Iodine-Mediated Aryl C−H Amination for the Synthesis of Benzimidazoles and Pyrido[1,2-a ]benzimidazoles

Recent Development of Benzimidazole-Containing Antibacterial Agents

(2016) Di Song et al.   ChemMedChem

Iodine mediated intramolecular C2-amidative cyclization of indoles: a facile access to indole fused tetracycles

(2016) Sindhura Badigenchala et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Intramolecular Dearomative Oxidative Coupling of Indoles: A Unified Strategy for the Total Synthesis of Indoline Alkaloids

(2015) Weiwei Zi et al.   ACCOUNTS OF CHEMICAL RESEARCH

The Conversion of 4-Anilinoquinazoline- and 3-Aryl-4-imino-3,4-dihydro-quinazoline-2-carbonitriles into Benzo[4,5]imidazo[1,2-c]quinazoline-6-carbonitriles via Oxidative and Nonoxidative C–N Couplings

(2015) Styliana I. Mirallai et al.   JOURNAL OF ORGANIC CHEMISTRY

I2/KI-Mediated Oxidative N–N Bond Formation for the Synthesis of 1,5-Fused 1,2,4-Triazoles from N-Aryl Amidines

(2015) Lina Song et al.   JOURNAL OF ORGANIC CHEMISTRY

Biologically Active Benzimidazole Derivatives

(2015) Subramaniyan Arulmurugan et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Recent Advances in Iodine-Mediated Organic Reactions

(2015) Jinjin Zhao et al.   CHINESE JOURNAL OF ORGANIC CHEMISTRY

I2-Mediated Oxidative C–N Bond Formation for Metal-Free One-Pot Synthesis of Di-, Tri-, and Tetrasubstituted Pyrazoles from α,β-Unsaturated Aldehydes/Ketones and Hydrazines

(2014) Xinting Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2-Amino-1,3,4-oxadiazoles and 2-Amino-1,3,4-thiadiazoles via Sequential Condensation and I2-Mediated Oxidative C–O/C–S Bond Formation

(2014) Pengfei Niu et al.   JOURNAL OF ORGANIC CHEMISTRY

Oxidant-Switchable Selective Synthesis of 2-Aminobenzimidazoles via C–H Amination/Acetoxylation of Guanidines

(2014) Yue Chi et al.   ORGANIC LETTERS

C–H cycloamination of N-aryl-2-aminopyridines and N-arylamidines catalyzed by an in situ generated hypervalent iodine(iii) reagent

(2013) Yimiao He et al.   CHEMICAL COMMUNICATIONS

Iodine-mediated intramolecular amination of ketones: the synthesis of 2-acylindoles and 2-acylindolines by tuning N-protecting groups

(2013) Wen-Chao Gao et al.   CHEMICAL COMMUNICATIONS

A Cascade Coupling Strategy for One-Pot Total Synthesis of β-Carboline and Isoquinoline-Containing Natural Products and Derivatives

(2013) Yan-Ping Zhu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Novel Research Strategies of Benzimidazole Derivatives: A Review

(2013) Kuldipsinh Barot et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Iodobenzene Catalyzed C–H Amination of N-Substituted Amidines Using m-Chloroperbenzoic Acid

(2013) Santhosh Kumar Alla et al.   ORGANIC LETTERS

Synthesis of pyrido[1,2-a]benzimidazoles and other fused imidazole derivatives with a bridgehead nitrogen atom

(2013) Roman S Begunov et al.   RUSSIAN CHEMICAL REVIEWS

Molecular iodine-catalyzed multicomponent reactions: an efficient catalyst for organic synthesis

(2013) Yi-Ming Ren et al.   RSC Advances

Iodine-mediated regioselective C2-amination of indoles and a concise total synthesis of (±)-folicanthine

(2012) Ying-Xiu Li et al.   CHEMICAL COMMUNICATIONS

Synthesis of Benzimidazoles by PIDA-Promoted Direct C(sp2)H Imidation ofN-Arylamidines

