The Direct Actions of GABA, 2’-Methoxy-6-Methylflavone and General Anaesthetics at β3γ2L GABAA Receptors: Evidence for Receptors with Different Subunit Stoichiometries

Dopamine Directly Modulates GABAA Receptors

(2015) P. Hoerbelt et al.   JOURNAL OF NEUROSCIENCE

Non-equivalent Ligand Selectivity of Agonist Sites in (α4β2)2α4 Nicotinic Acetylcholine Receptors

(2014) Simone Mazzaferro et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Multiple Propofol-binding Sites in a γ-Aminobutyric Acid Type A Receptor (GABAAR) Identified Using a Photoreactive Propofol Analog

(2014) Selwyn S. Jayakar et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Mutations at Beta N265 in γ-Aminobutyric Acid Type A Receptors Alter Both Binding Affinity and Efficacy of Potent Anesthetics

(2014) Deirdre S. Stewart et al.   PLoS One

Identification of novel positive allosteric modulators and null modulators at the GABAAreceptor α+β− interface

(2013) Zdravko Varagic et al.   BRITISH JOURNAL OF PHARMACOLOGY

Subtype selectivity of α+β− site ligands of GABAAreceptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors

(2013) Zdravko Varagic et al.   BRITISH JOURNAL OF PHARMACOLOGY

Etomidate produces similar allosteric modulation in α1β3δ and α1β3γ2L GABAAreceptors

(2013) H-J Feng et al.   BRITISH JOURNAL OF PHARMACOLOGY

Cysteine Substitutions Define Etomidate Binding and Gating Linkages in the α-M1 Domain of γ-Aminobutyric Acid Type A (GABAA) Receptors

(2013) Deirdre S. Stewart et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Specificity of Intersubunit General Anesthetic-binding Sites in the Transmembrane Domain of the Human α1β3γ2 γ-Aminobutyric Acid Type A (GABAA) Receptor

(2013) David C. Chiara et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Insights into functional pharmacology of α1 GABAA receptors: how much does partial activation at the benzodiazepine site matter?

(2013) Srđan Joksimović et al.   PSYCHOPHARMACOLOGY

Mapping General Anesthetic Binding Site(s) in Human α1β3 γ-Aminobutyric Acid Type A Receptors with [3H]TDBzl-Etomidate, a Photoreactive Etomidate Analogue

(2012) David C. Chiara et al.   BIOCHEMISTRY

Role of α1- and α2-GABAA receptors in mediating the respiratory changes associated with benzodiazepine sedation

(2011) S Masneuf et al.   BRITISH JOURNAL OF PHARMACOLOGY

2′-Methoxy-6-methylflavone: a novel anxiolytic and sedative with subtype selective activating and modulating actions at GABAA receptors

(2011) Nasiara Karim et al.   BRITISH JOURNAL OF PHARMACOLOGY

A novel GABAA receptor pharmacology: drugs interacting with the α+β- interface

(2011) Werner Sieghart et al.   BRITISH JOURNAL OF PHARMACOLOGY

Unraveling the High- and Low-Sensitivity Agonist Responses of Nicotinic Acetylcholine Receptors

(2011) K. Harpsoe et al.   JOURNAL OF NEUROSCIENCE

The GABAA Receptor  + - Interface: A Novel Target for Subtype Selective Drugs

(2011) J. Ramerstorfer et al.   JOURNAL OF NEUROSCIENCE

GABAA Receptor Trafficking-Mediated Plasticity of Inhibitory Synapses

(2011) Bernhard Luscher et al.   NEURON

γ-Amino Butyric Acid Type A Receptor Mutations at β2N265 Alter Etomidate Efficacy While Preserving Basal and Agonist-dependent Activity

(2009) Rooma Desai et al.   ANESTHESIOLOGY

Protein interactions involving the γ2 large cytoplasmic loop of GABAA receptors modulate conductance

(2009) Andrea B. Everitt et al.   FASEB JOURNAL

Estimating the efficiency of benzodiazepines on GABAA receptors comprising γ1 or γ2 subunits

(2008) I Baburin et al.   BRITISH JOURNAL OF PHARMACOLOGY

Histamine Action on Vertebrate GABAAReceptors

(2008) Arunesh Saras et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Tryptophan Mutations at Azi-Etomidate Photo-Incorporation Sites on  1 or  2 Subunits Enhance GABAA Receptor Gating and Reduce Etomidate Modulation

(2008) D. Stewart et al.   MOLECULAR PHARMACOLOGY

GABAA receptor trafficking and its role in the dynamic modulation of neuronal inhibition

(2008) Tija C. Jacob et al.   NATURE REVIEWS NEUROSCIENCE

International Union of Pharmacology. LXX. Subtypes of  -Aminobutyric AcidA Receptors: Classification on the Basis of Subunit Composition, Pharmacology, and Function. Update

(2008) R. W. Olsen et al.   PHARMACOLOGICAL REVIEWS