Catalyst-Controlled Divergent Reactions of 2,3-Disubstituted Indoles with Propargylic Alcohols: Synthesis of 3H-Benzo[b]azepines and Axially Chiral Tetrasubstituted Allenes

Chiral phosphoric acid-catalyzed regio- and enantioselective reactions of functionalized propargylic alcohols

(2022) Chenxiao Qian et al.   Organic Chemistry Frontiers

Recent Advances in Organocatalytic Enantioselective Synthesis of Axially Chiral Allenes

(2022) Xing Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Design of an Organocatalytic Asymmetric (4 + 3) Cycloaddition of 2-Indolylalcohols with Dienolsilanes

(2022) Jie Ouyang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Enantioselective 1,10-Addition of Alkynyl Indole Imine Methides with Thiazolones: An Access to Axially Chiral Tetrasubstituted Allenes

(2022) Xiao Lin et al.   ORGANIC LETTERS

Design and synthesis of axially chiral aryl-pyrroloindoles via the strategy of organocatalytic asymmetric (2 + 3) cyclization

(2022) Ping Wu et al.   Fundamental Research

Organocatalytic Enantioselective aza‐Michael Addition of Arylamines to 7‐Methide‐7H‐indoles

(2021) Fushuai Li et al.   ADVANCED SYNTHESIS & CATALYSIS

Dearomatization of 2,3-Disubstituted Indoles via 1,8-Addition of Propargylic (Aza)-para-Quinone Methides

(2021) Han-Peng Pan et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Enantioselective Construction of Axially Chiral Tetrasubstituted Allenes via 1,6‐Addition of Alkynyl Indole Imine Methides with 2‐Substituted Indoles

(2021) Yu Wu et al.   Asian Journal of Organic Chemistry

Allylic and Allenylic Dearomatization of Indoles promoted by Graphene Oxide via Covalent Grafting Activation Mode

(2020) Marco Bandini et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic Enantioselective Synthesis of Chiral Allenes: Remote Asymmetric 1,8‐Addition of Indole Imine Methides

(2020) Xingguang Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Formal (3 + 2) Cycloaddition toward Chiral Pyrrolo[1,2-a]indoles via Dynamic Kinetic Resolution of Allene Intermediates

(2020) Jian-Fei Bai et al.   ORGANIC LETTERS

Organocatalytic Regio- and Enantioselective 1,8-Additions of Nitrogen and Sulfur Nucleophiles to 6-Methylene-6H-indoles

(2020) Qianqian Song et al.   ORGANIC LETTERS

Enantioselective Dehydrative γ-Arylation of α-Indolyl Propargylic Alcohols with Phenols: Access to Chiral Tetrasubstituted Allenes and Naphthopyrans

(2020) Wen-Run Zhu et al.   ORGANIC LETTERS

Recent Advances in the Synthesis of Heterocyclics via Cascade Cyclization of Propargylic Alcohols

(2020) Xian‐Rong Song et al.   ADVANCED SYNTHESIS & CATALYSIS

Remote Stereocontrolled Construction of Vicinal Axially Chiral Tetrasubstituted Allenes and Heteroatom-Functionalized Quaternary Carbon Stereocenters

(2019) Pei Zhang et al.   ORGANIC LETTERS

2-Propargyl alcohols in Organic Synthesis

(2019) Hongwei Qian et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Synthesis of Chiral 1,4-Enynes through Organocatalytic Alkenylation of Propargyl Alcohols with Trialkenylboroxines

(2019) Jian-Fei Bai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Enantioconvergent Synthesis of Tetrasubstituted Allenes via Asymmetric 1,8-Addition to aza-para-Quinone Methides

(2019) Min Chen et al.   ORGANIC LETTERS

Organocatalytic Remote Stereocontrolled 1,8-Additions of Thiazolones to Propargylic Aza-p-quinone Methides

(2019) Lili Zhang et al.   ORGANIC LETTERS

Organocatalytic Enantioselective Synthesis of Tetrasubstituted α-Amino Allenoates by Dearomative γ-Addition of 2,3-Disubstituted Indoles to β,γ-Alkynyl-α-imino Esters

(2019) Junxian Yang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric Synthesis of Indole-Based Chiral Heterocycles: Strategies, Reactions, and Outreach

(2019) Yu-Chen Zhang et al.   ACCOUNTS OF CHEMICAL RESEARCH

Chiral Phosphoric Acid Catalyzed Asymmetric Synthesis of Hetero-triarylmethanes from Racemic Indolyl Alcohols

(2018) Caizhen Yue et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Harnessing the Polarizability of Conjugated Alkynes toward [2 + 2] Cycloaddition, Alkenylation, and Ring Expansion of Indoles

(2018) Tapas R. Pradhan et al.   ORGANIC LETTERS

Indolylmethanols as Reactants in Catalytic Asymmetric Reactions

(2017) Guang-Jian Mei et al.   JOURNAL OF ORGANIC CHEMISTRY

BF3-Promoted Divergent Reactions between Tryptophols and Propargylic Alcohols

(2017) Kai Huang et al.   ORGANIC LETTERS

Organocatalytic synthesis of chiral tetrasubstituted allenes from racemic propargylic alcohols

(2017) Deyun Qian et al.   Nature Communications

Catalyst-Controlled Chemoselective and Enantioselective Reactions of Tryptophols with Isatin-Derived Imines

(2017) Fei Jiang et al.   ACS Catalysis

Indoles — A promising scaffold for drug development

(2016) T.V. Sravanthi et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

Recent Advances in Chiral Phosphoric Acid Catalyzed Asymmetric Reactions for the Synthesis of Enantiopure Indole Derivatives

(2015) Hua Wu et al.   SYNTHESIS-STUTTGART

Brønsted Acid Mediated Alkenylation and Copper-Catalyzed Aerobic Oxidative Ring Expansion/Intramolecular Electrophilic Substitution of Indoles with Propargyl Alcohols: A Novel One-Pot Approach to Cyclopenta[c]quinolines

(2014) G. Gangadhararao et al.   ORGANIC LETTERS

Update 1 of: Synthesis and Functionalization of Indoles Through Palladium-Catalyzed Reactions

(2011) Sandro Cacchi et al.   CHEMICAL REVIEWS

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Transition Metal-Catalysed, Direct and Site-Selective N1-, C2- or C3-Arylation of the Indole Nucleus: 20 Years of Improvements

(2009) Lionel Joucla et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION