标题
Biologically active γ-lactams: synthesis and natural sources
作者
关键词
-
出版物
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 14, Issue 43, Pages 10134-10156
出版商
Royal Society of Chemistry (RSC)
发表日期
2016-10-07
DOI
10.1039/c6ob01349j
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- The anti-dementia drug candidate, (−)-clausenamide, improves memory impairment through its multi-target effect
- (2016) Shifeng Chu et al. PHARMACOLOGY & THERAPEUTICS
- Recent Advances in Chemistry of γ-Lactams: Part I. Synthesis Starting from Acyclic or Cyclic Precursors
- (2016) Gianluca Martelli et al. CURRENT ORGANIC CHEMISTRY
- Hydroxamic acid based histone deacetylase inhibitors with confirmed activity against the malaria parasite
- (2015) Giuseppe Giannini et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Selective CB2 receptor agonists. Part 2: Structure–activity relationship studies and optimization of proline-based compounds
- (2015) Doris Riether et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Recent Advances in Chemistry of γ-Lactams: Part II. Functionalization by C-C or CHeteroatom Bond Formation
- (2014) Gianluca Martelli et al. CURRENT ORGANIC CHEMISTRY
- Tetramic Acid Analogues Produced by Coculture of Saccharopolyspora erythraea with Fusarium pallidoroseum
- (2014) James Whitt et al. JOURNAL OF NATURAL PRODUCTS
- Recent progress towards transition metal-catalyzed synthesis of γ-lactams
- (2014) Long-Wu Ye et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- GAMMA-HYDROXYBUTYRIC ACID (GHB) MEASUREMENT BY GC-MS IN BLOOD, URINE AND GASTRIC CONTENTS, FOLLOWING AN ACUTE INTOXICATION IN BELGIUM
- (2014) Q. Bodson et al. ACTA CLINICA BELGICA
- Umpolung of Hemiaminals: Titanocene-Catalyzed Dehydroxylative Radical Coupling Reactions with Activated Alkenes
- (2013) Xiao Zheng et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- New route to the 5-((arylthio- and heteroarylthio)methylene)-3-(2,2,2-trifluoroethyl)-furan-2(5H)-ones—Key intermediates in the synthesis of 4-aminoquinoline γ-lactams as potent antimalarial compounds
- (2013) Oleksandr S. Kanishchev et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Novel Concise Synthesis of (−)-Clausenamide
- (2013) Di Liu et al. CHINESE JOURNAL OF CHEMISTRY
- Adjunctive brivaracetam for uncontrolled focal and generalized epilepsies: Results of a phase III, double-blind, randomized, placebo-controlled, flexible-dose trial
- (2013) Patrick Kwan et al. EPILEPSIA
- Adjunctive brivaracetam in adults with uncontrolled focal epilepsy: Results from a double-blind, randomized, placebo-controlled trial
- (2013) Philippe Ryvlin et al. EPILEPSIA
- The fusarin analog NG-391 impairs nucleic acid formation in K-562 leukemia cells
- (2013) Markus Bohnert et al. Phytochemistry Letters
- Evolution of secondary metabolites in legumes (Fabaceae)
- (2013) M. Wink SOUTH AFRICAN JOURNAL OF BOTANY
- Structure and property based design, synthesis and biological evaluation of γ-lactam based HDAC inhibitors: Part II
- (2012) Chulho Lee et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Natural and synthetic α-methylenelactones and α-methylenelactams with anticancer potential
- (2012) Anna Janecka et al. DRUG DISCOVERY TODAY
- (−)Clausenamide facilitates synaptic transmission at hippocampal Schaffer collateral-CA1 synapses
- (2012) Na Ning et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- Discovery, Synthesis, and Biological Evaluation of Orally Active Pyrrolidone Derivatives as Novel Inhibitors of p53–MDM2 Protein–Protein Interaction
- (2012) Chunlin Zhuang et al. JOURNAL OF MEDICINAL CHEMISTRY
- Property-Based Optimization of Hydroxamate-Based γ-Lactam HDAC Inhibitors to Improve Their Metabolic Stability and Pharmacokinetic Profiles
- (2012) Eunhyun Choi et al. JOURNAL OF MEDICINAL CHEMISTRY
- Incorporation of a 3-(2,2,2-Trifluoroethyl)-γ-hydroxy-γ-lactam Motif in the Side Chain of 4-Aminoquinolines. Syntheses and Antimalarial Activities
- (2012) Damien Cornut et al. JOURNAL OF MEDICINAL CHEMISTRY
- The enzymes of β-lactam biosynthesis
- (2012) Refaat B. Hamed et al. NATURAL PRODUCT REPORTS
- Bioinspired and Concise Synthesis of (±)-Stemoamide
- (2011) Yan Wang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Transformation of thiols to disulfides by epolactaene and its derivatives
- (2011) Kouji Kuramochi et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Recent Advances in the Synthesis of α-Alkylidene-Substituted δ-Lactones, γ-Lactams and δ-Lactams
- (2011) Anna Albrecht et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Total Synthesis of (−)-Salinosporamide A
- (2011) Nobuhiro Satoh et al. ORGANIC LETTERS
- Fusarin C acts like an estrogenic agonist and stimulates breast cancer cells in vitro
- (2011) T.E. Sondergaard et al. TOXICOLOGY LETTERS
- Design, synthesis and biological evaluation of γ-lactam hydroxamate based TACE inhibitors
- (2011) Anil Argade et al. MedChemComm
- Levetiracetam in the treatment of epilepsy
- (2011) Bassel Abou-Khalil Neuropsychiatric Disease and Treatment
- Salinosporamide Natural Products: Potent 20 S Proteasome Inhibitors as Promising Cancer Chemotherapeutics
- (2010) Tobias A. M. Gulder et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- The chemistry of Stemona alkaloids: An update
- (2010) Ronaldo Aloise Pilli et al. NATURAL PRODUCT REPORTS
- Histone Deacetylase Inhibitors: Recent Insights from Basic to Clinical Knowledge & Patenting of Anti-Cancer Actions
- (2010) Vincenzo Carafa et al. Recent Patents on Anti-Cancer Drug Discovery
- An alternate synthesis of levetiracetam
- (2010) Ravikumar Mylavarapu et al. Green Chemistry Letters and Reviews
- Gamma-lactams—A novel scaffold for highly potent and selective α7 nicotinic acetylcholine receptor agonists
- (2009) Albert Enz et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Pseurotin A and its analogues as inhibitors of immunoglobuline E production
- (2009) Minoru Ishikawa et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and activity in enhancing long-term potentiation (LTP) of clausenamide stereoisomers
- (2009) Zhiqiang Feng et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Flavan-3-ols Having a γ-Lactam from the Roots of Actinidia arguta Inhibit the Formation of Advanced Glycation End Products in Vitro
- (2009) Dae Sik Jang et al. CHEMICAL & PHARMACEUTICAL BULLETIN
- A Short and Efficient Synthesis of (−)-7-Methylomuralide, a Potent Proteasome Inhibitor
- (2009) Ryan A. Shenvi et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Chemistry and biology of non-tetramic γ-hydroxy-γ-lactams and γ-alkylidene-γ-lactams from natural sources
- (2009) Bastien Nay et al. NATURAL PRODUCT REPORTS
- From N-triisopropylsilylpyrrole to an optically active C-4 substituted pyroglutamic acid: total synthesis of penmacric acid
- (2009) Christophe Berini et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- A Synthesis of (±)-Stemoamide Using the Intramolecular Propargylic Barbier Reaction
- (2009) Roderick Bates et al. SYNLETT
- Efficient Total Synthesis of Novel Bioactive Microbial Metabolites
- (2008) Toshiaki Sunazuka et al. ACCOUNTS OF CHEMICAL RESEARCH
- Entry to Heterocycles Based on Indium-Catalyzed Conia-Ene Reactions: Asymmetric Synthesis of (−)-Salinosporamide A
- (2008) Keisuske Takahashi et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Discovery and development of the anticancer agent salinosporamide A (NPI-0052)
- (2008) William Fenical et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Diversity-Oriented Synthesis and Preliminary Biological Screening of Highly Substituted Five-Membered Lactones and Lactams Originating From an Allyboration of Aldehydes and Imines
- (2008) Tim G. Elford et al. JOURNAL OF COMBINATORIAL CHEMISTRY
- Organocatalytic Asymmetric Total Synthesis of (R)-Rolipram and Formal Synthesis of (3S,4R)-Paroxetine
- (2008) Peter S. Hynes et al. ORGANIC LETTERS
- Codinaeopsin, an Antimalarial Fungal Polyketide
- (2008) Renee Kontnik et al. ORGANIC LETTERS
- Antimicrobial Activity of Pyrrocidines fromAcremonium zeaeAgainst Endophytes and Pathogens of Maize
- (2008) Donald T. Wicklow et al. PHYTOPATHOLOGY
- A convenient synthesis and cytotoxic evaluation of N-unsubstituted α-methylene-γ-lactams
- (2008) Henryk Krawczyk et al. TETRAHEDRON
- Imine allylation using 2-alkoxycarbonyl allylboronates as an expedient three-component reaction to polysubstituted α-exo-methylene-γ-lactams
- (2008) Tim G. Elford et al. TETRAHEDRON LETTERS
- Chemoenzymatic total synthesis and determination of the absolute configuration of (S)-nebracetam
- (2008) Sho Yamashita et al. TETRAHEDRON-ASYMMETRY
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreAdd your recorded webinar
Do you already have a recorded webinar? Grow your audience and get more views by easily listing your recording on Peeref.
Upload Now