VEGFR2 and hepatocellular carcinoma inhibitory activities of trisubstituted triazole derivatives
出版年份 2021 全文链接
标题
VEGFR2 and hepatocellular carcinoma inhibitory activities of trisubstituted triazole derivatives
作者
关键词
1,2,4-triazole derivatives, Anti-VEGFR2 activity, HepG2, HCC cell lines, THLE3
出版物
JOURNAL OF MOLECULAR STRUCTURE
Volume 1250, Issue -, Pages 131832
出版商
Elsevier BV
发表日期
2021-11-02
DOI
10.1016/j.molstruc.2021.131832
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Synthesis of antimicrobial azoloazines and molecular docking for inhibiting COVID ‐19
- (2021) Zeinab A. Muhammad et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- Discovery of thiazole-based-chalcones and 4-hetarylthiazoles as potent anticancer agents: Synthesis, docking study and anticancer activity
- (2020) Thoraya A. Farghaly et al. BIOORGANIC CHEMISTRY
- Structure-based drug repositioning explains ibrutinib as VEGFR2 inhibitor
- (2020) Melissa F. Adasme et al. PLoS One
- Synthesis, structure elucidation, DNA binding and molecular docking studies of novel copper(II) complexes of two 1,3,4‐thiadiazolethiosemicarbazone derivatives
- (2020) Khadiga M. Takroni et al. APPLIED ORGANOMETALLIC CHEMISTRY
- 1,2,4-Triazolin-5-thione derivatives with anticancer activity as CK1γ kinase inhibitors
- (2020) Monika Pitucha et al. BIOORGANIC CHEMISTRY
- Discovery of novel indolyl-1,2,4-triazole hybrids as potent vascular endothelial growth factor receptor-2 (VEGFR-2) inhibitors with potential anti-renal cancer activity
- (2020) Sami A. Al-Hussain et al. BIOORGANIC CHEMISTRY
- Nano-sized formazan analogues: Synthesis, structure elucidation, antimicrobial activity and docking study for COVID-19
- (2020) Huda K. Mahmoud et al. BIOORGANIC CHEMISTRY
- A new reactive Ketenaminal: Synthesis, coupling reaction, tautomeric study, docking and antimicrobial evaluation of the products
- (2019) Huda K. Mahmoud et al. Medicinal Chemistry
- New Insight into Therapies Targeting Angiogenesis in Hepatocellular Carcinoma
- (2019) Mossenta et al. Cancers
- Synthesis and Antimicrobial Evaluation of Novel Pyrazolopyrimidines Incorporated with Mono- and Diphenylsulfonyl Groups
- (2019) Alsaedi et al. MOLECULES
- New azoloazine derivatives as antimicrobial agents: Synthesis under microwave irradiations, structure elucidation, and antimicrobial activity
- (2019) Asmaa F. Kassem et al. JOURNAL OF HETEROCYCLIC CHEMISTRY
- Cytotoxicity , docking study of new fluorinated fused pyrimidine scaffold: Thermal and microwave irradiation synthesis
- (2019) Alaa M. Abo Alnaja et al. Medicinal Chemistry
- 3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
- (2018) Romeo Romagnoli et al. BIOORGANIC CHEMISTRY
- Anti-Angiogenics: Current Situation and Future Perspectives
- (2018) Katja Zirlik et al. Oncology Research and Treatment
- Apatinib targets both tumor and endothelial cells in hepatocellular carcinoma
- (2018) Chaoxu Yang et al. Cancer Medicine
- The Role of Angiogenesis in Hepatocellular Carcinoma
- (2018) Michael A. Morse et al. CLINICAL CANCER RESEARCH
- Design, selective alkylation and X-ray crystal structure determination of dihydro-indolyl-1,2,4-triazole-3-thione and its 3-benzylsulfanyl analogue as potent anticancer agents
- (2017) Ahmed T.A. Boraei et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Recent Developments on 1,2,4-Triazole Nucleus in Anticancer Compounds: A Review
- (2016) Ramandeep Kaur et al. Anti-Cancer Agents in Medicinal Chemistry
- Design, synthesis and biological evaluation of novel 3-alkylsulfanyl-4-amino-1,2,4-triazole derivatives
- (2016) Pei-Liang Zhao et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and antiproliferative evaluation of novel 2-(4 H -1,2,4-triazole-3-ylthio)acetamide derivatives as inducers of apoptosis in cancer cells
- (2016) Necla Kulabaş et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of Potent VEGFR-2 Inhibitors based on Furopyrimidine and Thienopyrimidne Scaffolds as Cancer Targeting Agents
- (2016) Marwa A. Aziz et al. Scientific Reports
- Recent advances bioactive 1,2,4-triazole-3-thiones
- (2015) Ş.Güniz Küçükgüzel et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis of novel 1,2,4-triazoles and triazolo-thiadiazines as anticancer agents
- (2015) Thoraya Abd El-Reheem FARGHALY et al. TURKISH JOURNAL OF CHEMISTRY
- Quantitation of VEGFR2 (vascular endothelial growth factor receptor) inhibitors - review of assay methodologies and perspectives
- (2014) Kuldeep Sharma et al. BIOMEDICAL CHROMATOGRAPHY
- Benzenesulfonamide bearing 1,2,4-triazole scaffolds as potent inhibitors of tumor associated carbonic anhydrase isoforms hCA IX and hCA XII
- (2014) SitaRam et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis and biological evaluation of N-(4-hydroxy-3-mercaptonaphthalen-1-yl)amides as inhibitors of angiogenesis and tumor growth
- (2013) Fuming Xu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Nonclassical antifolates, part 4. 5-(2-Aminothiazol-4-yl)-4-phenyl-4H-1,2,4-triazole-3-thiols as a new class of DHFR inhibitors: Synthesis, biological evaluation and molecular modeling study
- (2013) Ghada S. Hassan et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- One-pot synthesis of novel isoindoline-1,3-dione derivatives bearing 1,2,4-triazole moiety and their preliminary biological evaluation
- (2012) Pei-Liang Zhao et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Molecular conformations, interactions, and properties associated with drug efficiency and clinical performance among VEGFR TK inhibitors
- (2012) M. McTigue et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- VEGF and angiopoietin signaling in tumor angiogenesis and metastasis
- (2011) Pipsa Saharinen et al. TRENDS IN MOLECULAR MEDICINE
- Discovery of Dual VEGFR-2 and Tubulin Inhibitors with in Vivo Efficacy
- (2010) Eugene L. Piatnitski Chekler et al. ACS Medicinal Chemistry Letters
- VEGF and endothelial guidance in angiogenic sprouting
- (2010) Holger Gerhardt Organogenesis
- Anti-angiogenic tyrosine kinase inhibitors: what is their mechanism of action?
- (2009) Kristy J. Gotink et al. ANGIOGENESIS
- Sorafenib
- (2009) Gillian M. Keating et al. DRUGS
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