Synthesis of bioactive and stabilized cyclic peptides by macrocyclization using C(sp3)–H activation
出版年份 2017 全文链接
标题
Synthesis of bioactive and stabilized cyclic peptides by macrocyclization using C(sp3)–H activation
作者
关键词
-
出版物
Chemical Science
Volume 8, Issue 6, Pages 4565-4570
出版商
Royal Society of Chemistry (RSC)
发表日期
2017-04-19
DOI
10.1039/c6sc05530c
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Butelase-Mediated Macrocyclization of d -Amino-Acid-Containing Peptides
- (2016) Giang K. T. Nguyen et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Metal-Catalyzed Annulations through Activation and Cleavage of C−H Bonds
- (2016) Moisés Gulías et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- A Simple and Versatile Amide Directing Group for C−H Functionalizations
- (2016) Ru-Yi Zhu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Nitrogen Arylation for Macrocyclization of Unprotected Peptides
- (2016) Guillaume Lautrette et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Oxadiazole grafts in peptide macrocycles
- (2016) John R. Frost et al. Nature Chemistry
- Organometallic palladium reagents for cysteine bioconjugation
- (2015) Ekaterina V. Vinogradova et al. NATURE
- Structure and biosynthesis of a macrocyclic peptide containing an unprecedented lysine-to-tryptophan crosslink
- (2015) Kelsey R. Schramma et al. Nature Chemistry
- New peptide architectures through C–H activation stapling between tryptophan–phenylalanine/tyrosine residues
- (2015) Lorena Mendive-Tapia et al. Nature Communications
- C–H Functionalization in the Synthesis of Amino Acids and Peptides
- (2014) Anaïs F. M. Noisier et al. CHEMICAL REVIEWS
- Site-Selective C(sp3)–H Functionalization of Di-, Tri-, and Tetrapeptides at the N-Terminus
- (2014) Wei Gong et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups
- (2013) Guy Rouquet et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Multifaceted Roles of Disulfide Bonds. Peptides as Therapeutics
- (2013) Miriam Góngora-Benítez et al. CHEMICAL REVIEWS
- New modalities in conformationally constrained peptides for potency, selectivity and cell permeation
- (2013) Ram Dharanipragada Future Medicinal Chemistry
- A Perfluoroaryl-Cysteine SNAr Chemistry Approach to Unprotected Peptide Stapling
- (2013) Alexander M. Spokoyny et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Screening Bicyclic Peptide Libraries for Protein–Protein Interaction Inhibitors: Discovery of a Tumor Necrosis Factor-α Antagonist
- (2013) Wenlong Lian et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals
- (2012) Junichiro Yamaguchi et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- The Future of Peptide-based Drugs
- (2012) David J. Craik et al. Chemical Biology & Drug Design
- Development of α-Helical Calpain Probes by Mimicking a Natural Protein–Protein Interaction
- (2012) Hyunil Jo et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Global Analysis of Peptide Cyclization Efficiency
- (2012) Amit Thakkar et al. ACS Combinatorial Science
- Cilengitide: The First Anti-Angiogenic Small Molecule Drug Candidate. Design, Synthesis and Clinical Evaluation
- (2011) Carlos Mas-Moruno et al. Anti-Cancer Agents in Medicinal Chemistry
- Carboxylate-Assisted Transition-Metal-Catalyzed C−H Bond Functionalizations: Mechanism and Scope
- (2011) Lutz Ackermann CHEMICAL REVIEWS
- Transition metal-catalyzed arylation of unactivated C(sp3)–H bonds
- (2011) Olivier Baudoin CHEMICAL SOCIETY REVIEWS
- Contemporary strategies for peptide macrocyclization
- (2011) Christopher J. White et al. Nature Chemistry
- Robust Generation of Lead Compounds for Protein-Protein Interactions by Computational and MCR Chemistry: p53/Hdm2 Antagonists
- (2010) Anna Czarna et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Macrocyclization of Linear Peptides Enabled by Amphoteric Molecules
- (2010) Ryan Hili et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Hydrocarbon double-stapling remedies the proteolytic instability of a lengthy peptide therapeutic
- (2010) G. H. Bird et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Total Synthesis of Celogentin C by Stereoselective CH Activation
- (2009) Yiqing Feng et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Protein-Protein Interactions: A Simple Strategy to Identify Binding Sites and Peptide Antagonists
- (2009) Annamaria Sandomenico et al. Chemical Biology & Drug Design
- Synthesis of chemically modified bioactive peptides: recent advances, challenges and developments for medicinal chemistry
- (2009) Soledad Royo Gracia et al. Future Medicinal Chemistry
- The exploration of macrocycles for drug discovery — an underexploited structural class
- (2008) Edward M. Driggers et al. NATURE REVIEWS DRUG DISCOVERY
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