Highly fluorinated 2,3-dihydro-1,3,4-thiadiazole derivatives via [3+2]-cycloadditions of tertiary thioamides with nitrile imines derived from trifluoroacetonitrile

The Huisgen Reaction: Milestones of the 1,3‐Dipolar Cycloaddition

(2020) Martin Breugst et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A straightforward access to 3-trifluoromethyl-1H-indazoles via (3+2)-cycloaddition of arynes with nitrile imines derived from trifluoroacetonitrile

(2020) Anna Kowalczyk et al.   JOURNAL OF FLUORINE CHEMISTRY

Progress in intermolecular and intramolecular reactions of thioamides with diazo compounds and azides

(2019) Vasiliy Bakulev et al.   TETRAHEDRON LETTERS

Synthesis of 4-polyfluoroalkyl-1,3-dithiolanes via [3+2] cycloaddition of thiocarbonyl ylide to polyfluoroalkanethioamides

(2019) Sergiy S. Mykhaylychenko et al.   Chemistry of Heterocyclic Compounds

Fluorine‐Containing Drugs Approved by the FDA in 2018

(2019) Haibo Mei et al.   CHEMISTRY-A EUROPEAN JOURNAL

A novel access to 4-trifluoromethyl-1,3-thiazole derivatives via an intermediate thiocarbonyl ylide

(2019) Emilia Obijalska et al.   JOURNAL OF FLUORINE CHEMISTRY

Trapping of trifluoroacetonitrile imines with mercaptoacetaldehyde and mercaptocarboxylic acids: An access to fluorinated 1,3,4-thiadiazine derivatives via (3+3)-annulation

(2019) Greta Utecht-Jarzyńska et al.   JOURNAL OF FLUORINE CHEMISTRY

Polysubstituted 3-trifluoromethylpyrazoles: regioselective (3 + 2)-cycloaddition of trifluoroacetonitrile imines with enol ethers and functional group transformations

(2018) Greta Utecht et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A Straightforward Access to Trifluoromethylated Spirobipyrazolines through a Double (3+2)-Cycloaddition of Fluorinated Nitrile Imines with Alkoxyallenes

(2018) Marcin Jasiński et al.   SYNLETT

Unravelling the Mysteries of [3+2] Cycloaddition Reactions

(2018) Mar Ríos-Gutiérez et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Expected and unexpected results in reactions of fluorinated nitrile imines with (cyclo)aliphatic thioketones

(2017) Greta Utecht et al.   JOURNAL OF FLUORINE CHEMISTRY

First (3+2)-Cycloadditions of Thiochalcones as C=S Dipolarophiles: Efficient Synthesis of 1,3,4-Thiadiazoles via Reactions with Fluorinated Nitrile Imines

(2017) Grzegorz Mlostoń et al.   SYNTHESIS-STUTTGART

Trifluoromethylated 2,3-dihydro-1,3,4-thiadiazoles via the regioselective [3+2]-cycloadditions of fluorinated nitrile imines with aryl, hetaryl, and ferrocenyl thioketones

(2016) Grzegorz Mlostoń et al.   JOURNAL OF FLUORINE CHEMISTRY

Aryl, hetaryl, and ferrocenyl thioketones as versatile building blocks for exploration in the organic chemistry of sulfur

(2016) Grzegorz Mlostoń et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

Synthesis of 5-(polyfluoroalkyl)-1,3-thiazolidines from polyfluoroalkanethiocarboxylic acid derivatives

(2015) Sergiy S. Mykhaylychenko et al.   Chemistry of Heterocyclic Compounds

1,3,4-Thiadiazoles: A potent multi targeted pharmacological scaffold

(2015) Saqlain Haider et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Selenophen-2-yl-Substituted Thiocarbonyl Ylides - at the Borderline of Dipolar and Biradical Reactivity

(2015) Grzegorz Mlostoń et al.   HELVETICA CHIMICA ACTA

Tautomeric equilibrium in trifluoroacetaldehyde arylhydrazones

(2015) Agata Wojciechowska et al.   TETRAHEDRON

Selective thioacylation of amines in water: a convenient preparation of secondary thioamides and thiazolines

(2015) Uma Pathak et al.   RSC Advances

1,3,4-Thiadiazole: Synthesis, Reactions, and Applications in Medicinal, Agricultural, and Materials Chemistry

(2014) Yang Hu et al.   CHEMICAL REVIEWS

Trifluoromethylated Heterocycles

(2014) Andrei Gakh et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

1,3,4-Thiadiazole and its Derivatives: A Review on Recent Progress in Biological Activities

(2013) Abhishek Kumar Jain et al.   Chemical Biology & Drug Design

Oxidation and chlorination reactions of perfluoroketene-N,S-acetals

(2009) Sergiy S. Mykhaylychenko et al.   JOURNAL OF FLUORINE CHEMISTRY

First synthesis of 2-aminosubstituted-2-perfluoroalkyl-3,6-dihydro-2H-thiopyrans by hetero-Diels–Alder reactions of fluorinated thioamides under microwave heating

(2009) Sergey S. Mikhailichenko et al.   TETRAHEDRON LETTERS

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS