New insights for the use of quercetin analogs in cancer treatment

Multifaceted properties of 1,4-dimethylcarbazoles: Focus on trimethoxybenzamide and trimethoxyphenylurea derivatives as novel human topoisomerase II inhibitors

(2017) Domenico Iacopetta et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

Structure related effects of flavonoid aglycones on cell cycle progression of HepG2 cells: Metabolic activation of fisetin and quercetin by catechol- O -methyltransferase (COMT)

(2016) Miklós Poór et al.   BIOMEDICINE & PHARMACOTHERAPY

Quercetin derivatives as novel antihypertensive agents: Synthesis and physiological characterization

(2016) Fedora Grande et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

Co-delivery with nano-quercetin enhances doxorubicin-mediated cytotoxicity against MCF-7 cells

(2016) Akbar Minaei et al.   MOLECULAR BIOLOGY REPORTS

Emerging Significance of Flavonoids as P-Glycoprotein Inhibitors in Cancer Chemotherapy

(2016) Tripta Bansal et al.   JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES

Synthesis and Bioactivity of Quercetin Aspirinates

(2014) Chenjuan Lu et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

Synthesis, characterization and cytotoxic activity on breast cancer cells of new half-titanocene derivatives

(2013) Esther Sirignano et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines

(2013) Marina Sala et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Site-Specific Anticancer Effects of Dietary Flavonoid Quercetin

(2013) Katrin Sak   NUTRITION AND CANCER-AN INTERNATIONAL JOURNAL

N-(Phenoxyalkyl)amides as MT1 and MT2 ligands: Antioxidant properties and inhibition of Ca2+/CaM-dependent kinase II

(2012) Alessia Carocci et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Life or death: Neuroprotective and anticancer effects of quercetin

(2012) Federico Dajas   JOURNAL OF ETHNOPHARMACOLOGY

Evaluation of Antioxidant and Immunity Activities of Quercetin in Isoproterenol-Treated Rats

(2012) Hui Liu et al.   MOLECULES

Enhancement of biological activities of nanostructured hydrophobic drug species

(2012) Qiusen Han et al.   Nanoscale

Induction of Apoptosis in Cancer Cells at Low Silver Nanoparticle Concentrations using Chitosan Nanocarrier

(2011) Pallab Sanpui et al.   ACS Applied Materials & Interfaces

Remarkable Stability and Cytostatic Effect of a Quercetin Conjugate, 3,7-Bis-O-Pivaloxymethyl (POM) Quercetin

(2011) Mi Kyoung Kim et al.   ChemMedChem

The pro-apoptotic effect of quercetin in cancer cell lines requires ERβ-dependent signals

(2011) Pamela Bulzomi et al.   JOURNAL OF CELLULAR PHYSIOLOGY

Genesis and development of DPPH method of antioxidant assay

(2011) Sagar B. Kedare et al.   JOURNAL OF FOOD SCIENCE AND TECHNOLOGY-MYSORE

Quercetin Diacylglycoside Analogues Showing Dual Inhibition of DNA Gyrase and Topoisomerase IV as Novel Antibacterial Agents

(2011) Abugafar M. L. Hossion et al.   JOURNAL OF MEDICINAL CHEMISTRY

Innovative antioxidant thermo-responsive hydrogels by radical grafting of catechin on inulin chain

(2010) U.G. Spizzirri et al.   CARBOHYDRATE POLYMERS

Antiproliferative and pro-apoptotic effects of quercetin on human pancreatic carcinoma cell lines EPP85-181P and EPP85-181RDB.

(2010) Sylwia Borska et al.   FOLIA HISTOCHEMICA ET CYTOBIOLOGICA

Inhibition of angiogenesis by quercetin in tamoxifen-resistant breast cancer cells

(2010) Soo Jin Oh et al.   FOOD AND CHEMICAL TOXICOLOGY

The Flavonol Isorhamnetin Exhibits Cytotoxic Effects on Human Colon Cancer Cells

(2010) Sara Jaramillo et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Enhanced Stability and Intracellular Accumulation of Quercetin by Protection of the Chemically or Metabolically Susceptible Hydroxyl Groups with a Pivaloxymethyl (POM) Promoiety

(2010) Mi Kyoung Kim et al.   JOURNAL OF MEDICINAL CHEMISTRY

Regioselective O-Derivatization of Quercetin via Ester Intermediates. An Improved Synthesis of Rhamnetin and Development of a New Mitochondriotropic Derivative

(2010) Andrea Mattarei et al.   MOLECULES

Distinct signalling mechanisms are involved in the dissimilar myocardial and coronary effects elicited by quercetin and myricetin, two red wine flavonols

(2010) T. Angelone et al.   NUTRITION METABOLISM AND CARDIOVASCULAR DISEASES

DNA Binding Ellipticine Analogues: Synthesis, Biological Evaluation, and Structure-Activity Relationships

(2009) Maria Grazia Ferlin et al.   ChemMedChem

Quercetin-induced apoptosis acts through mitochondrial- and caspase-3-dependent pathways in human breast cancer MDA-MB-231 cells

(2009) Su-Yu Chien et al.   HUMAN & EXPERIMENTAL TOXICOLOGY

Synthesis, inhibition of NO production and antiproliferative activities of some indole derivatives

(2009) Maria Stefania Sinicropi et al.   JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

Preventive effect of the flavonoid, quercetin, on hepatic cancer in rats via oxidant/antioxidant activity: molecular and histological evidences

(2009) AlaaEddeen M Seufi et al.   JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH

Cytotoxicity of flavones and flavonols to a human esophageal squamous cell carcinoma cell line (KYSE-510) by induction of G2/M arrest and apoptosis

(2009) Qiang Zhang et al.   TOXICOLOGY IN VITRO

Health effects of quercetin: From antioxidant to nutraceutical

(2008) Agnes W. Boots et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Quercetin inhibits lymphocyte activation and proliferation without inducing apoptosis in peripheral mononuclear cells

(2008) Enrico Lugli et al.   LEUKEMIA RESEARCH