Doubly stereoconvergent crystallization enabled by asymmetric catalysis

A Pd-Catalyzed [4 + 2] Annulation Approach to Fluorinated N-Heterocycles

(2021) Víctor García-Vázquez et al.   ORGANIC LETTERS

State of the Art in Crystallization‐Induced Diastereomer Transformations

(2021) Andrej Kolarovič et al.   ADVANCED SYNTHESIS & CATALYSIS

The application of modern reactions in large-scale synthesis

(2021) Kaitlyn Lovato et al.   Nature Reviews Chemistry

BIMP‐Catalyzed 1,3‐Prototropic Shift for the Highly Enantioselective Synthesis of Conjugated Cyclohexenones

(2020) Jonathan C. Golec et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Modular Tuning of Electrophilic Reactivity of Iridium Nitrenoids for the Intermolecular Selective α-Amidation of β-Keto Esters

(2020) Minhan Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bifunctional Iminophosphorane Superbase Catalysis: Applications in Organic Synthesis

(2020) Michele Formica et al.   ACCOUNTS OF CHEMICAL RESEARCH

Molecular Complexity as a Driver for Chemical Process Innovation in the Pharmaceutical Industry

(2019) Seb Caille et al.   JOURNAL OF ORGANIC CHEMISTRY

Curbing the costs of chemical manufacturing

(2019) Seb Caille   SCIENCE

Visible-Light-Driven N-Heterocyclic Carbene Catalyzed γ- and ϵ -Alkylation with Alkyl Radicals

(2019) Lei Dai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

SuFEx Chemistry of Thionyl Tetrafluoride (SOF4 ) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides, and Sulfonimidates

(2018) Bing Gao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stereodiversified Modular Synthesis of Non-planar Five-Membered Cyclic N -Hydroxylamidines: Reactivity Study and Application to the Synthesis of Cyclic Amidines

(2018) Mary Cruz Prieto-Ramírez et al.   ADVANCED SYNTHESIS & CATALYSIS

On the design of complex drug candidate syntheses in the pharmaceutical industry

(2017) Martin D. Eastgate et al.   Nature Reviews Chemistry

Asymmetric Synthesis of β-Amino Amides by Catalytic Enantioconvergent 2-Aza-Cope Rearrangement

(2015) C. Guy Goodman et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bifunctional Iminophosphorane Catalyzed Enantioselective Sulfa-Michael Addition to Unactivated α-Substituted Acrylate Esters

(2015) Alistair J. M. Farley et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

SHELXT– Integrated space-group and crystal-structure determination

(2015) George M. Sheldrick   Acta Crystallographica A-Foundation and Advances

Diazo- and Transition-Metal-Free CH Insertion: A Direct Synthesis of β-Lactams

(2014) Luis F. R. Gomes et al.   CHEMISTRY-A EUROPEAN JOURNAL

Bifunctional Iminophosphorane Organocatalysts for Enantioselective Synthesis: Application to the Ketimine Nitro-Mannich Reaction

(2013) Marta G. Núñez et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Aza-Michael-Michael Cascade Reactions: A Flexible Approach to 2,3,4-Trisubstituted Tetrahydroquinolines

(2012) Zhen-Xin Jia et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric and Diastereoselective Conjugate Addition Reactions: C–C Bond Formation at Large Scale

(2012) Gareth P. Howell   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Highly Asymmetric NHC-Catalyzed Hydroacylation of Unactivated Alkenes

(2011) Isabel Piel et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Expedient Synthesis of a 72-Membered Isoxazolino-β-ketoamide Library by a 2·3-Component Reaction

(2011) John M. Knapp et al.   ACS Combinatorial Science

Mechanism of Amido-Thiourea Catalyzed Enantioselective Imine Hydrocyanation: Transition State Stabilization via Multiple Non-Covalent Interactions

(2009) Stephan J. Zuend et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Synthesis of Functionalized Cyclopentanones via a Multicatalytic Secondary Amine/N-Heterocyclic Carbene Catalyzed Cascade Sequence

(2009) Stephen P. Lathrop et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Efficient Asymmetric Synthesis of Sitagliptin

(2009) Karl B. Hansen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-free Michael addition initiated multicomponent oxidative cyclodehydration route to polysubstituted pyridines from 1,3-dicarbonyls

(2008) Frédéric Liéby-Muller et al.   CHEMICAL COMMUNICATIONS