Brain uptake and distribution of the dopamine D3/D2receptor partial agonist [11C]cariprazine: An in vivo positron emission tomography study in nonhuman primates

Endogenous Opioid Release in the Human Brain Reward System Induced by Acute Amphetamine Administration

(2012) Alessandro Colasanti et al.   BIOLOGICAL PSYCHIATRY

Current State of Agonist Radioligands for Imaging of Brain Dopamine D2/D3 Receptors In Vivo with Positron Emission Tomography

(2012) Sjoerd J. Finnema et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

In vitro pharmacology of aripiprazole, its metabolite and experimental dopamine partial agonists at human dopamine D2 and D3 receptors

(2011) Yoshihiro Tadori et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

(2011) István Gyertyán et al.   NEUROCHEMISTRY INTERNATIONAL

Occupancy of dopamine D2 and D3 and serotonin 5-HT1A receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography

(2011) Nicholas Seneca et al.   PSYCHOPHARMACOLOGY

Absolute abundances and affinity states of dopamine receptors in mammalian brain: A review

(2011) Paul Cumming   SYNAPSE

Affinity and selectivity of [11C]-(+)-PHNO for the D3 and D2 receptors in the rhesus monkey brain in vivo

(2011) Jean-Dominique Gallezot et al.   SYNAPSE

Antipsychotic Occupancy of Dopamine Receptors in Schizophrenia

(2010) Magdalena Nord et al.   CNS Neuroscience & Therapeutics

PW01-188 - Characterization of cariprazine (RGH-188) D3/D2 receptor occupancy in healthy volunteers and schizophrenic patients by positron emission tomography (PET)

(2010) I. Laszlovszky et al.   EUROPEAN PSYCHIATRY

Cariprazine (RGH-188), a Dopamine D3 Receptor-Preferring, D3/D2 Dopamine Receptor Antagonist-Partial Agonist Antipsychotic Candidate: In Vitro and Neurochemical Profile

(2010) B. Kiss et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Imaging dopamine receptors in humans with [11C]-(+)-PHNO: Dissection of D3 signal and anatomy

(2010) Andri C. Tziortzi et al.   NEUROIMAGE

In Vivo Binding of Antipsychotics to D3 and D2 Receptors: A PET Study in Baboons with [11C]-(+)-PHNO

(2010) Ragy R Girgis et al.   NEUROPSYCHOPHARMACOLOGY

Advancement in PET quantification using 3D-OP-OSEM point spread function reconstruction with the HRRT

(2009) Andrea Varrone et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

In vivo quantification of regional dopamine-D3 receptor binding potential of (+)-PHNO: Studies in non-human primates and transgenic mice

(2009) Eugenii A. Rabiner et al.   SYNAPSE

In-target produced [11C]methane: Increased specific radioactivity

(2008) Jan Andersson et al.   APPLIED RADIATION AND ISOTOPES