Regioselective “hydroamination” of alk-3-ynones with non-symmetrical o-phenylenediamines. Synthesis of diversely substituted 3H-1,5-benzodiazepines via (Z)-3-amino-2-alkenones

Efficient Synthesis and Biological Evaluation of a Novel Series of 1,5-Benzodiazepine Derivatives as Potential Antimicrobial Agents

(2016) Ying-shuang An et al.   Chemical Biology & Drug Design

Construction of the 1,5-Benzodiazepine Skeleton from o-Phenylendiamine and Propargylic Alcohols via a Domino Gold-Catalyzed Hydroamination/Cyclization Process

(2016) Sandro Cacchi et al.   ORGANIC LETTERS

An intramolecular C–N cross-coupling of β-enaminones: a simple and efficient way to precursors of some alkaloids ofGalipea officinalis

(2015) Hana Doušová et al.   Beilstein Journal of Organic Chemistry

Phenyliodine(III) Diacetate Mediated Oxidative Cyclization of 1-Alkenoyl-1-carbamoyl Cycloalkanes: Access to Spiro-Fused Dihydrofuran-3(2H)-ones

(2015) Jingwen Yuan et al.   ORGANIC LETTERS

Facile and efficient synthesis of benzo[b][1,5]diazepines by three-component coupling of aromatic diamines, Meldrum’s acid, and isocyanides catalyzed by Fe3O4 nanoparticles

(2015) Mohammad Ali Ghasemzadeh et al.   RESEARCH ON CHEMICAL INTERMEDIATES

Facile synthesis of both perfluoroalkyl and phosphonate groups substituted trans-1,5-benzodiazepine and its derivatives via a one-pot catalyst-free process

(2015) Yangyong Shen et al.   TETRAHEDRON

Hydrogen–deuterium exchange of aromatic amines and amides using deuterated trifluoroacetic acid

(2015) Richard Giles et al.   TETRAHEDRON LETTERS

Synthesis, crystal structures and cytotoxic activity of new 1,3,4,5-tetrahydro-2H-1,5-benzodiazepine derivatives

(2015) Hassan M. Faidallah et al.   JOURNAL OF CHEMICAL RESEARCH

Discovery of novel 1,5-benzodiazepine-2,4-dione derivatives as potential anticancer agents

(2014) Yinbo Chen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

QSAR and 3D-QSAR studies applied to compounds with anticonvulsant activity

(2014) Juan C Garro Martinez et al.   Expert Opinion on Drug Discovery

Microwave-Assisted Synthesis of Benzo-fused Seven-membered Azaheterocycles

(2014) Rajeev Sakhuja et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Gold(I)-Catalyzed, Stereocontrolled Enamide Synthesis from Primary Amides and Propargyl Aldehydes Using a Tandem Strategy

(2014) Sang Min Kim et al.   ORGANIC LETTERS

Highly efficient one-pot, three-component synthesis of 1,5-benzodiazepine derivatives

(2013) Xiao-Qing Li et al.   CHINESE CHEMICAL LETTERS

Facile Synthesis of Perfluoroalkyl Substituted 1H-Benzo[b][1,4]-diazepine-2(3H)-ones via a Catalyst-Free Process

(2013) Shiyan Zhai et al.   CHINESE JOURNAL OF ORGANIC CHEMISTRY

One-pot microwave assisted synthesis of new 2-alkoxycarbonylmethylene-4-oxo-1,5-benzo-, naphtho-, and pyridodiazepines and assessment of their cytogenetic activity

(2013) Nicolaos Eleftheriadis et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Catalyst-free chemo-/regio-/stereo-selective amination of alk-3-ynones. Synthesis of 1,5-benzodiazepines and 3-amino-2-alkenones

(2013) Agnes Solan et al.   GREEN CHEMISTRY

Preyssler catalyst-promoted rapid, clean, and efficient condensation reactions for 3H-1,5-benzodiazepine synthesis in solvent-free conditions

(2013) Gustavo A. Pasquale et al.   TETRAHEDRON LETTERS

2,6-Pyridinedicarboxylic acid as organocatalyst for the synthesis of 1,5-benzodiazepines through one-pot reaction

(2013) Mohan Lal et al.   TETRAHEDRON LETTERS

Recyclable gallium(III) triflate-catalyzed [4+3] cycloaddition for synthesis of 2,4-disubstituted-3H-benzo[b][1,4]diazepines

(2013) Shi-Gang Huang et al.   TETRAHEDRON LETTERS

A theoretical study of the conformation and dynamic properties of 1,5-benzodiazepines and their derivatives

(2013) Rosa M. Claramunt et al.   Computational and Theoretical Chemistry

Studies on Elimination Pathways of β-Halovinyl Ketones Leading to Allenyl and Propargyl Ketones and Furans under the Action of Mild Bases

(2012) Hun Young Kim et al.   JOURNAL OF ORGANIC CHEMISTRY

Gold(I)-Catalyzed Synthesis of 1,5-Benzodiazepines Directly from o-Phenylenediamines and Alkynes

(2012) Jianqiang Qian et al.   JOURNAL OF ORGANIC CHEMISTRY

Room temperature syntheses of entirely diverse substituted β-fluorofurans

(2012) Yan Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of diversely 1,3,5-trisubstituted pyrazoles via 5-exo-dig cyclization

(2012) Dmitry A. Borkin et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Electrophilic Cyclizations of 2-Fluoroalk-3-yn-1-ones: Room-Temperature Synthesis of Diversely 2,5-Disubstituted 3,4-Fluorohalofurans

(2011) Yan Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

QSAR Study and Molecular Design of Open-Chain Enaminones as Anticonvulsant Agents

(2011) Juan Garro Martinez et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Gold(I)-Catalyzed Cycloisomerization of 2-Fluoroalk-3-yn-1-ones: Synthesis of 2,5-Substituted 3-Fluorofurans

(2010) Yan Li et al.   ADVANCED SYNTHESIS & CATALYSIS

The treatments of chronic insomnia: A review of benzodiazepine receptor agonists and psychological and behavioral therapies

(2009) Dieter Riemann et al.   SLEEP MEDICINE REVIEWS

Enaminones 8: CoMFA and CoMSIA studies on some anticonvulsant enaminones

(2008) Patrice L. Jackson et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Three-Component Synthesis of Cryofluorescent 2,4-Disubstituted 3H-1,5-Benzodiazepines - Conformational Control of ­Emission Properties

(2008) Benjamin Willy et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Zinc-Catalyzed Cycloisomerizations. Synthesis of Substituted Furans and Furopyrimidine Nucleosides

(2008) Adam Sniady et al.   JOURNAL OF ORGANIC CHEMISTRY