Synthesis of diversely 1,3,5-trisubstituted pyrazoles via 5-exo-dig cyclization

Room temperature syntheses of entirely diverse substituted β-fluorofurans

(2012) Yan Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Stereoselective synthesis of novel pyrazole derivatives using tert-butansulfonamide as a chiral auxiliary

(2012) Chang Min Park et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Terminal Alkyne Addition to Diazodicarboxylates: Synthesis of Hydrazide Linked Alkynes (Ynehydrazides)

(2012) Ramsay E. Beveridge et al.   ORGANIC LETTERS

1,3-Dipolar cycloaddition of nitrile imines with α,β-unsaturated lactones, thiolactones and lactams: synthesis of ring-fused pyrazoles

(2012) Jay Zumbar Chandanshive et al.   TETRAHEDRON

Gold-Catalyzed Hydroamination of Alkynes and Allenes with Parent Hydrazine

(2011) Rei Kinjo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent Advances in the Regioselective Synthesis of Pyrazoles

(2011) Joo-Yong Yoon et al.   CURRENT ORGANIC CHEMISTRY

Recent Advances in the Chemistry of Pyrazoles. Properties, Biological Activities, and Syntheses

(2011) Andreas Schmidt et al.   CURRENT ORGANIC CHEMISTRY

Microwave-Assisted Heterogeneous Catalysis: An Environmentally Benign Tool for Contemporary Organic Synthesis

(2011) Seema Bag et al.   CURRENT ORGANIC SYNTHESIS

Electrophilic Cyclizations of 2-Fluoroalk-3-yn-1-ones: Room-Temperature Synthesis of Diversely 2,5-Disubstituted 3,4-Fluorohalofurans

(2011) Yan Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Environmentally benign synthesis of heterocyclic compounds by combined microwave-assisted heterogeneous catalytic approaches†

(2011) Arif Daştan et al.   GREEN CHEMISTRY

Design, Synthesis, Docking, and Biological Evaluation of Novel Diazide-Containing Isoxazole- and Pyrazole-Based Histone Deacetylase Probes

(2011) Raghupathi Neelarapu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Discovery of a Novel Class of Orally Active Trypanocidal N-Myristoyltransferase Inhibitors

(2011) Stephen Brand et al.   JOURNAL OF MEDICINAL CHEMISTRY

Tri- and Tetrasubstituted Pyrazole Derivates: Regioisomerism Switches Activity from p38MAP Kinase to Important Cancer Kinases

(2011) Bassam Abu Thaher et al.   JOURNAL OF MEDICINAL CHEMISTRY

Microwave-Assisted and Continuous Flow Multistep Synthesis of 4-(Pyrazol-1-yl)carboxanilides

(2011) David Obermayer et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Pyrazoles via Electrophilic Cyclization

(2011) Metin Zora et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Selective Synthesis of Pyrazole and Spiropyrazoline Phosphonates via Base-Assisted Reaction of the Bestmann–Ohira Reagent with Enones

(2011) Deepti Verma et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Pyrazoles via CuI-Mediated Electrophilic Cyclizations of α,β-Alkynic Hydrazones

(2011) Metin Zora et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Substituted Pyrazoles via Tandem Cross-Coupling/Electrocyclization of Enol Triflates and Diazoacetates

(2011) David J. Babinski et al.   JOURNAL OF ORGANIC CHEMISTRY

Heterogeneous Catalytic Hydrogenation of Unprotected Indoles in Water: A Green Solution to a Long-Standing Challenge

(2011) Aditya Kulkarni et al.   ORGANIC LETTERS

Gold(I)-Catalyzed Cycloisomerization of 2-Fluoroalk-3-yn-1-ones: Synthesis of 2,5-Substituted 3-Fluorofurans

(2010) Yan Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Discovery of novel, potent, selective, and orally active human glucagon receptor antagonists containing a pyrazole core

(2010) Dong-Ming Shen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Microwave-assisted multicomponent domino cyclization–aromatization: an efficient approach for the synthesis of substituted quinolines

(2010) Aditya Kulkarni et al.   GREEN CHEMISTRY

Discovery ofN-[(4R)-6-(4-Chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2H-pyrano[2,3-b]pyridin-4-yl]-5-methyl-1H-pyrazole-3-carboxamide (MK-5596) as a Novel Cannabinoid-1 Receptor (CB1R) Inverse Agonist for the Treatment of Obesity

(2010) Lin Yan et al.   JOURNAL OF MEDICINAL CHEMISTRY

Access to 2,5-Diamidopyrroles and 2,5-Diamidofurans by Au(I)-Catalyzed Double Hydroamination or Hydration of 1,3-Diynes

(2010) Søren Kramer et al.   ORGANIC LETTERS

New Synthesis of Fluorinated Pyrazoles

(2010) Riccardo Surmont et al.   ORGANIC LETTERS

Antitumor Efficacy of the Novel RAF Inhibitor GDC-0879 Is Predicted by BRAFV600E Mutational Status and Sustained Extracellular Signal-Regulated Kinase/Mitogen-Activated Protein Kinase Pathway Suppression

(2009) K. P. Hoeflich et al.   CANCER RESEARCH

Synthesis of Celecoxib Analogues Possessing aN-Difluoromethyl-1,2-dihydropyrid-2-one 5-Lipoxygenase Pharmacophore: Biological Evaluation as Dual Inhibitors of Cyclooxygenases and 5-Lipoxygenase with Anti-Inflammatory Activity

(2009) Morshed A. Chowdhury et al.   JOURNAL OF MEDICINAL CHEMISTRY

Pharmacodynamics of 2- ethan-1-ol (GDC-0879), a Potent and Selective B-Raf Kinase Inhibitor: Understanding Relationships between Systemic Concentrations, Phosphorylated Mitogen-Activated Protein Kinase Kinase 1 Inhibition, and Efficacy

(2009) H. Wong et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Pd-Catalyzed Cross-Coupling of Functionalized Organozinc Reagents with Thiomethyl-Substituted Heterocycles

(2009) Albrecht Metzger et al.   ORGANIC LETTERS

APPLICATION OF CLAY CATALYSTS IN ORGANIC SYNTHESIS. A REVIEW

(2009) Sujaya Dasgupta et al.   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

Zinc-Catalyzed Cycloisomerizations. Synthesis of Substituted Furans and Furopyrimidine Nucleosides

(2008) Adam Sniady et al.   JOURNAL OF ORGANIC CHEMISTRY