Palladium-catalyzed coupling of functionalized primary and secondary amines with aryl and heteroaryl halides: two ligands suffice in most cases

A flow-based synthesis of Imatinib: the API of Gleevec

(2010) Mark D. Hopkin et al.   CHEMICAL COMMUNICATIONS

Switching the Chemoselectivity in the Amination of 4-Chloroquinazolines with Aminopyrazoles

(2010) Zhenlu Shen et al.   ORGANIC LETTERS

Recent Applications of Palladium-Catalyzed Coupling Reactions in the Pharmaceutical, Agrochemical, and Fine Chemical Industries

(2009) Christian Torborg et al.   ADVANCED SYNTHESIS & CATALYSIS

Triarylamine: a promising core unit for efficient photovoltaic materials

(2009) Zhijun Ning et al.   CHEMICAL COMMUNICATIONS

An Efficient Process for Pd-Catalyzed C−N Cross-Coupling Reactions of Aryl Iodides: Insight Into Controlling Factors

(2009) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of imatinib: a convergent approach revisited

(2009) Andrey S. Ivanov et al.   MONATSHEFTE FUR CHEMIE

An improved synthesis of N-aryl and N-heteroaryl substituted homopiperazines—from conventional thermal conditions to scaling-up using microwave heating

(2009) Uwe Schön et al.   TETRAHEDRON

Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

(2008) John F. Hartwig   ACCOUNTS OF CHEMICAL RESEARCH

Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles†

(2008) Dawei Ma et al.   ACCOUNTS OF CHEMICAL RESEARCH

Well-Defined N-Heterocyclic Carbenes−Palladium(II) Precatalysts for Cross-Coupling Reactions

(2008) Nicolas Marion et al.   ACCOUNTS OF CHEMICAL RESEARCH

Discovery of Selective Aminothiazole Aurora Kinase Inhibitors

(2008) Carsten B. Andersen et al.   ACS Chemical Biology

Biaryl Phosphane Ligands in Palladium-Catalyzed Amination

(2008) David S. Surry et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Evaluation of indazole-based compounds as a new class of potent KDR/VEGFR-2 inhibitors

(2008) David Bauer et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery of piperidine carboxamide TRPV1 antagonists

(2008) Wing S. Cheung et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Hole-transporting hydrazones

(2008) Ramūnas Lygaitis et al.   CHEMICAL SOCIETY REVIEWS

A Highly Active Catalyst for Pd-Catalyzed Amination Reactions: Cross-Coupling Reactions Using Aryl Mesylates and the Highly Selective Monoarylation of Primary Amines Using Aryl Chlorides

(2008) Brett P. Fors et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Reactive, General and Long-Lived Catalysts for Palladium-Catalyzed Amination of Heteroaryl and Aryl Chlorides, Bromides, and Iodides: Scope and Structure–Activity Relationships

(2008) Qilong Shen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A New Class of Easily Activated Palladium Precatalysts for Facile C−N Cross-Coupling Reactions and the Low Temperature Oxidative Addition of Aryl Chlorides

(2008) Mark R. Biscoe et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of End-Functionalized Polyanilines

(2008) Rienk Eelkema et al.   MACROMOLECULES

[(CyPF-tBu)PdCl2]: An Air-Stable, One-Component, Highly Efficient Catalyst for Amination of Heteroaryl and Aryl Halides

(2008) Qilong Shen et al.   ORGANIC LETTERS

A Facile Total Synthesis of Imatinib Base and Its Analogues

(2008) Yi-Feng Liu et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

N-Heterocyclic Carbenes (NHCs) ContainingN-C-Palladacycle Complexes: Synthesis and Reactivity in Aryl Amination Reactions

(2008) Julie Broggi et al.   ORGANOMETALLICS

Development of CXCR3 antagonists. Part 4: Discovery of 2-amino-(4-tropinyl)quinolines

(2007) Roland L. Knight et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS