthesis of Indoles and Aniline Derivatives from Nitroarenes under Hydrogenation Condition with Supported Gold Nanoparticles

(2009) Yoshihiro Yamane et al.   ORGANIC LETTERS

Palladium-Catalyzed Direct Arylation of (Hetero)Arenes with Aryl Boronic Acids

(2008) Shang-Dong Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Aplicyanins A–F, new cytotoxic bromoindole derivatives from the marine tunicate Aplidium cyaneum

(2008) Fernando Reyes et al.   TETRAHEDRON

Indium-HI-mediated one-pot reaction of 1-(2-arylethynyl)-2-nitroarenes to 2-arylindoles

(2008) Ji Sook Kim et al.   TETRAHEDRON LETTERS

Palladium-Catalyzed Aryl Amination–Heck Cyclization Cascade: A One-Flask Approach to 3-Substituted Indoles

(2007) Thomas Jensen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION