Monoamine Oxidase Inhibitory Activity: Methyl- versus Chlorochalcone Derivatives

Identification of Indole-Based Chalcones: Discovery of a Potent, Selective, and Reversible Class of MAO-B Inhibitors

(2016) Rani Sasidharan et al.   ARCHIV DER PHARMAZIE

Potent and Selective Monoamine Oxidase-B Inhibitory Activity: Fluoro-vs. Trifluoromethyl-4-hydroxylated Chalcone Derivatives

(2016) Bijo Mathew et al.   CHEMISTRY & BIODIVERSITY

Synthesis, Biochemistry, and Computational Studies of Brominated Thienyl Chalcones: A New Class of Reversible MAO-B Inhibitors

(2016) Bijo Mathew et al.   ChemMedChem

Design and synthesis of novel chalcones as potent selective monoamine oxidase-B inhibitors

(2016) Arwa Hammuda et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Exploration of chlorinated thienyl chalcones: A new class of monoamine oxidase-B inhibitors

(2016) Bijo Mathew et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Discovery of New Chemical Entities for Old Targets: Insights on the Lead Optimization of Chromone-Based Monoamine Oxidase B (MAO-B) Inhibitors

(2016) Joana Reis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Screening of Human Monoamine Oxidase-A Inhibitor Effect of New 2-Pyrazoline and Hydrazone Derivatives

(2015) Begüm Evranos-Aksöz et al.   ARCHIV DER PHARMAZIE

Synthesis of a series of unsaturated ketone derivatives as selective and reversible monoamine oxidase inhibitors

(2015) Ji Won Choi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Monoamine oxidase inhibitory activities of heterocyclic chalcones

(2015) Corné Minders et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Development of fluorinated methoxylated chalcones as selective monoamine oxidase-B inhibitors: Synthesis, biochemistry and molecular docking studies

(2015) Bijo Mathew et al.   BIOORGANIC CHEMISTRY

Monoamine oxidase inhibitory activity of 2-aryl-4H-chromen-4-ones

(2015) Vishnu Nayak Badavath et al.   BIOORGANIC CHEMISTRY

Discovery of 3-Hydroxy-3-phenacyloxindole Analogues of Isatin as Potential Monoamine Oxidase Inhibitors

(2015) Rati K. P. Tripathi et al.   ChemMedChem

New Frontiers in Selective Human MAO-B Inhibitors

(2015) Simone Carradori et al.   JOURNAL OF MEDICINAL CHEMISTRY

Development of Fluorinated Thienylchalcones as Monoamine Oxidase-B Inhibitors: Design, Synthesis, Biological Evaluation and Molecular Docking Studies

(2015) Bijo Mathew et al.   LETTERS IN ORGANIC CHEMISTRY

Monoamine Oxidase Inhibition and Molecular Modeling Studies of Piperidyl-thienyl and 2-Pyrazoline Derivatives of Chalcones

(2015) Sumera Zaib et al.   Medicinal Chemistry

Quinolinyl-Thienyl Chalcones as Monoamine Oxidase Inhibitors and their In Silico Modeling Studies

(2015) Sumera Zaib et al.   Medicinal Chemistry

Synthesis and evaluation of 6-substituted 3-arylcoumarin derivatives as multifunctional acetylcholinesterase/monoamine oxidase B dual inhibitors for the treatment of Alzheimer’s disease

(2015) Zhi-Min Wang et al.   RSC Advances

Synthesis of some novel hydrazone and 2-pyrazoline derivatives: Monoamine oxidase inhibitory activities and docking studies

(2014) Begüm Evranos-Aksöz et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, Biological Evaluation, and Molecular Simulation of Chalcones and Aurones as Selective MAO-B Inhibitors

(2014) Nicole Morales-Camilo et al.   Chemical Biology & Drug Design

Recent developments in biological activities of chalcones: A mini review

(2014) Parvesh Singh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Update on the pharmacology of selective inhibitors of MAO-A and MAO-B: Focus on modulation of CNS monoamine neurotransmitter release

(2014) John P.M. Finberg   PHARMACOLOGY & THERAPEUTICS

Chromenylchalcones with inhibitory effects on monoamine oxidase B

(2013) Geunhyeong Jo et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Selected furanochalcones as inhibitors of monoamine oxidase

(2013) Sarel J. Robinson et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Inhibitor Design for Monoamine Oxidases

(2013) Rona R. Ramsay   CURRENT PHARMACEUTICAL DESIGN

Monoamine oxidase inhibitory activity of 3,5-biaryl-4,5-dihydro-1H-pyrazole-1-carboxylate derivatives

(2013) B. Vishnu Nayak et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

The interactions of caffeine with monoamine oxidase

(2013) Anél Petzer et al.   LIFE SCIENCES

Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors

(2010) Franco Chimenti et al.   BIOORGANIC & MEDICINAL CHEMISTRY

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

(2009) Garrett M. Morris et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY

Chalcones: A Valid Scaffold for Monoamine Oxidases Inhibitors

(2009) Franco Chimenti et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Stereochemical Identification, and Selective Inhibitory Activity against Human Monoamine Oxidase-B of 2-Methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones

(2008) Franco Chimenti et al.   JOURNAL OF MEDICINAL CHEMISTRY