A practical approach to asymmetric synthesis of dolastatin 10

Design and Synthesis of a Novel N-(1H-tetrazol-5-yl)methyl Cyclic Peptoid Using Nosyl-protected N-(1-trityl-1H-tetrazol-5-yl)methyl Substituted Glycine

(2017) Girish Prabhu et al.   International Journal of Peptide Research and Therapeutics

Peptide hormones and lipopeptides: from self-assembly to therapeutic applications

(2017) J. A. Hutchinson et al.   JOURNAL OF PEPTIDE SCIENCE

An efficient approach to trans-4-hydroxy-5-substituted 2-pyrrolidinones through a stereoselective tandem Barbier process: divergent syntheses of (3R,4S)-statines, (+)-preussin and (−)-hapalosin

(2017) Chang-Mei Si et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis and biological activity evaluation of dolastatin 10 analogues with N-terminal modifications

(2017) Xin Wang et al.   TETRAHEDRON

Synthesis and structure revision of symplocin A

(2017) Lu-Ping Shao et al.   Organic Chemistry Frontiers

A Theoretical Study of Benzene Dimers in the Excited States: Wavefunction Delocalization, Charge-Transfer Admixture, and Electronic Coupling

(2017) Dongwook Kim   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Design and synthesis of novel triazole derivatives containing γ-lactam as potential antifungal agents

(2016) Yuan-Yuan Xu et al.   CHINESE CHEMICAL LETTERS

Design, synthesis and antibacterial activity of novel pleuromutilin derivatives with 4 H -pyran-4-one and pyridin-4-one substitution in the C-14 side chain

(2016) Chen-Yu Ling et al.   CHINESE CHEMICAL LETTERS

Lipopeptides: a novel antigen repertoire presented by major histocompatibility complex class I molecules

(2016) Daisuke Morita et al.   IMMUNOLOGY

Asymmetric Synthesis of Apratoxin E

(2016) Zhuo-Ya Mao et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis and Biological Evaluation of Natural and Designed Tubulysins

(2016) K. C. Nicolaou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric syntheses of epohelmins A and B by In-mediated allylation

(2016) Yi-Wen Liu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

An enantioselective total synthesis of tubulysin V

(2016) Wei Tao et al.   TETRAHEDRON

Asymmetric synthesis of epohelmins A, B and 3-epi ent- epohelmin A

(2016) Chang-Mei Si et al.   TETRAHEDRON

Studies toward asymmetric synthesis of hoiamides A and B

(2016) Ming Li et al.   TETRAHEDRON LETTERS

Asymmetric synthesis of emericellamide B

(2015) Rong-Guo Ren et al.   CHINESE CHEMICAL LETTERS

Divergent Method to trans-5-Hydroxy-6-alkynyl/alkenyl-2-piperidinones: Syntheses of (−)-Epiquinamide and (+)-Swainsonine

(2015) Chang-Mei Si et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent Advances in the Development of New Auristatins: Structural Modifications and Application in Antibody Drug Conjugates

(2015) Andreas Maderna et al.   MOLECULAR PHARMACEUTICS

Tetrahydrofuran amino acid-containing gramicidin S analogues with improved biological profiles

(2015) Sudip Pal et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Lipopeptides as the Antifungal and Antibacterial Agents: Applications in Food Safety and Therapeutics

(2015) Khem Raj Meena et al.   Biomed Research International

Stereoselective formation of chiral trans-4-hydroxy-5-substituted 2-pyrrolidinones: syntheses of streptopyrrolidine and 3-epi-epohelmin A

(2015) Chang-Mei Si et al.   Organic Chemistry Frontiers

Specific Labeling of Streptavidin for Better Understanding of Ligand Modification in Modular Method for Affinity Labeling (MoAL)

(2014) Munetaka Kunishima et al.   CHEMICAL & PHARMACEUTICAL BULLETIN

Discovery of Cytotoxic Dolastatin 10 Analogues with N-Terminal Modifications

(2014) Andreas Maderna et al.   JOURNAL OF MEDICINAL CHEMISTRY

Lipopeptides from the Tropical Marine Cyanobacterium Symploca sp.

(2014) Emily Mevers et al.   JOURNAL OF NATURAL PRODUCTS

Diastereoconvergent Synthesis of trans-5-Hydroxy-6-Substituted-2-Piperidinones by Addition–Cyclization–Deprotection Process

(2014) Chang-Mei Si et al.   ORGANIC LETTERS

A total synthesis of a highly N-methylated cyclodepsipeptide [2S,3S-Hmp]-aureobasidin L using solid-phase methods

(2014) Rani Maharani et al.   TETRAHEDRON

Dolastatin, along with Celecoxib, stimulates apoptosis by a mechanism involving oxidative stress, membrane potential change and PI3-K/AKT pathway down regulation

(2013) Honit Piplani et al.   BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS

Benzazepinones and Benzoxazepinones as Antagonists of Inhibitor of Apoptosis Proteins (IAPs) Selective for the Second Baculovirus IAP Repeat (BIR2) Domain

(2013) Andrew F. Donnell et al.   JOURNAL OF MEDICINAL CHEMISTRY

Diverse Synthesis of Marine Cyclic Depsipeptide Lagunamide A and Its Analogues

(2013) Wei Huang et al.   JOURNAL OF ORGANIC CHEMISTRY

Peptide Coupling Reagents, More than a Letter Soup

(2011) Ayman El-Faham et al.   CHEMICAL REVIEWS

Synthesis of Vaniprevir (MK-7009): Lactamization To Prepare a 22-Membered Macrocycle

(2011) Zhiguo J. Song et al.   JOURNAL OF ORGANIC CHEMISTRY

N-Linked Peptidoresorc[4]arene-Based Receptors as Noncompetitive Inhibitors for α-Chymotrypsin

(2011) Ilaria D’Acquarica et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis and Stereochemical Assignment of Burkholdac B, a Depsipeptide HDAC Inhibitor

(2011) Hanae Benelkebir et al.   ORGANIC LETTERS

Synthesis and Applications oftert-Butanesulfinamide

(2010) MaryAnn T. Robak et al.   CHEMICAL REVIEWS

Further Studies toward the Stereocontrolled Synthesis of Silicon-Containing Peptide Mimics

(2010) Dácil Hernández et al.   JOURNAL OF ORGANIC CHEMISTRY

Total synthesis of spiruchostatin B, a potent histone deacetylase inhibitor, from a microorganism

(2008) Toshiya Takizawa et al.   CHEMICAL COMMUNICATIONS

Diastereoselective Synthesis of Heteroaromatic Glycine Derivatives

(2008) Trygve Andreassen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Simple Microscale Method for Determining the Relative Stereochemistry of Statine Units

(2008) Alejandro Preciado et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis of Cruentaren B

(2008) Tushar Kanti Chakraborty et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Total Synthesis of (+)-Largazole, a Potent Inhibitor of Histone Deacetylase†

(2008) Arun K. Ghosh et al.   ORGANIC LETTERS