Direct Synthesis of 4-Aryl-1,2,3-triazoles via I2-Promoted Cyclization under Metal- and Azide-Free Conditions

A Scalable, Metal-, Azide- and Halogen-Free Method for the Preparation of Triazoles

(2020) Peter Clark et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Sulfenyl Ynamides in Gold Catalysis: Synthesis of Oxo‐functionalised 4‐aminoimidazolyl Fused Compounds by Intermolecular Annulation Reactions

(2020) Elsa M. Arce et al.   ADVANCED SYNTHESIS & CATALYSIS

Iodine-Mediated Condensation-Cyclization of α-Azido Ketones with p -Toluenesulfonyl Hydrazide for Synthesis of 4-Aryl-NH -1,2,3-Triazoles

(2020) Ming-Tian Ren et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Photocatalytic Vicinal Aminopyridylation of Methyl Ketones by a Double Umpolung Strategy

(2020) Honggu Im et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Selective 1,2‐Aminoisothiocyanation of 1,3‐Dienes Under Visible‐Light Photoredox Catalysis

(2020) Weisi Guo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Comprehensive review on the anti-bacterial activity of 1,2,3-triazole hybrids

(2019) Bo Zhang   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal-Free Cascade [4 + 1] Cyclization Access to 4-Aryl-NH-1,2,3-triazoles from N-Tosylhydrazones and Sodium Azide

(2019) Wen-Ming Shu et al.   JOURNAL OF ORGANIC CHEMISTRY

Regiospecific Three-Component Aminofluorination of Olefins via Photoredox Catalysis

(2018) Jia-Nan Mo et al.   ORGANIC LETTERS

Facile Synthesis of 1,3,5-Triarylbenzenes and 4-Aryl-NH -1,2,3-Triazoles Using Mesoporous Pd-MCM-41 as Reusable Catalyst

(2018) Arijit Saha et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Multicomponent Domino Reaction of 2-Bromobenzaldehydes, Aryl Methyl Ketones, and Sodium Azide: Access to 1H-[1,2,3]Triazolo[4,5-c]quinoline Derivatives

(2018) Cheng Xu et al.   JOURNAL OF ORGANIC CHEMISTRY

Assembly of a biocompatible triazole-linked gene by one-pot click-DNA ligation

(2017) Mikiembo Kukwikila et al.   Nature Chemistry

A mini review of the synthesis of poly-1,2,3-triazole-based functional materials

(2017) Jingpei Huo et al.   RSC Advances

Aluminium(III) Chloride-Catalyzed Three-Component Condensation of Aromatic Aldehydes, Nitroalkanes and Sodium Azide for the Synthesis of 4-Aryl-NH-1,2,3-triazoles

(2016) Qinquan Hu et al.   ADVANCED SYNTHESIS & CATALYSIS

A single-step acid catalyzed reaction for rapid assembly of NH-1,2,3-triazoles

(2016) Joice Thomas et al.   CHEMICAL COMMUNICATIONS

Reaction between Azidyl Radicals and Alkynes: A Straightforward Approach to NH -1,2,3-Triazoles

(2015) Long Hu et al.   CHEMISTRY-A EUROPEAN JOURNAL

I2–TBHP-Catalyzed Oxidative Cross-Coupling of N-Sulfonyl Hydrazones and Isocyanides to 5-Aminopyrazoles

(2015) Gopal Chandru Senadi et al.   ORGANIC LETTERS

Preparation of 1H-1,2,3-Triazoles by Cuprous Ion Mediated Cycloaddition of Terminal Alkyne and Sodium Azide

(2015) Li-Hui Lu et al.   JOURNAL OF THE CHINESE CHEMICAL SOCIETY

Metal-Free CN- and NN-Bond Formation: Synthesis of 1,2,3-Triazoles from Ketones,N-Tosylhydrazines, and Amines in One Pot

