Design, synthesis and anti-diabetic activity of novel 1, 2, 3-triazole-5-carboximidamide derivatives as dipeptidyl peptidase-4 inhibitors

Synthesis and biological evaluation of triazole based uracil derivatives as novel DPP-4 inhibitors

(2016) Qing Li et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Design, Synthesis and Biological Evaluation of Imidazo[1,2-a]pyridine Derivatives as Novel DPP-4 Inhibitors

(2015) Qing Li et al.   Chemical Biology & Drug Design

Glucagon-like Peptide-1 (GLP-1) Analogs: Recent Advances, New Possibilities, and Therapeutic Implications

(2014) Bikash Manandhar et al.   JOURNAL OF MEDICINAL CHEMISTRY

A comparative study of the binding modes of recently launched dipeptidyl peptidase IV inhibitors in the active site

(2013) Mika Nabeno et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Synthesis and biological evaluation of pyrrolidine-2-carbonitrile and 4-fluoropyrrolidine-2-carbonitrile derivatives as dipeptidyl peptidase-4 inhibitors for the treatment of type 2 diabetes

(2013) Jiang Wang et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Empagliflozin, a novel selective sodium glucose cotransporter-2 (SGLT-2) inhibitor: characterisation and comparison with other SGLT-2 inhibitors

(2011) R. Grempler et al.   DIABETES OBESITY & METABOLISM

Linagliptin

(2011) Lesley J. Scott   DRUGS

Alogliptin

(2010) Lesley J. Scott   DRUGS

Sitagliptin

(2010) Sohita Dhillon   DRUGS

Vildagliptin

(2010) Gillian M. Keating   DRUGS

Design and Synthesis of Pyrimidinone and Pyrimidinedione Inhibitors of Dipeptidyl Peptidase IV

(2010) Zhiyuan Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

One-Pot Three-Step Synthesis of 1,2,3-Triazoles by Copper-Catalyzed Cycloaddition of Azides with Alkynes formed by a Sonogashira Cross-Coupling and Desilylation

(2010) Frédéric Friscourt et al.   ORGANIC LETTERS

Medicinal chemistry approaches to the inhibition of dipeptidyl peptidase-4 for the treatment of type 2 diabetes

(2009) Shrikanth H. Havale et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Diagnosis and Classification of Diabetes Mellitus

(2009)   DIABETES CARE

Saxagliptin

(2009) Sohita Dhillon et al.   DRUGS

Dipeptidyl peptidase IV (DPP IV) and related molecules in type 2 diabetes

(2008) Peter et al.   Frontiers in Bioscience-Landmark

Involvement of DPP-IV catalytic residues in enzyme-saxagliptin complex formation

(2008) William J. Metzler et al.   PROTEIN SCIENCE