Asymmetric Synthesis of Spiro[Azetidine‐3,3′‐Indoline]‐2,2′‐Diones via Copper(I)‐Catalyzed Kinugasa/C−C Coupling Cascade Reaction

Visible Light‐Mediated Dearomative Hydrogen Atom Abstraction/ Cyclization Cascade of Indoles

(2022) Yang Xiong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Diastereoselective [3 + 1] Cyclization Reaction of Oxindolyl Azaoxyallyl Cations with Sulfur Ylides: Assembly of 3,3′-Spiro[β-lactam]-oxindoles

(2021) Hai-Jun Leng et al.   ORGANIC LETTERS

Modular Synthesis of α‐Quaternary Chiral β‐Lactams by a Synergistic Copper/Palladium‐Catalyzed Multicomponent Reaction

(2021) Jialin Qi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Mechanism of the Kinugasa Reaction Revisited

(2021) Stefano Santoro et al.   JOURNAL OF ORGANIC CHEMISTRY

Access to Triazolopiperidine Derivatives via Copper(I)‐Catalyzed [3+2] Cycloaddition/Alkenyl C−N Coupling Tandem Reactions

(2021) Guorong Xiao et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper(I)‐Catalyzed Interrupted Click/Sulfenylation Cascade: One‐Pot Synthesis of Sulfur Cycle Fused 1,2,3‐Triazoles

(2020) Weiguo Wang et al.   CHINESE JOURNAL OF CHEMISTRY

Copper(I)‐Catalyzed Asymmetric Interrupted Kinugasa Reaction: Synthesis of α‐Thiofunctional Chiral β‐Lactams

(2020) Jialin Qi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric synthesis of spirooxindole β-lactams via isothiourea-catalyzed Mannich/lactamization reaction of aryl acetic acids with isatin-derived ketimines

(2019) Jing-Hai Jin et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Exclusively 4-Substituted β-Lactams through the Kinugasa Reaction Utilizing Calcium Carbide

(2019) Abolfazl Hosseini et al.   ORGANIC LETTERS

Intramolecular Copper(I)-Catalyzed Interrupted Click/Acylation Domino Reaction

(2019) Egor M. Larin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Synthesis of Spirocyclic β-Lactams through Copper-Catalyzed Kinugasa/Michael Domino Reactions

(2018) Tao Shu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic asymmetric synthesis of spirooxindoles: recent developments

(2018) Guang-Jian Mei et al.   CHEMICAL COMMUNICATIONS

New development in the enantioselective synthesis of spiro compounds

(2018) Aishun Ding et al.   CHEMICAL SOCIETY REVIEWS

A Revised Mechanism for the Kinugasa Reaction

(2018) Thomas C. Malig et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Discovery of 3,3′-Spiro[Azetidine]-2-oxo-indoline Derivatives as Fusion Inhibitors for Treatment of RSV Infection

(2018) Weihua Shi et al.   ACS Medicinal Chemistry Letters

Bench-Stable 5-Stannyl Triazoles by a Copper(I)-Catalyzed Interrupted Click Reaction: Bridge to Trifluoromethyltriazoles and Trifluoromethylthiotriazoles

(2017) Fang Wei et al.   ORGANIC LETTERS

Regioselective synthesis of multisubstituted 1,2,3-triazoles: moving beyond the copper-catalyzed azide–alkyne cycloaddition

(2016) Fang Wei et al.   CHEMICAL COMMUNICATIONS

Studies on the Enantioselective Kinugasa Reaction: Efficient Synthesis of β-Lactams Catalyzed byN-PINAP/CuX Complexes

(2016) Karol Wolosewicz et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper(I)-Catalyzed Three-Component Click/Alkynylation: One-Pot Synthesis of 5-Alkynyl-1,2,3-triazoles

(2016) Weiguo Wang et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Three-Component Coupling ofN-Tosylhydrazones, Alkynes and Azides: Synthesis of Trisubstituted 1,2,3-Triazoles

(2015) Zhikun Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper(I)-Catalyzed Interrupted Click Reaction: Synthesis of Diverse 5-Hetero-Functionalized Triazoles

(2015) Weiguo Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Theoretical Study of Mechanism and Stereoselectivity of Catalytic Kinugasa Reaction

(2015) Stefano Santoro et al.   JOURNAL OF ORGANIC CHEMISTRY

Mild Cu(I)-Catalyzed Cascade Reaction of Cyclic Diaryliodoniums, Sodium Azide, and Alkynes: Efficient Synthesis of Triazolophenanthridines

(2014) Zhenquan Liu et al.   ORGANIC LETTERS

Bifunctional N-Heterocyclic Carbene-Catalyzed Highly Enantioselective Synthesis of Spirocyclic Oxindolo-β-lactams

(2014) Han-Ming Zhang et al.   ORGANIC LETTERS

Preparation of 1,4,5-Trisubstituted 5-Acyl-1,2,3-triazoles by Selective Acylation between Copper(I)-Carbon(sp) and Copper(I)-Carbon(sp2) Bonds with Acyl Chlorides

(2013) Bo Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Towards a General Synthesis of 3-Metal-Substituted β-Lactams

(2013) Beatriz Baeza et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric Synthesis oftrans-β-Lactams by a Kinugasa Reaction on Water

(2013) Zhenling Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Tandem Reaction of 1-Copper(I) Alkynes for the Synthesis of 1,4,5-Trisubstituted 5-Chloro-1,2,3-triazoles

(2013) Bo Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Easy preparation of 1,4,5-trisubstituted 5-(2-alkoxy-1,2-dioxoethyl)-1,2,3-triazoles by chemoselective trapping of copper(I)–carbon bond with alkoxalyl chloride

(2013) Bo Wang et al.   TETRAHEDRON LETTERS

Isatins As Privileged Molecules in Design and Synthesis of Spiro-Fused Cyclic Frameworks

(2012) Girija S. Singh et al.   CHEMICAL REVIEWS

Synthesis of [1,2,3]Triazolo[1,5-a]quinoxalin-4(5H)-ones through Copper-Catalyzed Tandem Reactions of N-(2-Haloaryl)propiolamides with Sodium Azide

(2012) Jiajie Yan et al.   ORGANIC LETTERS

A CuAAC/Ullmann C–C Coupling Tandem Reaction: Copper-Catalyzed Reactions of Organic Azides with N-(2-Iodoaryl)propiolamides or 2-Iodo-N-(prop-2-ynyl)benzenamines

(2012) Qian Cai et al.   ORGANIC LETTERS

Asymmetric Kinugasa reaction involving six-membered cyclic nitrones

(2012) Barbara Grzeszczyk et al.   TETRAHEDRON

Copper-catalysed approach to spirocyclic oxindoles via a direct C–H, Ar-H functionalisation

(2012) Catherine L. Moody et al.   TETRAHEDRON LETTERS

Copper-Catalyzed Tandem Reaction of Isocyanides withN-(2-Haloaryl)propiolamides for the Synthesis of Pyrrolo[3,2-c]quinolin-4-ones

(2011) Fengtao Zhou et al.   JOURNAL OF ORGANIC CHEMISTRY

A Formal Synthesis of Ezetimibe via Cycloaddition/Rearrangement Cascade Reaction

(2011) Michał Michalak et al.   JOURNAL OF ORGANIC CHEMISTRY

CuBr-NCS-Mediated Multicomponent Azide-Alkyne Cycloaddition: Mild and Efficient Synthesis of 5-Bromo-1,4-Disubstituted-1,2,3-Triazoles

(2011) Lingjun Li et al.   SYNLETT

The future of the β-lactams

(2010) Leticia I Llarrull et al.   CURRENT OPINION IN MICROBIOLOGY

Design, synthesis and in vitro antibacterial and antifungal activities of some novel spiro[azetidine-2,3′-indole]-2,4(1′H)-dione

(2010) Ravi J. Shah et al.   MEDICINAL CHEMISTRY RESEARCH

Copper-Catalyzed Tandem Reactions of 1-(2-Iodoary)-2-yn-1-ones with Isocyanides for the Synthesis of 4-Oxo-indeno[1,2-b]pyrroles

(2010) Qian Cai et al.   ORGANIC LETTERS

Studies of multicomponent Kinugasa reactions in aqueous media

(2009) Craig S. McKay et al.   TETRAHEDRON LETTERS

A Convenient Preparation of 5-Iodo-1,4-disubstituted-1,2,3-triazole: Multicomponent One-Pot Reaction of Azide and Alkyne Mediated by CuI−NBS

(2008) Lingjun Li et al.   JOURNAL OF ORGANIC CHEMISTRY