Application of nucleophilic substitution of hydrogen in nitroarenes to the chemistry of indoles

Indole synthesis through transition metal-catalyzed C–H activation

(2015) Tenglong Guo et al.   TETRAHEDRON LETTERS

Reactions of Nucleophiles with Nitroarenes: Multifacial and Versatile Electrophiles

(2014) Mieczysław Mąkosza   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and Antiproliferative Activity of Substituted 3[2-(1H-indol-3-yl)- 1,3-thiazol-4-yl]-1H-pyrrolo[3,2-b]pyridines, Marine Alkaloid Nortopsentin Analogues

(2014) A. Carbone et al.   CURRENT MEDICINAL CHEMISTRY

KOtBu-Mediated Aerobic Transition-Metal-Free Regioselective β-Arylation of Indoles: Synthesis of β-(2-/4-Nitroaryl)-indoles

(2014) Shailesh Kumar et al.   ORGANIC LETTERS

Synthesis of Heterocycles via Nucleophilic Substitution of Hydrogen in Nitroarenes

(2013) Mieczysław Mąkosza et al.   HETEROCYCLES

Synthesis and biological evaluation of novel isoxazolo[4,3-e]indoles as antibacterial agents

(2013) Mehdi Pordel et al.   RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY

Synthesis of Pentafluorosulfanyl-Containing Indoles and Oxindoles

(2013) Petr Beier et al.   SYNLETT

Synthesis of Pyrroles, Indoles, and Carbazoles through Transition-Metal-Catalyzed CH Functionalization

(2013) Naohiko Yoshikai et al.   Asian Journal of Organic Chemistry

Nucleophilic Substitution Reaction of 1-Methoxyindole-3-carbaldehyde

(2012) Masanori Somei et al.   HETEROCYCLES

Development of Scalable Manufacturing Routes to AZD1981. Application of the Semmler–Wolff Aromatisation for Synthesis of the Indole-4-amide Core

(2012) Manjunatha Sulur et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Expedient Synthesis of 1-Hydroxy-4- and 1-Hydroxy-6-nitroindoles

(2012) Krzysztof Wojciechowski et al.   SYNLETT

Straightforward protocol for the efficient synthesis of varied N1-acylated (aza)indole 2-/3-alkanoic acids and esters: optimization and scale-up

(2012) Andy J. Liedtke et al.   TETRAHEDRON

An efficient one-pot synthesis of a new heterocyclic system with high-fluorescent properties

(2011) Mohammad Rahimizadeh et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Oligonucleotides containing substituted 4-nitroindoles: Synthesis and study of their DNA duplexes

(2011) E. N. Timofeev et al.   RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY

Nucleophilic Substitution of Hydrogen in Nitroarenes: A New Chapter of Aromatic Chemistry

(2011) Mieczysław Mąkosza   SYNTHESIS-STUTTGART

A base-modulated chemoselective synthesis of 3-cyanoindoles or 4-cyanoquinolines using a palladium-catalyzed N-heterocyclization

(2011) Serge R. Banini et al.   TETRAHEDRON

3-(Arylsulfonyl)-1-(azacyclyl)-1H-indoles are 5-HT6 receptor modulators

(2010) Ronald C. Bernotas et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Nucleophilic substitution of hydrogen in electron-deficient arenes, a general process of great practical value

(2010) Mieczysław Mąkosza   CHEMICAL SOCIETY REVIEWS

Synthesis and evaluation of 9-benzylideneamino derivatives of homocamptothecin as potent inhibitors of DNA topoisomerase I

(2010) Wei Guo et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of polycyclic indole derivatives from 2,4,6-trinitrotoluene

(2010) Maxim A. Bastrakov et al.   MENDELEEV COMMUNICATIONS

Short and Simple Method of Synthesis of Some Pyrrolo[3,2-b]quinoline Derivatives from Easily Available Nitrobenzene Derivatives

(2010) Zbigniew Wróbel et al.   SYNLETT

Simple Synthesis of N-Aryl-2-nitrosoanilines in the Reaction of Nitroarenes with Aniline Anion Derivatives

(2010) Zbigniew Wróbel et al.   SYNTHESIS-STUTTGART

Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part I: Exploration of 5–6 fused rings as alternative S1 moieties

(2009) Kenji Yoshikawa et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Dual acting norepinephrine reuptake inhibitors and 5-HT2A receptor antagonists: Identification, synthesis and activity of novel 4-aminoethyl-3-(phenylsulfonyl)-1H-indoles

(2009) Gavin D. Heffernan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Nucleophilic Substitution Reaction in Indole Chemistry: 1-Methoxy-6-nitroindole-3-carbaldehyde as a Versatile Building Block for 2,3,6-Trisubstituted Indoles1,#

(2009) Masanori Somei et al.   HETEROCYCLES

Functionalization of 4,6-dinitro-2-phenylindole at position 7

(2009) M. A. Bastrakov et al.   RUSSIAN CHEMICAL BULLETIN

Convenient access to C-2 or C-5 substituted 4-azaindole derivatives

(2009) Fabienne Saab et al.   TETRAHEDRON

Substituent Effects on the Electrophilic Activity of Nitroarenes in Reactions with Carbanions

(2008) Sylwia Błażej et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and adrenolytic activity of 1-(1H-indol-4-yloxy)-3-{[2-(2-methoxyphenoxy)ethyl]amino}propan-2-ol and its enantiomers. Part 1

(2008) Grażyna Groszek et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of C3-Substituted 4-Azaindoles: An Easy Access to 4-Azamelatonin and Protected 4-Azatryptophan

(2008) Matthieu Jeanty et al.   JOURNAL OF ORGANIC CHEMISTRY

One-pot three component synthesis of heteroarylated arylacetates via VNSAr-SN reaction using N-methylpyrrolidone as general solvent

(2008) Song Cao et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Eudistomin C and E: Improved Preparation of the Indole Unit

(2008) Hiroaki Yamagishi et al.   ORGANIC LETTERS

Palladium-Catalyzed Synthesis of 3-Indolecarboxylic Acid Derivatives

(2008) Björn Söderberg et al.   SYNTHESIS-STUTTGART