Organocatalytic Enantioselective Friedel-Crafts Alkylation of 1-Naphthol Derivatives and Activated Phenols with Ethyl Trifluoropyruvate

Bifunctional Amine-Squaramides: Powerful Hydrogen-Bonding Organocatalysts for Asymmetric Domino/Cascade Reactions

(2015) Pankaj Chauhan et al.   ADVANCED SYNTHESIS & CATALYSIS

Organocatalytic Asymmetric Addition of Naphthols and Electron-Rich Phenols to Isatin-Derived Ketimines: Highly Enantioselective Construction of Tetrasubstituted Stereocenters

(2015) Marc Montesinos-Magraner et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Strategies for the asymmetric functionalization of indoles: an update

(2015) Renato Dalpozzo   CHEMICAL SOCIETY REVIEWS

Catalytic asymmetric conjugate addition of terminal alkynes to β-trifluoromethyl α,β-enones

(2014) Amparo Sanz-Marco et al.   CHEMICAL COMMUNICATIONS

Chiral transition-metal complexes as Brønsted-acid catalysts for the asymmetric Friedel–Crafts hydroxyalkylation of indoles

(2014) Daniel Carmona et al.   DALTON TRANSACTIONS

Lignans from the Aerial Parts of Saururus chinensis: Isolation, Structural Characterization, and Their Effects on Platelet Aggregation

(2014) Wei-Jern Tsai et al.   JOURNAL OF NATURAL PRODUCTS

Syntheses of the Fungal Metabolites Boletopsins 7, 11, and 12 from the Papua New Guinea Medicinal Mushroom Boletopsis sp.

(2014) Andrew M. Beekman et al.   JOURNAL OF ORGANIC CHEMISTRY

N,N′-Dioxide–Scandium(III)-Catalyzed Asymmetric Aza-Friedel–Crafts Reaction of Sesamol with Aldimines

(2014) Sha Bai et al.   JOURNAL OF ORGANIC CHEMISTRY

C3-Symmetric chiral trisimidazoline-catalyzed Friedel–Crafts (FC)-type reaction

(2014) Shinobu Takizawa et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Chiral Brønsted Acid Catalysts. Activation of Methyl 3,3,3-Trifluoropyruvate by Hydroxymethylpyridine-Containing Half-Sandwich Complexes

(2014) Daniel Carmona et al.   ORGANOMETALLICS

Organocatalytic asymmetric Friedel–Crafts reaction of 1-naphthols with isatins: an enantioselective synthesis of 3-aryl-3-hydroxy-2-oxindoles

(2014) Jasneet Kaur et al.   TETRAHEDRON LETTERS

Catalytic and highly enantioselective Friedel–Crafts type reactions of heteroaromatic compounds with trifluoropyruvate and glyoxylate by a dicationic palladium complex

(2014) Kohsuke Aikawa et al.   TETRAHEDRON-ASYMMETRY

Asymmetric synthesis of trans-dihydroarylfurans in a Friedel–Crafts/substitution domino reaction under squaramide catalysis

(2013) Carlos Jarava-Barrera et al.   CHEMICAL COMMUNICATIONS

Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

(2013) Jiang Wang et al.   CHEMICAL REVIEWS

Enantioselective inhibition of reverse transcriptase (RT) of HIV-1 by non-racemic indole-based trifluoropropanoates developed by asymmetric catalysis using recyclable organocatalysts

(2013) Xin Han et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Organocatalytic asymmetric Michael addition of 2-naphthols to alkylideneindolenines generated in situ from arenesulfonylalkylindoles

(2013) Liangliang Yu et al.   TETRAHEDRON LETTERS

Organocatalytic enantioselective aza-Friedel–Crafts reaction of sesamols with N-sulfonylimines catalyzed by 6′-OH Cinchona alkaloids

(2013) Pankaj Chauhan et al.   TETRAHEDRON LETTERS

Organocatalytic Enantioselective Friedel-Crafts Reaction of 1-Naphthols with Isatins and an Unexpected Spontaneous Dehydration Process

(2013) Deyan Wu et al.   Asian Journal of Organic Chemistry

Iminium ion catalysis: the enantioselective Friedel–Crafts alkylation–acetalization cascade of naphthols with α,β-unsaturated cyclic ketones

(2012) Enrico Paradisi et al.   CHEMICAL COMMUNICATIONS

Asymmetric Calcium Catalysis: Highly Enantioselective Carbonyl-Ene and Friedel-Crafts Reactions for the Synthesis of Quaternary α-Hydroxy Esters Bearing a Trifluoromethyl Group

(2012) Magnus Rueping et al.   Chemistry-An Asian Journal

Vanadium-catalyzed enantioselective Friedel–Crafts-type reactions

(2012) Shinobu Takizawa et al.   DALTON TRANSACTIONS

Enhanced efficiency of recyclable C3-symmetric cinchonine-squaramides in the asymmetric Friedel–Crafts reaction of indoles with alkyl trifluoropyruvate

