Supramolecular hosts that recognize methyllysines and disrupt the interaction between a modified histone tail and its epigenetic reader protein

A Fluorescence-Based Supramolecular Tandem Assay for Monitoring Lysine Methyltransferase Activity in Homogeneous Solution

(2012) Mara Florea et al.   CHEMISTRY-A EUROPEAN JOURNAL

Antibody-Free Reading of the Histone Code Using a Simple Chemical Sensor Array

(2012) Samuel A. Minaker et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Epigenetic protein families: a new frontier for drug discovery

(2012) Cheryl H. Arrowsmith et al.   NATURE REVIEWS DRUG DISCOVERY

Synthesis of New Trisulfonated Calix[4]arenes Functionalized at the Upper Rim, and Their Complexation with the Trimethyllysine Epigenetic Mark

(2012) Kevin D. Daze et al.   ORGANIC LETTERS

A bacteria colony-based screen for optimal linker combinations in genetically encoded biosensors

(2011) Andreas Ibraheem et al.   BMC BIOTECHNOLOGY

Biochemistry of anionic calix[n]arenes

(2011) Florent Perret et al.   CHEMICAL COMMUNICATIONS

Recognition of amino acids by functionalized calixarenes

(2011) Lucia Mutihac et al.   CHEMICAL SOCIETY REVIEWS

Small-Molecule Ligands of Methyl-Lysine Binding Proteins

(2011) J. Martin Herold et al.   JOURNAL OF MEDICINAL CHEMISTRY

Operational calixarene-based fluorescent sensing systems for choline and acetylcholine and their application to enzymatic reactions

(2011) Dong-Sheng Guo et al.   Chemical Science

A small molecule receptor that selectively recognizes trimethyl lysine in a histone peptide with native protein-like affinity

(2010) Lindsey A. Ingerman et al.   CHEMICAL COMMUNICATIONS

Recognition and Specificity Determinants of the Human Cbx Chromodomains

(2010) Lilia Kaustov et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Pharmacophore Screening of the Protein Data Bank for Specific Binding Site Chemistry

(2010) Valérie Campagna-Slater et al.   Journal of Chemical Information and Modeling

A review of calixarene applications in nuclear industries

(2010) Bahram Mokhtari et al.   JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY

Finding Inspiration in the Protein Data Bank to Chemically Antagonize Readers of the Histone Code

(2010) Valérie Campagna-Slater et al.   Molecular Informatics

Combined epigenetic therapy with the histone methyltransferase EZH2 inhibitor 3-deazaneplanocin A and the histone deacetylase inhibitor panobinostat against human AML cells

(2009) W. Fiskus et al.   BLOOD

A Simple Calixarene Recognizes Post-translationally Methylated Lysine

(2009) Cory S. Beshara et al.   CHEMBIOCHEM

Protein methyltransferases as a target class for drug discovery

(2009) Robert A. Copeland et al.   NATURE REVIEWS DRUG DISCOVERY

Cancer treatment of the future: Inhibitors of histone methyltransferases

(2008) Astrid Spannhoff et al.   INTERNATIONAL JOURNAL OF BIOCHEMISTRY & CELL BIOLOGY

Complexation of amino acids derivatives in water by calix[4]arene phosphonic acids

(2008) Joanna Dziemidowicz et al.   JOURNAL OF INCLUSION PHENOMENA AND MACROCYCLIC CHEMISTRY

Chemical Sensors Based on Cyclodextrin Derivatives

(2008) Tomoki Ogoshi et al.   SENSORS