Asymmetric [4+2] annulations to construct norcamphor scaffolds with 2-cyclopentenone via double amine–thiol catalysis

Switchable regioselectivity in amine-catalysed asymmetric cycloadditions

(2017) Zhi Zhou et al.   Nature Chemistry

γ′-Selective Functionalization of Cyclic Enones: Construction of a Chiral Quaternary Carbon Center by [4+2] Cycloaddition/Retro-Mannich Reaction with 3-Substituted Maleimides

(2016) Chuncheng Zou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Combinations of Aminocatalysts and Metal Catalysts: A Powerful Cooperative Approach in Selective Organic Synthesis

(2016) Samson Afewerki et al.   CHEMICAL REVIEWS

Dual Catalysis Strategies in Photochemical Synthesis

(2016) Kazimer L. Skubi et al.   CHEMICAL REVIEWS

Asymmetric Diels-Alder Cycloadditions of Trifluoromethylated Dienophiles Under Trienamine Catalysis

(2016) Xin Yuan et al.   CHEMISTRY-A EUROPEAN JOURNAL

The addition of polyfluoroalkanesulfenic acids to alkenes

(2016) Xiao-Bo Li et al.   JOURNAL OF FLUORINE CHEMISTRY

Asymmetric Lewis acid organocatalysis of the Diels-Alder reaction by a silylated C-H acid

(2016) T. Gatzenmeier et al.   SCIENCE

Pushing the Limits of Aminocatalysis: Enantioselective Transformations of α-Branched β-Ketocarbonyls and Vinyl Ketones by Chiral Primary Amines

(2015) Long Zhang et al.   ACCOUNTS OF CHEMICAL RESEARCH

Direct Catalytic Asymmetric Doubly Vinylogous Michael Addition of α,β-Unsaturated γ-Butyrolactams to Dienones

(2015) Xiaodong Gu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct Access to Multifunctionalized Norcamphor Scaffolds by Asymmetric Organocatalytic Diels-Alder Reactions

(2015) Rasmus Mose et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cinchona Alkaloid Squaramide-Catalyzed Asymmetric Michael Addition of α-Aryl Isocyanoacetates to β-Trifluoromethylated Enones and Its Applications in the Synthesis of Chiral β-Trifluoromethylated Pyrrolines

(2015) Mei-Xin Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Enantioselective Formal [4 + 2] Cycloaddition of Enones with Cyclic N-Sulfonylimines and Methylene Chromene for Chiral Spirocyclic Compounds

(2015) Jie Fei et al.   ORGANIC LETTERS

Diastereo- and Enantioselective [4+2] Cycloadditions of Cyclic Enones with Cyclic 1-Azadienes

(2015) Rong Zhou et al.   ACTA CHIMICA SINICA

Catalytic asymmetric conjugate addition of terminal alkynes to β-trifluoromethyl α,β-enones

(2014) Amparo Sanz-Marco et al.   CHEMICAL COMMUNICATIONS

Novel Organocatalytic Activation of Unmodified Morita-Baylis-Hillman Alcohols for the Synthesis of Bicyclic α-Alkylidene-Ketones

(2014) Julian Stiller et al.   CHEMISTRY-A EUROPEAN JOURNAL

Chiral silicon Lewis acids having a pentacoordinate stereogenic silicon center: 29Si NMR studies and application to asymmetric Diels–Alder reactions

(2013) Yuhsuke Sakaguchi et al.   CHEMICAL COMMUNICATIONS

Highly Diastereo- and Enantioselective Cross-Cascade Reactions of Different Enones

(2013) Huicai Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Stereospecific Asymmetric N-Heterocyclic Carbene (NHC)-Catalyzed Redox Synthesis of Trifluoromethyl Dihydropyranones and Mechanistic Insights

(2013) Alyn T. Davies et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalytic Asymmetric Construction of Chiral Hydropyridazines via Conjugate Addition of N-Monosubstituted Hydrazones to Enones

(2013) Wenbin Wu et al.   ORGANIC LETTERS

Asymmetric organocatalysis mediated by primary amines derived from cinchona alkaloids: recent advances

(2013) Jindian Duan et al.   Catalysis Science & Technology

Hydrogen-Bond-Mediated Supramolecular Iminium Ion Catalysis

(2012) Yao Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cinchona-based Primary Amine Catalysis in the Asymmetric Functionalization of Carbonyl Compounds

(2012) Paolo Melchiorre   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic enantioselective synthesis of β-trifluoromethyl pyrrolines

(2012) Hiroyuki Kawai et al.   CHEMICAL COMMUNICATIONS

Stereodivergence in Amine-Catalyzed Regioselective [4 + 2] Cycloadditions of β-Substituted Cyclic Enones and Polyconjugated Malononitriles

(2012) Xin Feng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(i)-catalyzed 1,4-conjugate arylation toward β-fluoroalkylated electron-deficient alkenes: a new entry to a construction of a tertiary carbon center possessing a fluoroalkyl group

(2012) Atsunori Morigaki et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Chiral Primary Amine Catalyzed Asymmetric Direct Cross-Aldol Reaction of Acetaldehyde

(2011) Shenshen Hu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Evaluation of the Metabolites of AMG 221, a Clinical Candidate for the Treatment of Type 2 Diabetes

(2011) Aiwen Li et al.   ACS Medicinal Chemistry Letters

Recent advances in asymmetric catalysis with cinchona alkaloid-based primary amines

(2011) Lin Jiang et al.   Catalysis Science & Technology

Synthesis of Functionalized Indoles with a Trifluoromethyl-Substituted Stereogenic Tertiary Carbon Atom Through an Enantioselective Friedel-Crafts Alkylation with β-Trifluoromethyl-α,β-enones

(2010) Gonzalo Blay et al.   CHEMISTRY-A EUROPEAN JOURNAL

Development of a Cysteine-Catalyzed Enantioselective Rauhut−Currier Reaction

(2010) Carrie E. Aroyan et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Cooperative Catalysis of Strong Bronsted Acid-Promoted Reactions Using Chiral Ureas

(2010) H. Xu et al.   SCIENCE

ortho-Acidic aromatic thiols as efficient catalysts of intramolecular Morita–Baylis–Hillman and Rauhut–Currier reactions

(2010) Philipp S. Selig et al.   TETRAHEDRON LETTERS

Organocascade Reactions of Enones Catalyzed by a Chiral Primary Amine

(2009) Li-Yuan Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

In Situ Enamine Activation in Aqueous Salt Solutions: Highly Efficient Asymmetric Organocatalytic Diels-Alder Reaction of Cyclohexenones with Nitroolefins

(2009) Dan-Qian Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Targeting Structural and Stereochemical Complexity by Organocascade Catalysis: Construction of Spirocyclic Oxindoles Having Multiple Stereocenters

(2009) Giorgio Bencivenni et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of tricyclic 5,6-dihydro-1H-pyridin-2-ones as novel, potent, and orally bioavailable inhibitors of HCV NS5B polymerase

(2009) Frank Ruebsam et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A new domino autocatalytic reaction leading to polyfunctionalized spiro[5.5]undecanes and dispiro[4.2.5.2]pentadecanes

(2009) Bo Jiang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Sordarin, an antifungal agent with a unique mode of action

(2008) Huan Liang   Beilstein Journal of Organic Chemistry

Double cascade reactions based on the Barbas dienamine platform: highly stereoselective synthesis of functionalized cyclohexanes for cardiovascular agents

(2008) Dhevalapally B. Ramachary et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The Development of Asymmetric Primary Amine Catalysts Based on Cinchona Alkaloids

(2008) Ying-Chun Chen   SYNLETT

A first high enantiocontrol of an asymmetric tertiary carbon center attached with a fluoroalkyl group via Rh(I)-catalyzed conjugate addition reaction

(2008) Tsutomu Konno et al.   TETRAHEDRON LETTERS