Cetirizine and Levetiracetam as Inhibitors of Monoacylglycerol Lipase: Investigating Their Repurposing Potential as Novel Osteoarthritic Pain Therapies
出版年份 2023 全文链接
标题
Cetirizine and Levetiracetam as Inhibitors of Monoacylglycerol Lipase: Investigating Their Repurposing Potential as Novel Osteoarthritic Pain Therapies
作者
关键词
-
出版物
Pharmaceuticals
Volume 16, Issue 11, Pages 1563
出版商
MDPI AG
发表日期
2023-11-06
DOI
10.3390/ph16111563
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Monoacylglycerol Lipase Inhibitor JJKK048 Ameliorates ABCG2 Transporter-Mediated Regorafenib Resistance Induced by Hypoxia in Triple Negative Breast Cancer Cells
- (2023) Elena Puris et al. JOURNAL OF PHARMACEUTICAL SCIENCES
- Inhibition of Monoacylglycerol Lipase Decreases Angiogenic Features of Endothelial Cells via Release of Tissue Inhibitor of Metalloproteinase-1 from Lung Cancer Cells
- (2023) Felix Wittig et al. Cells
- Pristimerin, a triterpene that inhibits monoacylglycerol lipase activity, prevents the development of paclitaxel-induced allodynia in mice
- (2022) Altaf Al-Romaiyan et al. Frontiers in Pharmacology
- Pharmacological activation of mediodorsal thalamic GABA-A receptors modulates morphine/cetirizine-induced changes in the prefrontal cortical GFAP expression in a rat model of neuropathic pain
- (2022) Niyusha Asgharpour-Masouleh et al. BEHAVIOURAL BRAIN RESEARCH
- ‘SMASH’ recommendations for standardised microscopic arthritis scoring of histological sections from inflammatory arthritis animal models
- (2021) Silvia Hayer et al. ANNALS OF THE RHEUMATIC DISEASES
- Anticancer Potential of Small‐Molecule Inhibitors of Fatty Acid Amide Hydrolase and Monoacylglycerol Lipase
- (2021) Shivani Jaiswal et al. ChemMedChem
- Targeting Monoacylglycerol Lipase in Pursuit of Therapies for Neurological and Neurodegenerative Diseases
- (2021) Anca Zanfirescu et al. MOLECULES
- The burden of OA-health services and economics
- (2021) V.P. Leifer et al. OSTEOARTHRITIS AND CARTILAGE
- Identifying FAAH Inhibitors as New Therapeutic Options for the Treatment of Chronic Pain through Drug Repurposing
- (2021) Anca Zanfirescu et al. Pharmaceuticals
- Andrographolide ameliorates oxidative stress, inflammation and histological outcome in complete Freund's adjuvant-induced arthritis
- (2020) Shasha Luo et al. CHEMICO-BIOLOGICAL INTERACTIONS
- An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present)
- (2020) Giulia Bononi et al. EXPERT OPINION ON THERAPEUTIC PATENTS
- Histamine, histamine receptors and neuropathic pain relief
- (2019) Ilona Obara et al. BRITISH JOURNAL OF PHARMACOLOGY
- Therapeutic options for targeting inflammatory osteoarthritis pain
- (2019) Philip G. Conaghan et al. Nature Reviews Rheumatology
- Mitodepressive, antioxidant, antifungal and anti-inflammatory effects of wild-growing Romanian native Arctium lappa L. ( Asteraceae ) and Veronica persica Poiret ( Plantaginaceae )
- (2018) Radu Claudiu Fierascu et al. FOOD AND CHEMICAL TOXICOLOGY
- Design, synthesis, and evaluation of piperazinyl pyrrolidin-2-ones as a novel series of reversible monoacylglycerol lipase inhibitors
- (2018) Jumpei Aida et al. JOURNAL OF MEDICINAL CHEMISTRY
- Chronic Monosodium Glutamate Administration Induced Hyperalgesia in Mice
- (2017) Anca Zanfirescu et al. Nutrients
- Methods Used to Evaluate Pain Behaviors in Rodents
- (2017) Jennifer R. Deuis et al. Frontiers in Molecular Neuroscience
- Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain
- (2016) Margherita Brindisi et al. JOURNAL OF MEDICINAL CHEMISTRY
- Randall Selitto pressure algometry for assessment of bone-related pain in rats
- (2015) S. Falk et al. EUROPEAN JOURNAL OF PAIN
- The effect of FAAH, MAGL, and Dual FAAH/MAGL inhibition on inflammatory and colorectal distension-induced visceral pain models in Rodents
- (2015) Y. S. Sakin et al. NEUROGASTROENTEROLOGY AND MOTILITY
- In vivocharacterization of the highly selective monoacylglycerol lipase inhibitor KML29: antinociceptive activity without cannabimimetic side effects
- (2013) B M Ignatowska-Jankowska et al. BRITISH JOURNAL OF PHARMACOLOGY
- The adverse effects profile of levetiracetam in epilepsy: a more detailed look
- (2013) Gashirai K. Mbizvo et al. INTERNATIONAL JOURNAL OF NEUROSCIENCE
- Levetiracetam Interacts Synergistically With Nonsteroidal Analgesics and Caffeine to Produce Antihyperalgesia in Rats
- (2013) Maja A. Tomić et al. JOURNAL OF PAIN
- KIAA1199, a deafness gene of unknown function, is a new hyaluronan binding protein involved in hyaluronan depolymerization
- (2013) H. Yoshida et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- The Local Peripheral Antihyperalgesic Effect of Levetiracetam and Its Mechanism of Action in an Inflammatory Pain Model
- (2012) Radica M. Stepanović-Petrović et al. ANESTHESIA AND ANALGESIA
- The antinociceptive triterpene β-amyrin inhibits 2-arachidonoylglycerol (2-AG) hydrolysis without directly targeting cannabinoid receptors
- (2012) A Chicca et al. BRITISH JOURNAL OF PHARMACOLOGY
- The Endocannabinoid System and Pain
- (2012) Josee Guindon et al. CNS & Neurological Disorders-Drug Targets
- The monoacylglycerol lipase inhibitor JZL184 suppresses inflammatory pain in the mouse carrageenan model
- (2012) Sudeshna Ghosh et al. LIFE SCIENCES
- Physiological roles of 2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand
- (2009) Takayuki Sugiura BIOFACTORS
- AutoDock Vina: Improving the speed and accuracy of docking with a new scoring function, efficient optimization, and multithreading
- (2009) Oleg Trott et al. JOURNAL OF COMPUTATIONAL CHEMISTRY
- Analgesic Effects Of H1 Receptor Antagonists In The Rat Model Of Formalin-Induced Pain
- (2009) Hazem Adel Ashmawi et al. Revista Brasileira de Anestesiologia
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