(2014) Zhengkai Chen et al.   CHEMISTRY-A EUROPEAN JOURNAL

p-Toluenesulfonic Acid Mediated 1,3-Dipolar Cycloaddition of Nitroolefins with NaN3 for Synthesis of 4-Aryl-NH-1,2,3-triazoles

(2014) Xue-Jing Quan et al.   ORGANIC LETTERS

Copper-Mediated Synthesis of 1,2,3-Triazoles fromN-Tosylhydrazones and Anilines

(2013) Zhengkai Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Click Chemistry for Drug Development and Diverse Chemical–Biology Applications

(2013) Prakasam Thirumurugan et al.   CHEMICAL REVIEWS

Development and Optimization of Piperidyl-1,2,3-Triazole Ureas as Selective Chemical Probes of Endocannabinoid Biosynthesis

(2013) Ku-Lung Hsu et al.   JOURNAL OF MEDICINAL CHEMISTRY

Catalytic Asymmetric Synthesis of Pyrroloindolines via a Rhodium(II)-Catalyzed Annulation of Indoles

(2013) Jillian E. Spangler et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Sulfonyl-1,2,3-Triazoles: Convenient Synthones for Heterocyclic Compounds

(2012) Mikhail Zibinsky et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Heterocyclic methylsulfone hydroxamic acid LpxC inhibitors as Gram-negative antibacterial agents

(2012) Laura A. McAllister et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Preparation of reusable Ag-decorated graphene oxide catalysts for decarboxylative cycloaddition

(2012) Ji Dang Kim et al.   JOURNAL OF MATERIALS CHEMISTRY

Rational Design of 4-Aryl-1,2,3-Triazoles for Indoleamine 2,3-Dioxygenase 1 Inhibition

(2012) Ute F. Röhrig et al.   JOURNAL OF MEDICINAL CHEMISTRY

Click Dendrimers and Triazole-Related Aspects: Catalysts, Mechanism, Synthesis, and Functions. A Bridge between Dendritic Architectures and Nanomaterials

(2011) Didier Astruc et al.   ACCOUNTS OF CHEMICAL RESEARCH

Intermolecular and Selective Synthesis of 2,4,5-Trisubstituted Oxazoles by a Gold-Catalyzed Formal [3+2] Cycloaddition

(2011) Paul W. Davies et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly N2-Selective Palladium-Catalyzed Arylation of 1,2,3-Triazoles

(2011) Satoshi Ueda et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Catalyzed Denitrogenative Transannulation: Converting Triazoles into Other Heterocyclic Systems

(2011) Buddhadeb Chattopadhyay et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structure–activity relationship and enzyme kinetic studies on 4-aryl-1H-1,2,3-triazoles as indoleamine 2,3-dioxygenase (IDO) inhibitors

(2011) Qiang Huang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Synthesis of 4-Aryl-1H-1,2,3-triazoles from 1,1-Dibromoalkenes and Sodium Azide

(2011) Xiaokun Wang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Click-generated triazole ureas as ultrapotent in vivo–active serine hydrolase inhibitors

(2011) Alexander Adibekian et al.   Nature Chemical Biology

Acid-catalyzed synthesis of 10-substituted triazolyl artemisinins and their growth inhibitory activity against various cancer cells

(2010) Sangtae Oh et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Click polymerization

(2010) Anjun Qin et al.   CHEMICAL SOCIETY REVIEWS

Click chemistry with DNA

(2010) Afaf H. El-Sagheer et al.   CHEMICAL SOCIETY REVIEWS

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

Marrying click chemistry with polymerization: expanding the scope of polymeric materials

(2009) Patricia L. Golas et al.   CHEMICAL SOCIETY REVIEWS

Bromo-DirectedN-2 Alkylation ofNH-1,2,3-Triazoles: Efficient Synthesis of Poly-Substituted 1,2,3-Triazoles

(2009) Xiao-jun Wang et al.   ORGANIC LETTERS

Conformational control in the regioselective synthesis of N-2-substituted-1,2,3-triazoles

(2008) Yunfeng Chen et al.   CHEMICAL COMMUNICATIONS