Formation of Kiss1R/GPER Heterocomplexes Negatively Regulates Kiss1R-mediated Signalling through Limiting Receptor Cell Surface Expression

Does GPER Really Function as a G Protein-Coupled Estrogen Receptor in vivo?

(2020) Jing Luo et al.   Frontiers in Endocrinology

GIP receptor suppresses PAC1 receptor‐mediated neuronal differentiation via formation of a receptor heterocomplex

(2020) Ran Ke et al.   JOURNAL OF NEUROCHEMISTRY

Crosstalk between Notch, HIF-1α and GPER in Breast Cancer EMT

(2018) Ernestina De Francesco et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Separating Actin-Dependent Chemokine Receptor Nanoclustering from Dimerization Indicates a Role for Clustering in CXCR4 Signaling and Function

(2018) Laura Martínez-Muñoz et al.   MOLECULAR CELL

Homocysteine directly interacts and activates the angiotensin II type I receptor to aggravate vascular injury

(2018) Tuoyi Li et al.   Nature Communications

Allosteric Modulation of GPCRs: New Insights and Potential Utility for Treatment of Schizophrenia and Other CNS Disorders

(2017) Daniel J. Foster et al.   NEURON

Inhibitory action of gonadotropin-inhibitory hormone on the signaling pathways induced by kisspeptin and vasoactive intestinal polypeptide in GnRH neuronal cell line, GT1-7

(2016) You Lee Son et al.   FASEB JOURNAL

PRESTO-Tango as an open-source resource for interrogation of the druggable human GPCRome

(2015) Wesley K Kroeze et al.   NATURE STRUCTURAL & MOLECULAR BIOLOGY

Nicolaus Copernicus and the rapid vascular responses to aldosterone

(2015) Matthias Barton et al.   TRENDS IN ENDOCRINOLOGY AND METABOLISM

PRESTO-Tango as an open-source resource for interrogation of the druggable human GPCRome

(2015) Wesley K Kroeze et al.   NATURE STRUCTURAL & MOLECULAR BIOLOGY

Transmembrane peptides as unique tools to demonstrate the in vivo action of a cross-class GPCR heterocomplex

(2014) Leo T. O. Lee et al.   FASEB JOURNAL

The kisspeptin-GnRH pathway in human reproductive health and disease

(2014) Karolina Skorupskaite et al.   HUMAN REPRODUCTION UPDATE

Disrupted Kisspeptin Signaling in GnRH Neurons Leads to Hypogonadotrophic Hypogonadism

(2014) Horacio J. Novaira et al.   MOLECULAR ENDOCRINOLOGY

GPER activates Notch signaling in breast cancer cells and cancer-associated fibroblasts (CAFs)

(2013) Marco Pupo et al.   INTERNATIONAL JOURNAL OF BIOCHEMISTRY & CELL BIOLOGY

Cross-talk between GPER and growth factor signaling

(2013) Rosamaria Lappano et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Applying Physics-Based Scoring to Calculate Free Energies of Binding for Single Amino Acid Mutations in Protein-Protein Complexes

(2013) Hege Beard et al.   PLoS One

Minireview: G Protein-Coupled Estrogen Receptor-1, GPER-1: Its Mechanism of Action and Role in Female Reproductive Cancer, Renal and Vascular Physiology

(2012) Edward J. Filardo et al.   ENDOCRINOLOGY

Hormonal Regulation of Female Reproduction

(2012) A. Christensen et al.   HORMONE AND METABOLIC RESEARCH

Position paper: The membrane estrogen receptor GPER – Clues and questions

(2012) Matthias Barton   STEROIDS

Mathematical Models for Quantitative Assessment of Bioluminescence Resonance Energy Transfer: Application to Seven Transmembrane Receptors Oligomerization

(2012) Luka Drinovec et al.   Frontiers in Endocrinology

Update 1 of: Computational Modeling Approaches to Structure–Function Analysis of G Protein-Coupled Receptors

(2011) Francesca Fanelli et al.   CHEMICAL REVIEWS

GPR30 Expression Is Required for the Mineralocorticoid Receptor–Independent Rapid Vascular Effects of Aldosterone

(2011) Robert Gros et al.   HYPERTENSION

Regulation of Embryonic Kidney Branching Morphogenesis and Glomerular Development by KISS1 Receptor (Gpr54) through NFAT2- and Sp1-mediated Bmp7 Expression

(2010) Tingfang Yi et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Time-resolved FRET between GPCR ligands reveals oligomers in native tissues

(2010) Laura Albizu et al.   Nature Chemical Biology

Regulation of GPR54 Signaling by GRK2 and β-Arrestin

(2009) Macarena Pampillo et al.   MOLECULAR ENDOCRINOLOGY

FireDock: a web server for fast interaction refinement in molecular docking

(2008) E. Mashiach et al.   NUCLEIC ACIDS RESEARCH