Tetrahydrofuran amino acid-containing gramicidin S analogues with improved biological profiles

Structure–activity relationships of the antimicrobial peptide gramicidin S and its analogs: Aqueous solubility, self-association, conformation, antimicrobial activity and interaction with model lipid membranes

(2014) Thomas Abraham et al.   BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES

Thiazole-Based γ-Building Blocks as Reverse-Turn Mimetic to Design a Gramicidin S Analogue: Conformational and Biological Evaluation

(2014) Baptiste Legrand et al.   CHEMISTRY-A EUROPEAN JOURNAL

Multidrug-resistant and extensively drug-resistant tuberculosis: a review of current concepts and future challenges

(2014) G. Gunther   CLINICAL MEDICINE

Furan-Based Locked Z-Vinylogous γ-Amino Acid Stabilizing Protein α-Turn in Water-Soluble Cyclic α3γ Tetrapeptides

(2014) Yarkali Krishna et al.   ORGANIC LETTERS

Peptidomimetics with tunable tertiary amide bond containing substituted β-proline and β-homoproline

(2014) Sandip Basu et al.   TETRAHEDRON

Cationic amphipathic D-enantiomeric antimicrobial peptides with in vitro and ex vivo activity against drug-resistant Mycobacterium tuberculosis

(2014) Yun Lan et al.   TUBERCULOSIS

A compendium of cyclic sugar amino acids and their carbocyclic and heterocyclic nitrogen analogues

(2013) Martijn Risseeuw et al.   AMINO ACIDS

Rational Design of Engineered Cationic Antimicrobial Peptides Consisting Exclusively of Arginine and Tryptophan, and Their Activity against Multidrug-Resistant Pathogens

(2013) Berthony Deslouches et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Differential spontaneous folding of mycolic acids from Mycobacterium tuberculosis

(2013) Wilma Groenewald et al.   CHEMISTRY AND PHYSICS OF LIPIDS

Dissociation of Antimicrobial and Hemolytic Activities of Gramicidin S through N-Methylation Modification

(2013) Yangmei Li et al.   ChemMedChem

Tetrahydrofuran amino acids of the past decade

(2013) Vitālijs Rjabovs et al.   TETRAHEDRON

Getting in Shape: Controlling Peptide Bioactivity and Bioavailability Using Conformational Constraints

(2012) Jonathan E. Bock et al.   ACS Chemical Biology

Polycationic Gramicidin S Analogues with Both High Antibiotic Activity and Very Low Hemolytic Activity

(2012) Makoto Tamaki et al.   CHEMICAL & PHARMACEUTICAL BULLETIN

Robust Turn Structures in α3β Cyclic Tetrapeptides Induced and Controlled by Carbo-β3 Amino Acid

(2012) Anindra Sharma et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and evaluation of strand and turn modified ring-extended gramicidin S derivatives

(2011) Annemiek D. Knijnenburg et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The Role of Antimicrobial Peptides in Preventing Multidrug-Resistant Bacterial Infections and Biofilm Formation

(2011) Seong-Cheol Park et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Design and syntheses of gramicidin S analogs, cyclo(-X-Leu-X-D-Phe-Pro-)2 (X=His, Lys, Orn, Dab and Dap)

(2011) Makoto Tamaki et al.   JOURNAL OF ANTIBIOTICS

Towards the synthesis of sugar amino acid containing antimicrobial noncytotoxic CAP conjugates with gold nanoparticles and a mechanistic study of cell disruption

(2011) Sudip Pal et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Structure–activity relationships of gramicidin S analogs containing (β-3-pyridyl)-α,β-dehydroalanine residues on membrane permeability

(2011) Keiichi Yamada et al.   MedChemComm

Influence of glucose-templated proline mimetics on the β-turn conformation of the peptide fragment Ac-Leu-d-Phe-Pro-Val-NMe2 found in Gramicidin S

(2010) Kaidong Zhang et al.   CARBOHYDRATE RESEARCH

Sequence Inversion and Phenylalanine Surrogates at the β-Turn Enhance the Antibiotic Activity of Gramicidin S

(2010) Concepción Solanas et al.   JOURNAL OF MEDICINAL CHEMISTRY

Development of CHARMM Polarizable Force Field for Nucleic Acid Bases Based on the Classical Drude Oscillator Model

(2010) Christopher M. Baker et al.   JOURNAL OF PHYSICAL CHEMISTRY B

The Structural Basis of Peptide-Protein Binding Strategies

(2010) Nir London et al.   STRUCTURE

Gramicidin S and polymyxins: the revival of cationic cyclic peptide antibiotics

(2009) Tatsushi Mogi et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

Therapeutic Index of Gramicidin S is Strongly Modulated byd-Phenylalanine Analogues at the β-Turn

(2009) Concepción Solanas et al.   JOURNAL OF MEDICINAL CHEMISTRY

Extensively drug-resistant tuberculosis: new strains, new challenges

(2008) Ritu Banerjee et al.   Expert Review of Anti-Infective Therapy

Identification of new inhibitors for alternative NADH dehydrogenase (NDH-II)

(2008) Tatsushi Mogi et al.   FEMS MICROBIOLOGY LETTERS