Differential Requirement of the Extracellular Domain in Activation of Class B G Protein-coupled Receptors
出版年份 2016 全文链接
标题
Differential Requirement of the Extracellular Domain in Activation of Class B G Protein-coupled Receptors
作者
关键词
-
出版物
JOURNAL OF BIOLOGICAL CHEMISTRY
Volume 291, Issue 29, Pages 15119-15130
出版商
American Society for Biochemistry & Molecular Biology (ASBMB)
发表日期
2016-05-14
DOI
10.1074/jbc.m116.726620
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Extra-helical binding site of a glucagon receptor antagonist
- (2016) Ali Jazayeri et al. NATURE
- Conformational states of the full-length glucagon receptor
- (2015) Linlin Yang et al. Nature Communications
- The non-peptide GLP-1 receptor agonist WB4-24 blocks inflammatory nociception by stimulating β-endorphin release from spinal microglia
- (2014) Hui Fan et al. BRITISH JOURNAL OF PHARMACOLOGY
- Structure of Class B GPCRs: new horizons for drug discovery
- (2014) Andrea Bortolato et al. BRITISH JOURNAL OF PHARMACOLOGY
- A potentiator of orthosteric ligand activity at GLP-1R acts via covalent modification
- (2014) Whitney M Nolte et al. Nature Chemical Biology
- Structure of class B GPCR corticotropin-releasing factor receptor 1
- (2013) Kaspar Hollenstein et al. NATURE
- Structure of the human glucagon class B G-protein-coupled receptor
- (2013) Fai Yiu Siu et al. NATURE
- A continued saga of Boc5, the first non-peptidic glucagon-like peptide-1 receptor agonist with in vivo activities
- (2012) Min He et al. ACTA PHARMACOLOGICA SINICA
- Structure and mechanism for recognition of peptide hormones by Class B G-protein-coupled receptors
- (2012) Kuntal Pal et al. ACTA PHARMACOLOGICA SINICA
- Small Molecule Drug Discovery at the Glucagon-Like Peptide-1 Receptor
- (2012) Francis S. Willard et al. Experimental Diabetes Research
- Molecular basis for negative regulation of the glucagon receptor
- (2012) C. M. Koth et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Fusion Partner Toolchest for the Stabilization and Crystallization of G Protein-Coupled Receptors
- (2012) Eugene Chun et al. STRUCTURE
- Cyclobutane Derivatives As Novel Nonpeptidic Small Molecule Agonists of Glucagon-Like Peptide-1 Receptor
- (2011) Qing Liu et al. JOURNAL OF MEDICINAL CHEMISTRY
- Crystal Structure of the PAC1R Extracellular Domain Unifies a Consensus Fold for Hormone Recognition by Class B G-Protein Coupled Receptors
- (2011) Shiva Kumar et al. PLoS One
- Structural insights into RAMP modification of secretin family G protein-coupled receptors: implications for drug development
- (2011) Julia K. Archbold et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- Non-peptidic glucose-like peptide-1 receptor agonists: aftermath of a serendipitous discovery
- (2010) Ming-wei Wang et al. ACTA PHARMACOLOGICA SINICA
- Novel Small Molecule Glucagon-Like Peptide-1 Receptor Agonist Stimulates Insulin Secretion in Rodents and From Human Islets
- (2010) K. W. Sloop et al. DIABETES
- Structural Basis for Hormone Recognition by the Human CRFR2α G Protein-coupled Receptor
- (2010) Kuntal Pal et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- NMR Structure of the First Extracellular Domain of Corticotropin-releasing Factor Receptor 1 (ECD1-CRF-R1) Complexed with a High Affinity Agonist
- (2010) Christy Rani R. Grace et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Allosteric Ligands of the Glucagon-Like Peptide 1 Receptor (GLP-1R) Differentially Modulate Endogenous and Exogenous Peptide Responses in a Pathway-Selective Manner: Implications for Drug Screening
- (2010) C. Koole et al. MOLECULAR PHARMACOLOGY
- Crystal Structure of Glucagon-like Peptide-1 in Complex with the Extracellular Domain of the Glucagon-like Peptide-1 Receptor
- (2009) Christina Rye Underwood et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Homozygous P86S Mutation of the Human Glucagon Receptor Is Associated With Hyperglucagonemia, α Cell Hyperplasia, and Islet Cell Tumor
- (2009) Cuiqi Zhou et al. PANCREAS
- Membrane-tethered ligands are effective probes for exploring class B1 G protein-coupled receptor function
- (2009) J.-P. Fortin et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Passing the baton in class B GPCRs: peptide hormone activation via helix induction?
- (2009) Christoph Parthier et al. TRENDS IN BIOCHEMICAL SCIENCES
- Molecular Recognition of Corticotropin-releasing Factor by Its G-protein-coupled Receptor CRFR1
- (2008) Augen A. Pioszak et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Molecular recognition of parathyroid hormone by its G protein-coupled receptor
- (2008) Augen A. Pioszak et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
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