Discovery of natural naphthoquinones as sortase A inhibitors and potential anti‐infective solutions against Staphylococcus aureus

Quinone skeleton as a new class of irreversible inhibitors against Staphylococcus aureus sortase A

(2018) Xiaochen Hou et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Molecular Docking and Screening Studies of New Natural Sortase A Inhibitors

(2017) Georgiana Nitulescu et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

New 2-Phenylthiazoles as Potential Sortase A Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

(2017) Smaranda Oniga et al.   MOLECULES

Burdock (Arctium lappa) Leaf Extracts Increase the In Vitro Antimicrobial Efficacy of Common Antibiotics on Gram-positive and Gram-negative Bacteria

(2017) Lucia Pirvu et al.   Open Chemistry

Structural Analysis of Sortase A Inhibitors

(2016) Georgiana Nitulescu et al.   MOLECULES

Optimizing the production of the biosurfactant lichenysin and its application in biofilm control

(2015) J. Coronel-León et al.   JOURNAL OF APPLIED MICROBIOLOGY

Sortase A Inhibitors: Recent Advances and Future Perspectives

(2015) Stella Cascioferro et al.   JOURNAL OF MEDICINAL CHEMISTRY

Streptococcus pyogenes Sortase Mutants Are Highly Susceptible to Killing by Host Factors Due to Aberrant Envelope Physiology

(2015) Assaf Raz et al.   PLoS One

Assessment of the potential health benefits of certain total extracts from Vitis vinifera, Aesculus hyppocastanum and Curcuma longa

(2015) DENISA MARGINĂ et al.   Experimental and Therapeutic Medicine

Ultrasound-assisted synthesis and anticancer evaluation of new pyrazole derivatives as cell cycle inhibitors

(2015) George Mihai Nitulescu et al.   Arabian Journal of Chemistry

Discovery and structure–activity relationship studies of irreversible benzisothiazolinone-based inhibitors against Staphylococcus aureus sortase A transpeptidase

(2014) Dmitrijs Zhulenkovs et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A New Approach to Radial Basis Function Approximation and Its Application to QSAR

(2014) Alexey V. Zakharov et al.   Journal of Chemical Information and Modeling

Sortase A: An ideal target for anti-virulence drug development

(2014) Stella Cascioferro et al.   MICROBIAL PATHOGENESIS

Antiinfective therapy with a small molecule inhibitor ofStaphylococcus aureussortase

(2014) Jie Zhang et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Learning from our mistakes: The ‘unknown knowns’ in fragment screening

(2013) Ben J. Davis et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery ofStaphylococcus aureusSortase A Inhibitors Using Virtual Screening and the Relaxed Complex Scheme

(2013) Albert H. Chan et al.   Chemical Biology & Drug Design

lazar: a modular predictive toxicology framework

(2013) Andreas Maunz et al.   Frontiers in Pharmacology

Beta-carboline alkaloids derived from the ascidian Synoicum sp.

(2012) Tae Hyung Won et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Substituent Effects on the Reactivity of Benzoquinone Derivatives with Thiols

(2012) Wilbes Mbiya et al.   CHEMICAL RESEARCH IN TOXICOLOGY

Sortase enzymes in Gram-positive bacteria

(2011) Thomas Spirig et al.   MOLECULAR MICROBIOLOGY

Sortase transpeptidases: Insights into mechanism, substrate specificity, and inhibition

(2010) Kathleen W. Clancy et al.   BIOPOLYMERS

Synthesis and structure activity relationship studies of novel Staphylococcus aureus Sortase A inhibitors

(2010) Bala Chandra Chenna et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Probing of the cis-5-phenyl proline scaffold as a platform for the synthesis of mechanism-based inhibitors of the Staphylococcus aureus sortase SrtA isoform

(2009) Konstantin V. Kudryavtsev et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery and structure–activity relationship analysis of Staphylococcus aureus sortase A inhibitors

(2009) Nuttee Suree et al.   BIOORGANIC & MEDICINAL CHEMISTRY