Old drugs with new skills: fenoprofen as an allosteric enhancer at melanocortin receptor 3
出版年份 2016 全文链接
标题
Old drugs with new skills: fenoprofen as an allosteric enhancer at melanocortin receptor 3
作者
关键词
Inflammation, Arthritis, GPCR, Drug repositioning, Resolution of inflammation
出版物
CELLULAR AND MOLECULAR LIFE SCIENCES
Volume 74, Issue 7, Pages 1335-1345
出版商
Springer Nature
发表日期
2016-11-17
DOI
10.1007/s00018-016-2419-3
参考文献
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注意：仅列出部分参考文献，下载原文获取全部文献信息。- Can you teach old drugs new tricks?
- (2016) Nicola Nosengo NATURE
- Biased Agonism as a Novel Strategy To Harness the Proresolving Properties of Melanocortin Receptors without Eliciting Melanogenic Effects
- (2015) Trinidad Montero-Melendez et al. JOURNAL OF IMMUNOLOGY
- ACTH: The forgotten therapy
- (2015) Trinidad Montero-Melendez SEMINARS IN IMMUNOLOGY
- Resolution Pharmacology: Opportunities for Therapeutic Innovation in Inflammation
- (2015) Mauro Perretti et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- Association between Periodontal Disease and Inflammatory Arthritis Reveals Modulatory Functions by Melanocortin Receptor Type 3
- (2014) Trinidad Montero-Melendez et al. AMERICAN JOURNAL OF PATHOLOGY
- Melanocortin peptides protect chondrocytes from mechanically induced cartilage injury
- (2014) Magdalena K. Kaneva et al. BIOCHEMICAL PHARMACOLOGY
- Melanocortin Peptides: Potential Targets in Systemic Lupus Erythematosus
- (2014) Lisa Carole Loram et al. INFLAMMATION
- Positive allosteric modulators to peptide GPCRs: a promising class of drugs
- (2013) Tamas Bartfai et al. ACTA PHARMACOLOGICA SINICA
- Emerging paradigms in GPCR allostery: implications for drug discovery
- (2013) Denise Wootten et al. NATURE REVIEWS DRUG DISCOVERY
- Multiple Sclerosis, Relapses, and the Mechanism of Action of Adrenocorticotropic Hormone
- (2013) Amy Perrin Ross et al. Frontiers in Neurology
- Chondroprotective and anti-inflammatory role of melanocortin peptides in TNF-α activated human C-20/A4 chondrocytes
- (2012) Magdalena K Kaneva et al. BRITISH JOURNAL OF PHARMACOLOGY
- Gene expression signature-based approach identifies a pro-resolving mechanism of action for histone deacetylase inhibitors
- (2012) T Montero-Melendez et al. CELL DEATH AND DIFFERENTIATION
- Diagnosing the decline in pharmaceutical R&D efficiency
- (2012) Jack W. Scannell et al. NATURE REVIEWS DRUG DISCOVERY
- Treatment of Acute Relapses in Multiple Sclerosis
- (2012) Regina Berkovich Neurotherapeutics
- 2012 American College of Rheumatology guidelines for management of gout. Part 2: Therapy and antiinflammatory prophylaxis of acute gouty arthritis
- (2012) Dinesh Khanna et al. ARTHRITIS CARE & RESEARCH
- The Melanocortin Agonist AP214 Exerts Anti-Inflammatory and Proresolving Properties
- (2011) Trinidad Montero-Melendez et al. AMERICAN JOURNAL OF PATHOLOGY
- Melanocortin MC4 receptor agonists counteract late inflammatory and apoptotic responses and improve neuronal functionality after cerebral ischemia
- (2011) Luca Spaccapelo et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- Development of a high throughput screen for allosteric modulators of melanocortin-4 receptor signaling using a real time cAMP assay
- (2011) Jacques Pantel et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- The resolution of inflammation: the devil in the flask and in the details
- (2011) Charles N. Serhan FASEB JOURNAL
- Allosteric Modulation of Seven Transmembrane Spanning Receptors: Theory, Practice, and Opportunities for Central Nervous System Drug Discovery
- (2011) Bruce J. Melancon et al. JOURNAL OF MEDICINAL CHEMISTRY
- The renaissance of corticotropin therapy in proteinuric nephropathies
- (2011) Rujun Gong Nature Reviews Nephrology
- The Melanocortin System in Control of Inflammation
- (2011) Anna Catania et al. TheScientificWorldJOURNAL
- Melanocortins counteract inflammatory and apoptotic responses to prolonged myocardial ischemia/reperfusion through a vagus nerve-mediated mechanism
- (2010) Alessandra Ottani et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- Anti-inflammatory and antiosteoclastogenesis properties of endogenous melanocortin receptor type 3 in experimental arthritis
- (2010) Hetal B. Patel et al. FASEB JOURNAL
- ACTH protects against glucocorticoid-induced osteonecrosis of bone
- (2010) M. Zaidi et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Melanocortin peptides inhibit urate crystal-induced activation of phagocytic cells
- (2009) Franco Capsoni et al. ARTHRITIS RESEARCH & THERAPY
- Predominance of cyclooxygenase 1 over cyclooxygenase 2 in the generation of proinflammatory prostaglandins in autoantibody-driven K/BxN serum–transfer arthritis
- (2008) Mei Chen et al. ARTHRITIS AND RHEUMATISM
- Design and Microwave-Assisted Synthesis of Novel Macrocyclic Peptides Active at Melanocortin Receptors: Discovery of Potent and Selective hMC5R Receptor Antagonists
- (2008) Paolo Grieco et al. JOURNAL OF MEDICINAL CHEMISTRY
- A role for MC3R in modulating lung inflammation
- (2008) Stephen J. Getting et al. PULMONARY PHARMACOLOGY & THERAPEUTICS
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