(2012) Jinbo Huang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Developments in the Synthesis of Five- and Six-Membered Heterocycles Using Molecular Iodine

(2012) Prakash T. Parvatkar et al.   CHEMISTRY-A EUROPEAN JOURNAL

Highly Regioselective C–N Bond Formation through C–H Azolation of Indoles Promoted by Iodine in Aqueous Media

(2012) Wen-Bin Wu et al.   ORGANIC LETTERS

Direct One-Pot Synthesis of Luotonin F and Analogues via Rational Logical Design

(2012) Yan-ping Zhu et al.   ORGANIC LETTERS

Iodine-Mediated Intramolecular Electrophilic Aromatic Cyclization in Allylamines: A General Route to Synthesis of Quinolines, Pyrazolo[4,3-b]pyridines, and Thieno[3,2-b]pyridines

(2012) Harikrishna Batchu et al.   ORGANIC LETTERS

I2-promoted direct one-pot synthesis of 2-aryl-3-(pyridine-2-ylamino)imidazo[1,2-a]pyridines from aromatic ketones and 2-aminopyridines

(2012) Zhuan Fei et al.   TETRAHEDRON LETTERS

Palladium-catalyzed aerobic oxidative C–H amination: synthesis of 2-unsubstituted and 2-substituted N-aryl benzimidazoles

(2012) Rapolu Kiran Kumar et al.   RSC Advances

Synthesis of Heterocycles via Electrophilic Cyclization of Alkynes Containing Heteroatom

(2011) Benhur Godoi et al.   CHEMICAL REVIEWS

Molecular Iodine: Recent Application in Heterocyclic Synthesis

(2011) Hojat Veisi   CURRENT ORGANIC CHEMISTRY

Antimalarial Pyrido[1,2-a]benzimidazoles

(2011) Albert J. Ndakala et al.   JOURNAL OF MEDICINAL CHEMISTRY

The synthesis, characterization and optical properties of novel pyrido[1,2-a]benzimidazole derivatives

(2010) Yan Qing Ge et al.   DYES AND PIGMENTS

Optimization of Phenyl-Substituted Benzimidazole Carboxamide Poly(ADP-Ribose) Polymerase Inhibitors: Identification of (S)-2-(2-Fluoro-4-(pyrrolidin-2-yl)phenyl)-1H-benzimidazole-4-carboxamide (A-966492), a Highly Potent and Efficacious Inhibitor

(2010) Thomas D. Penning et al.   JOURNAL OF MEDICINAL CHEMISTRY

Iodine-Induced Regioselective C−C and C−N Bonds Formation ofN-Protected Indoles

(2010) Ying-Xiu Li et al.   JOURNAL OF ORGANIC CHEMISTRY

A Direct Intramolecular C−H Amination Reaction Cocatalyzed by Copper(II) and Iron(III) as Part of an Efficient Route for the Synthesis of Pyrido[1,2-a]benzimidazoles fromN-Aryl-2-aminopyridines

(2010) Honggen Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iodine-catalyzed transformation of molecules containing oxygen functional groups

(2010) Marjan Jereb et al.   TETRAHEDRON

Direct Imidation to Construct 1H-Benzo[d]imidazole through PdII-Catalyzed CH Activation Promoted by Thiourea

(2009) Qing Xiao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Molecular Iodine—An Expedient Reagent for Oxidative Aromatization Reactions of α,β-Unsaturated Cyclic Compounds

(2009) Malose Jack Mphahlele   MOLECULES

Molecular Iodine-Mediated Cyclization of Tethered Heteroatom-Containing Alkenyl or Alkynyl Systems

(2009) Malose Jack Mphahlele   MOLECULES

CH Functionalization/CN Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

(2008) Gordon Brasche et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of the Poly(ADP-ribose) Polymerase (PARP) Inhibitor 2-[(R)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide (ABT-888) for the Treatment of Cancer

(2008) Thomas D. Penning et al.   JOURNAL OF MEDICINAL CHEMISTRY