(2012) Xin Han et al.   TETRAHEDRON-ASYMMETRY

Asymmetric Friedel-Crafts Reaction of Indoles with Ethyl Trifluoropyruvate Using a Copper(I)-Bisoxazolidine Catalyst

(2011) Christian Wolf et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly enantioselective Friedel–Crafts alkylation reaction catalyzed by rosin-derived tertiary amine–thiourea: synthesis of modified chromanes with anticancer potency

(2011) Xianxing Jiang et al.   CHEMICAL COMMUNICATIONS

Squaramides: physical properties, synthesis and applications

(2011) R. Ian Storer et al.   CHEMICAL SOCIETY REVIEWS

Squaramides: Bridging from Molecular Recognition to Bifunctional Organocatalysis

(2011) José Alemán et al.   CHEMISTRY-A EUROPEAN JOURNAL

Linking Conformational Flexibility and Kinetics: Catalytic 1,4-Type Friedel-Crafts Reactions of Phenols Utilizing 1,3-Diamine-Tethered Guanidine/Bisthiourea Organocatalysts

(2011) Yoshihiro Sohtome et al.   Chemistry-An Asian Journal

Asymmetric Organocatalytic Aza-Friedel-Crafts Reaction of Naphthols with N-Sulfonyl Imines

(2011) Pankaj Chauhan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Enantioselective Friedel−Crafts Reactions of 1-Naphthols with Aldimines

(2011) Guixia Liu et al.   ORGANIC LETTERS

Asymmetric synthesis of the 6-cyanoindole derivatives as non-steroidal glucocorticoid receptor modulators using (+)- and (−)-tert-butyl 6-cyano-3-[3-ethoxy-1,1,1-trifluoro-2-hydroxy-3-oxopropan-2-yl]-1H-indole-1-carboxylate

(2011) Takaaki Sumiyoshi et al.   TETRAHEDRON-ASYMMETRY

Highly Enantioselective Zinc-Catalyzed Friedel-Crafts Alkylation of Indoles with Ethyl Trifluoropyruvate

(2010) Yonghai Hui et al.   ADVANCED SYNTHESIS & CATALYSIS

Entropy-Controlled Catalytic Asymmetric 1,4-Type Friedel-Crafts Reaction of Phenols Using Conformationally Flexible Guanidine/Bisthiourea Organocatalyst

(2010) Yoshihiro Sohtome et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Construction of Stereogenic Carbon Centers Featuring a Trifluoromethyl Group from Prochiral Trifluoromethylated Substrates

(2010) Jing Nie et al.   CHEMICAL REVIEWS

Organocatalytic strategies for the asymmetric functionalization of indoles

(2010) Giuseppe Bartoli et al.   CHEMICAL SOCIETY REVIEWS

Synthesis of Functionalized Indoles with a Trifluoromethyl-Substituted Stereogenic Tertiary Carbon Atom Through an Enantioselective Friedel-Crafts Alkylation with β-Trifluoromethyl-α,β-enones

(2010) Gonzalo Blay et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalyst-free and catalytic Friedel–Crafts alkylations of indoles in Solkane® 365mfc, an environmentally benign alternative solvent

(2010) Xiu-Hua Xu et al.   GREEN CHEMISTRY

Enantioselective Friedel–Crafts alkylation of indole derivatives catalyzed by new Yb(OTf)3-pyridylalkylamine complexes as chiral Lewis acids

(2010) Guillaume Grach et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Efavirenz in the therapy of HIV infection

(2009) Natella Y Rakhmanina et al.   Expert Opinion on Drug Metabolism & Toxicology

Organocatalytic Asymmetric Friedel−Crafts Alkylation/Cyclization Cascade Reaction of 1-Naphthols and α,β-Unsaturated Aldehydes: An Enantioselective Synthesis of Chromanes and Dihydrobenzopyranes

(2009) Liang Hong et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalyzed Friedel–Craft-type reaction of 2-naphthol with β,γ-unsaturated α-keto ester to form novel optically active naphthopyran derivatives

(2009) Xiao-Sheng Wang et al.   TETRAHEDRON-ASYMMETRY

Novel EnantiocomplementaryC2‐Symmetric Chiral Bis(imidazoline) Ligands: Highly Enantioselective Friedel–Crafts Alkylation of Indoles with Ethyl 3,3,3‐Trifluoropyruvate

(2008) Shuichi Nakamura et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Enantioselective Zirconium-Catalyzed Friedel−Crafts Alkylation of Pyrrole with Trifluoromethyl Ketones

(2008) Gonzalo Blay et al.   ORGANIC LETTERS

Organocatalytic enantioselective Friedel–Crafts alkylation of simple phenols with trifluoropyruvate

(2008) Jun-Ling Zhao et al.   TETRAHEDRON LETTERS

Enantioselective synthesis of naphthopyran derivatives catalyzed by bifunctional thiourea-tertiary amines

(2008) Xiao-Sheng Wang et al.   TETRAHEDRON-ASYMMETRY

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS